KR101409277B1 - 펩티드 성장 호르몬 분비촉진제와 유사한 화합물 및 이를 포함하는 제형 - Google Patents
펩티드 성장 호르몬 분비촉진제와 유사한 화합물 및 이를 포함하는 제형 Download PDFInfo
- Publication number
- KR101409277B1 KR101409277B1 KR1020087023543A KR20087023543A KR101409277B1 KR 101409277 B1 KR101409277 B1 KR 101409277B1 KR 1020087023543 A KR1020087023543 A KR 1020087023543A KR 20087023543 A KR20087023543 A KR 20087023543A KR 101409277 B1 KR101409277 B1 KR 101409277B1
- Authority
- KR
- South Korea
- Prior art keywords
- ghrelin
- ghs
- growth hormone
- peptide
- receptor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/60—Growth hormone-releasing factor [GH-RF], i.e. somatoliberin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Zoology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Toxicology (AREA)
- Gastroenterology & Hepatology (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Child & Adolescent Psychology (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Fodder In General (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20060050A CU23558A1 (es) | 2006-02-28 | 2006-02-28 | Compuestos análogos a los secretagogos peptidicos de la hormona de crecimiento |
| CU2006-0050 | 2006-02-28 | ||
| PCT/CU2007/000007 WO2007098716A1 (es) | 2006-02-28 | 2007-02-28 | Compuestos analogos a los secretagogos peptidicos de la hormona de crecimiento y preparaciones que los contienen |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20080110763A KR20080110763A (ko) | 2008-12-19 |
| KR101409277B1 true KR101409277B1 (ko) | 2014-06-24 |
Family
ID=40130780
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020087023543A Expired - Fee Related KR101409277B1 (ko) | 2006-02-28 | 2007-02-28 | 펩티드 성장 호르몬 분비촉진제와 유사한 화합물 및 이를 포함하는 제형 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US8367620B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP1997827B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP5183496B2 (cg-RX-API-DMAC7.html) |
| KR (1) | KR101409277B1 (cg-RX-API-DMAC7.html) |
| CN (1) | CN101432294B (cg-RX-API-DMAC7.html) |
| AR (1) | AR059646A1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2007219569B2 (cg-RX-API-DMAC7.html) |
| BR (1) | BRPI0708366A2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2637593C (cg-RX-API-DMAC7.html) |
| CL (2) | CL2007000528A1 (cg-RX-API-DMAC7.html) |
| CU (1) | CU23558A1 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2441441T3 (cg-RX-API-DMAC7.html) |
| MX (1) | MX2008011142A (cg-RX-API-DMAC7.html) |
| MY (1) | MY184130A (cg-RX-API-DMAC7.html) |
| NO (1) | NO20084118L (cg-RX-API-DMAC7.html) |
| RU (1) | RU2416618C2 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2007098716A1 (cg-RX-API-DMAC7.html) |
| ZA (1) | ZA200807162B (cg-RX-API-DMAC7.html) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4831551B2 (ja) * | 2008-11-06 | 2011-12-07 | 国立大学法人名古屋大学 | 非虚血性心筋障害に対する医薬 |
| CU24473B1 (es) * | 2016-11-01 | 2020-02-04 | Centro De Ingenieria Genetica Y Biotecnologia Biocubafarma | Composición vacunal que comprende un péptido secretagogo de la hormona de crecimiento como adyuvante vacunal |
| RU2734835C1 (ru) * | 2020-02-11 | 2020-10-23 | Федеральное государственное бюджетное учреждение науки Лимнологический институт Сибирского отделение Российской академии наук (ЛИН СО РАН) | Способ повышения жизнестойкости эмбрионов рыб в аквакультуре |
Family Cites Families (92)
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| UA53716C2 (uk) | 1997-06-25 | 2003-02-17 | Пфайзер Продактс Інк. | Тартратна сіль заміщеного дипептиду, спосіб її одержання, проміжні сполуки та спосіб їх одержання, фармацевтична композиція (варіанти), спосіб підвищення рівнів ендогенного гормону росту та спосіб лікування або профілактики захворювань (варіанти) |
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| KR100680085B1 (ko) | 1998-08-20 | 2007-02-28 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 성장호르몬 방출촉진제로서 옥신돌 유도체 |
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| ES2333097T3 (es) | 2000-05-31 | 2010-02-17 | Raqualia Pharma Inc | Uso de secretagogos de la hormona de crecimiento para estimular la motilidad gastrointestinal. |
| CN1232507C (zh) | 2000-06-13 | 2005-12-21 | 曾塔里斯股份公司 | 生长激素促分泌剂 |
| EP1297839A4 (en) | 2000-06-23 | 2005-12-07 | Kaken Pharma Co Ltd | PREVENTIVA OR THERAPEUTIC AGAINST HEART FAILURE |
| ITMI20011445A1 (it) | 2001-07-06 | 2003-01-06 | Europ Geie | Analoghi della cortistantina capaci di legarsi selettivamente ai recettori dei secretagoghi dell'ormone della crescita |
| CU23043A1 (es) | 2001-12-20 | 2005-05-20 | Ct Ingenieria Genetica Biotech | Composicion farmaceutica que contiene factor de crecimiento epidrmico (egf) para la prevencion de la amputacion de pie diabetico. |
| US7476653B2 (en) | 2003-06-18 | 2009-01-13 | Tranzyme Pharma, Inc. | Macrocyclic modulators of the ghrelin receptor |
| WO2005039625A1 (en) | 2003-10-28 | 2005-05-06 | Rheoscience A/S | Growth hormone secretagogue receptor agonists |
| EP1682136A4 (en) | 2003-11-04 | 2009-06-03 | Elixir Pharmaceuticals Inc | THERAPEUTIC COMPOUNDS AND CORRESPONDING USES THEREOF |
| WO2005048916A2 (en) | 2003-11-20 | 2005-06-02 | Biovitrum Ab | Tetrahydrospiro-beta-carboline-1,3 '-pyrrolidine derivatives and their use in ghsr-related disorders |
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| Eur. J. Clin. Invest. 5(2): 165-175(1975. 4.) * |
| Experientia 43(11-12):1211-1212(1987. 12. 1.) * |
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| ZA200807162B (en) | 2009-06-24 |
| CU23558A1 (es) | 2010-07-20 |
| CA2637593A1 (en) | 2007-09-07 |
| JP2009528303A (ja) | 2009-08-06 |
| BRPI0708366A2 (pt) | 2011-05-24 |
| RU2416618C2 (ru) | 2011-04-20 |
| KR20080110763A (ko) | 2008-12-19 |
| WO2007098716A8 (es) | 2008-12-18 |
| CA2637593C (en) | 2015-04-14 |
| US8367620B2 (en) | 2013-02-05 |
| MX2008011142A (es) | 2008-09-08 |
| AU2007219569B2 (en) | 2012-03-15 |
| CN101432294A (zh) | 2009-05-13 |
| WO2007098716A1 (es) | 2007-09-07 |
| CL2016001648A1 (es) | 2017-02-24 |
| NO20084118L (no) | 2008-09-29 |
| ES2441441T3 (es) | 2014-02-04 |
| EP1997827B1 (en) | 2013-10-09 |
| CL2007000528A1 (es) | 2008-01-18 |
| AR059646A1 (es) | 2008-04-16 |
| AU2007219569A1 (en) | 2007-09-07 |
| US20100055118A1 (en) | 2010-03-04 |
| EP1997827A1 (en) | 2008-12-03 |
| CN101432294B (zh) | 2013-09-11 |
| MY184130A (en) | 2021-03-19 |
| JP5183496B2 (ja) | 2013-04-17 |
| RU2008138569A (ru) | 2010-04-10 |
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