BR9610887A - Processo para a preparação de um composto - Google Patents

Processo para a preparação de um composto

Info

Publication number
BR9610887A
BR9610887A BR9610887A BR9610887A BR9610887A BR 9610887 A BR9610887 A BR 9610887A BR 9610887 A BR9610887 A BR 9610887A BR 9610887 A BR9610887 A BR 9610887A BR 9610887 A BR9610887 A BR 9610887A
Authority
BR
Brazil
Prior art keywords
compound
preparation
Prior art date
Application number
BR9610887A
Other languages
English (en)
Inventor
Peter G Houghton
Ioannis Houpis
Audrey Molina
Joseph E Lynch
Ralph P Volante
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9602949.1A external-priority patent/GB9602949D0/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of BR9610887A publication Critical patent/BR9610887A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06017Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
BR9610887A 1995-10-27 1996-10-23 Processo para a preparação de um composto BR9610887A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US589895P 1995-10-27 1995-10-27
GBGB9602949.1A GB9602949D0 (en) 1996-02-13 1996-02-13 Process for the preparation of a growth hormone secretagogue
PCT/US1996/016954 WO1997015573A1 (en) 1995-10-27 1996-10-23 Process for the preparation of a growth hormone secretagogue

Publications (1)

Publication Number Publication Date
BR9610887A true BR9610887A (pt) 1999-07-13

Family

ID=26308687

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9610887A BR9610887A (pt) 1995-10-27 1996-10-23 Processo para a preparação de um composto

Country Status (14)

Country Link
EP (1) EP0863900A1 (pt)
JP (1) JPH11513984A (pt)
KR (1) KR19990067097A (pt)
AR (1) AR004124A1 (pt)
AU (1) AU7468596A (pt)
BR (1) BR9610887A (pt)
CA (1) CA2235511A1 (pt)
CZ (1) CZ128298A3 (pt)
HR (1) HRP960494A2 (pt)
HU (1) HUP9902095A3 (pt)
PL (1) PL326428A1 (pt)
SK (1) SK51198A3 (pt)
WO (1) WO1997015573A1 (pt)
YU (1) YU56596A (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9601724D0 (en) * 1996-01-29 1996-03-27 Merck Sharp & Dohme Therapeutic agents
WO1998018815A1 (en) * 1996-10-25 1998-05-07 Merck & Co., Inc. Convergent process for the preparation of a growth hormone secretagogue
US6329342B1 (en) 1997-08-19 2001-12-11 Eli Lilly And Company Treatment of congestive heart failure with growth hormone secretagogues
US6639076B1 (en) 1998-08-18 2003-10-28 Eli Lilly And Company Growth hormone secretagogues
US6828331B1 (en) 1999-02-19 2004-12-07 Eli Lilly And Company Growth hormone secretagogues
EP1159964B1 (en) 2000-05-31 2009-10-28 Pfizer Products Inc. Use of growth hormone secretagogues for stimulating gastrointestinal motility
US7125840B2 (en) 2001-10-09 2006-10-24 Eli Lilly And Company Substituted dipeptides as growth hormone secretagogues
ATE332307T1 (de) 2002-04-09 2006-07-15 Lilly Co Eli Wachstumhormonsekretionsförderer
US7476653B2 (en) 2003-06-18 2009-01-13 Tranzyme Pharma, Inc. Macrocyclic modulators of the ghrelin receptor
CU23558A1 (es) 2006-02-28 2010-07-20 Ct Ingenieria Genetica Biotech Compuestos análogos a los secretagogos peptidicos de la hormona de crecimiento
BRPI0807046A2 (pt) 2007-02-09 2015-05-26 Tranzyme Pharma Inc Composto, composição farmacêutica, métodos de tratar um distúrbio, uma doença cardiovascular e um paciente que sofre de motilidade gastrointestinal reduzida ou disfuncional e, kit.
US9119832B2 (en) 2014-02-05 2015-09-01 The Regents Of The University Of California Methods of treating mild brain injury
US20170121385A1 (en) 2015-10-28 2017-05-04 Oxeia Biopharmaceuticals, Inc. Methods of treating neurodegenerative conditions

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RO115804B1 (ro) * 1992-12-11 2000-06-30 Merck & Co Inc Derivati de spiropiperidine, procedee de preparare si compozitii farmaceutice ale acestora

Also Published As

Publication number Publication date
EP0863900A1 (en) 1998-09-16
MX9803316A (es) 1998-09-30
AR004124A1 (es) 1998-09-30
HRP960494A2 (en) 1998-04-30
PL326428A1 (en) 1998-09-14
CA2235511A1 (en) 1997-05-01
WO1997015573A1 (en) 1997-05-01
CZ128298A3 (cs) 1998-07-15
SK51198A3 (en) 1998-11-04
HUP9902095A2 (hu) 1999-10-28
YU56596A (sh) 1999-09-27
KR19990067097A (ko) 1999-08-16
JPH11513984A (ja) 1999-11-30
AU7468596A (en) 1997-05-15
HUP9902095A3 (en) 2001-05-28

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law