PT877738E - Processo para a preparacao de derivados de fenil-imidazolidina - Google Patents

Processo para a preparacao de derivados de fenil-imidazolidina

Info

Publication number
PT877738E
PT877738E PT96938306T PT96938306T PT877738E PT 877738 E PT877738 E PT 877738E PT 96938306 T PT96938306 T PT 96938306T PT 96938306 T PT96938306 T PT 96938306T PT 877738 E PT877738 E PT 877738E
Authority
PT
Portugal
Prior art keywords
phenyl
preparation
imidazolidine derivatives
imidazolidine
derivatives
Prior art date
Application number
PT96938306T
Other languages
English (en)
Inventor
Philippe Mackiewicz
Raphael Bouchet
Daniel Guilmard
Michel Delthil
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of PT877738E publication Critical patent/PT877738E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72Two oxygen atoms, e.g. hydantoin
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
PT96938306T 1995-11-16 1996-11-14 Processo para a preparacao de derivados de fenil-imidazolidina PT877738E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9513589A FR2741346B1 (fr) 1995-11-16 1995-11-16 Nouveau procede de preparation de derives phenylimidazolidine

Publications (1)

Publication Number Publication Date
PT877738E true PT877738E (pt) 2003-09-30

Family

ID=9484624

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96938306T PT877738E (pt) 1995-11-16 1996-11-14 Processo para a preparacao de derivados de fenil-imidazolidina

Country Status (29)

Country Link
US (1) US6107488A (pt)
EP (1) EP0877738B1 (pt)
JP (1) JP2000500150A (pt)
KR (1) KR100466991B1 (pt)
CN (1) CN1131219C (pt)
AR (1) AR004965A1 (pt)
AT (1) ATE240300T1 (pt)
AU (1) AU718832B2 (pt)
BR (1) BR9611573A (pt)
CA (1) CA2235335A1 (pt)
CU (1) CU22890A3 (pt)
CZ (1) CZ144498A3 (pt)
DE (1) DE69628203T2 (pt)
DK (1) DK0877738T3 (pt)
EA (1) EA002658B1 (pt)
ES (1) ES2193271T3 (pt)
FR (1) FR2741346B1 (pt)
HU (1) HUP9904034A3 (pt)
IL (1) IL124382A0 (pt)
MX (1) MX9803730A (pt)
NO (1) NO316514B1 (pt)
PL (1) PL189697B1 (pt)
PT (1) PT877738E (pt)
SI (1) SI0877738T1 (pt)
TR (1) TR199800865T2 (pt)
TW (1) TW404942B (pt)
UA (1) UA67720C2 (pt)
WO (1) WO1997018197A1 (pt)
ZA (1) ZA969442B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2299266A1 (en) * 2003-12-19 2011-03-23 The Regents of the University of California Methods and materials for assessing prostate cancer therapies
NZ550102A (en) * 2004-02-24 2010-10-29 Univ California Methods and materials for assessing prostate cancer therapies and compounds (thiohydantoine derivatives)
US7709517B2 (en) * 2005-05-13 2010-05-04 The Regents Of The University Of California Diarylhydantoin compounds
LT3100727T (lt) 2006-03-27 2018-12-10 The Regents Of The University Of California Androgeno receptoriaus moduliatorius, skirtas prostatos vėžio ir su androgeno receptoriumi susijusių ligų gydymui
WO2007127010A2 (en) 2006-03-29 2007-11-08 The Regents Of The University Of California Diarylthiohydantoin compounds
EP2220050A2 (en) 2007-10-26 2010-08-25 The Regents Of The University Of California Diarylhydantoin compounds as androgen receptor modulators
US20120238533A1 (en) 2009-09-11 2012-09-20 Bayer Pharma Aktiengesellschaft (Heteroarylmethyl) Thiohydantoins as anticancer drugs
AU2010265775B2 (en) 2009-09-15 2013-09-12 Mylan Group Copolymers, polymeric particles comprising said copolymers and copolymeric binders for radiation-sensitive coating compositions for negative-working radiation-sensitive lithographic printing plates
EA201792046A1 (ru) 2010-02-16 2018-05-31 Арагон Фармасьютикалс, Инк. Модуляторы рецептора андрогенов и их применение
UA106533C2 (uk) 2010-09-14 2014-09-10 Майлен Груп Співполімери для чутливих у близькій інфрачервоній області випромінювання композицій для покриття позитивних термічних літографічних друкарських форм
NZ744456A (en) 2012-09-26 2019-09-27 Aragon Pharmaceuticals Inc Anti-androgens for the treatment of non-metastatic castrate-resistant prostate cancer
JOP20200097A1 (ar) 2013-01-15 2017-06-16 Aragon Pharmaceuticals Inc معدل مستقبل أندروجين واستخداماته
TWI726969B (zh) 2016-01-11 2021-05-11 比利時商健生藥品公司 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物
JOP20200076A1 (ar) 2017-10-16 2020-04-30 Aragon Pharmaceuticals Inc مضادات أندروجين لعلاج سرطان البروستاتا غير النقيلي المقاوم للاستئصال
CN108218784A (zh) * 2018-01-16 2018-06-29 吴江信凯医药科技有限公司 一种尼鲁米特的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4916937B1 (pt) * 1970-01-21 1974-04-25
JPS5136332B1 (pt) * 1970-12-09 1976-10-07
CH544491A (de) * 1971-03-16 1973-11-30 Ciba Geigy Ag Herbizides Mittel
MC1220A1 (fr) * 1977-10-28 1979-07-20 Hoffmann La Roche Nouveaux derives d'imidazolidine
JPS57197268A (en) * 1981-05-29 1982-12-03 Sumitomo Chem Co Ltd Substituted phenylhydantoin derivative, its preparation, and herbicide containing the same as active ingredient
JPS62298562A (ja) * 1986-06-17 1987-12-25 Nippon Kayaku Co Ltd ブロモアニリン類の製造法
FR2656302B1 (fr) * 1989-12-22 1992-05-07 Roussel Uclaf Nouveau procede de preparation de l'anandron et derives de l'anandron.
US5411981A (en) * 1991-01-09 1995-05-02 Roussel Uclaf Phenylimidazolidines having antiandrogenic activity
FR2694290B1 (fr) * 1992-07-08 1994-09-02 Roussel Uclaf Nouvelles phénylimidazolidines éventuellement substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.

Also Published As

Publication number Publication date
CN1131219C (zh) 2003-12-17
NO316514B1 (no) 2004-02-02
DE69628203D1 (de) 2003-06-18
NO982237L (no) 1998-07-10
DE69628203T2 (de) 2004-02-05
EP0877738A1 (fr) 1998-11-18
UA67720C2 (en) 2004-07-15
IL124382A0 (en) 1998-12-06
WO1997018197A1 (fr) 1997-05-22
JP2000500150A (ja) 2000-01-11
NO982237D0 (no) 1998-05-15
TR199800865T2 (xx) 1998-08-21
KR100466991B1 (ko) 2005-04-06
MX9803730A (es) 1998-11-30
FR2741346B1 (fr) 1997-12-19
US6107488A (en) 2000-08-22
ATE240300T1 (de) 2003-05-15
PL326491A1 (en) 1998-09-28
HUP9904034A3 (en) 2001-08-28
CU22890A3 (es) 2004-01-23
CA2235335A1 (fr) 1997-05-22
AR004965A1 (es) 1999-04-07
AU718832B2 (en) 2000-04-20
EA002658B1 (ru) 2002-08-29
CZ144498A3 (cs) 1998-09-16
SI0877738T1 (en) 2003-10-31
TW404942B (en) 2000-09-11
PL189697B1 (pl) 2005-09-30
DK0877738T3 (da) 2003-09-08
BR9611573A (pt) 1999-05-11
HUP9904034A2 (hu) 2000-05-28
AU7577396A (en) 1997-06-05
KR19990067639A (ko) 1999-08-25
ES2193271T3 (es) 2003-11-01
ZA969442B (en) 1997-11-11
FR2741346A1 (fr) 1997-05-23
CN1207732A (zh) 1999-02-10
EP0877738B1 (fr) 2003-05-14
EA199800378A1 (ru) 1998-10-29

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