BR9608471A - Processo para a preparação de um composto - Google Patents

Processo para a preparação de um composto

Info

Publication number
BR9608471A
BR9608471A BR9608471A BR9608471A BR9608471A BR 9608471 A BR9608471 A BR 9608471A BR 9608471 A BR9608471 A BR 9608471A BR 9608471 A BR9608471 A BR 9608471A BR 9608471 A BR9608471 A BR 9608471A
Authority
BR
Brazil
Prior art keywords
compound
preparation
Prior art date
Application number
BR9608471A
Other languages
English (en)
Inventor
Mogens Engelstoft
Bjorn Bentzen
Soren Lehman
John Bondo Hansen
Svend Treppendahl
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of BR9608471A publication Critical patent/BR9608471A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
BR9608471A 1995-05-17 1996-04-25 Processo para a preparação de um composto BR9608471A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK56395 1995-05-17
PCT/DK1996/000185 WO1996036636A1 (en) 1995-05-17 1996-04-25 Process for preparing 4-aryl-piperidine derivatives

Publications (1)

Publication Number Publication Date
BR9608471A true BR9608471A (pt) 1998-12-29

Family

ID=8094959

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9608471A BR9608471A (pt) 1995-05-17 1996-04-25 Processo para a preparação de um composto

Country Status (11)

Country Link
EP (1) EP0828735A1 (pt)
JP (1) JPH11505229A (pt)
CN (1) CN1068597C (pt)
AU (1) AU721257B2 (pt)
BR (1) BR9608471A (pt)
CA (1) CA2220963A1 (pt)
HU (1) HUP9900318A3 (pt)
IL (1) IL118294A0 (pt)
NZ (1) NZ307479A (pt)
WO (1) WO1996036636A1 (pt)
ZA (1) ZA963951B (pt)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9526645D0 (en) * 1995-12-28 1996-02-28 Chiroscience Ltd Stereoselective synthesis
ES2117557B1 (es) * 1996-02-29 1999-07-01 Ferrer Int Nuevo procedimiento de obtencion de (-)-trans -n-p-fluorobenzoilmetil-4-(p-fluorofenil)-3- ((3,4-(metilendioxi)fenoxi ) metil)-piperidina.
EP0812827B1 (en) 1996-06-13 2009-09-02 Sumitomo Chemical Company, Limited Piperidine derivative as intermediates for the preparation of paroxetine and process for their preparation
HU221921B1 (hu) * 1996-07-08 2003-02-28 Richter Gedeon Vegyészeti Gyár Rt. N-benzil-piperidin- és tetrahidropiridinszármazékok és eljárás azok előállítására
GB9623359D0 (en) * 1996-11-09 1997-01-08 Smithkline Beecham Plc Novel process
GB9700690D0 (en) 1997-01-15 1997-03-05 Smithkline Beecham Plc Novel process
GB9710004D0 (en) * 1997-05-17 1997-07-09 Knoll Ag Chemical process
JP2002514222A (ja) 1997-05-29 2002-05-14 スミスクライン・ビーチャム・コーポレイション 新規方法
WO1998056787A1 (en) * 1997-06-10 1998-12-17 Synthon B.V. 4-Phenylpiperidine compounds
CH689805A8 (fr) * 1998-07-02 2000-02-29 Smithkline Beecham Plc Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
GB9826175D0 (en) * 1998-11-28 1999-01-20 Smithkline Beecham Plc Novel process
GB9828767D0 (en) * 1998-12-29 1999-02-17 Smithkline Beecham Plc Novel process
IT1308629B1 (it) * 1999-02-23 2002-01-09 Recordati Chem Pharm Processo per la produzione di paroxetina.
IT1313702B1 (it) * 1999-08-02 2002-09-09 Chemi Spa Processo per la preparazione di derivati 3-sostituiti di 4-fenil-piperidine.
WO2001032178A1 (en) * 1999-10-29 2001-05-10 Novo Nordisk A/S Use of 3,4-substituted piperidines
GB9930577D0 (en) * 1999-12-23 2000-02-16 Smithkline Beecham Plc Novel process
EP1280775A1 (en) 2000-05-12 2003-02-05 Synthon B.V. TOSYLATE SALTS OF 4-(p-FLUOROPHENYL)-PIPERIDINE-3-CARBINOLS
WO2002006275A1 (en) * 2000-07-17 2002-01-24 Smithkline Beecham P.L.C. Novel processes for the preparation of 4-phenylpiperidine derivatives
GB0021147D0 (en) * 2000-08-30 2000-10-11 Knoll Ag Chemical process
GB0021145D0 (en) * 2000-08-30 2000-10-11 Knoll Ag Chemical process
AU2001211337A1 (en) * 2000-10-06 2002-04-15 Smithkline Beecham Plc Process for the preparation of aryl-piperidine carbinols and intermediates thereof
NZ526874A (en) * 2001-01-04 2005-07-29 Ferrer Internacional S Process for preparing (+/-) trans-4-p-fluorophenyl-3-hydroxymethyl-1-methylpiperidine
WO2015071831A1 (en) * 2013-11-18 2015-05-21 Piramal Enterprises Limited An improved process for minimising the formation of dehalogenated byproducts

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1422263A (en) * 1973-01-30 1976-01-21 Ferrosan As 4-phenyl-piperidine compounds
US4593036A (en) * 1984-02-07 1986-06-03 A/S Ferrosan (-)-Trans-4-(4-fluorophenyl)-3-[(4-methoxyphenoxy)methyl]-1-methylpiperidine useful as 5-HT potentiator
IE66332B1 (en) * 1986-11-03 1995-12-27 Novo Nordisk As Piperidine compounds and their preparation and use
DK715988D0 (da) * 1988-12-22 1988-12-22 Ferrosan As Etherifikation og dealkylering af piperidin-derivater samt intermediater

Also Published As

Publication number Publication date
AU721257B2 (en) 2000-06-29
EP0828735A1 (en) 1998-03-18
WO1996036636A1 (en) 1996-11-21
JPH11505229A (ja) 1999-05-18
HUP9900318A3 (en) 2001-09-28
CN1068597C (zh) 2001-07-18
IL118294A0 (en) 1996-09-12
CN1184476A (zh) 1998-06-10
HUP9900318A2 (hu) 1999-09-28
AU5684596A (en) 1996-11-29
NZ307479A (en) 1999-08-30
ZA963951B (en) 1997-01-21
CA2220963A1 (en) 1996-11-21

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Legal Events

Date Code Title Description
EG Technical examination (opinion): publication of technical examination (opinion)
FC Decision: refusal