ATE240300T1 - Verfahren zur herstellung von phenylimidazolin- derivaten - Google Patents

Verfahren zur herstellung von phenylimidazolin- derivaten

Info

Publication number
ATE240300T1
ATE240300T1 AT96938306T AT96938306T ATE240300T1 AT E240300 T1 ATE240300 T1 AT E240300T1 AT 96938306 T AT96938306 T AT 96938306T AT 96938306 T AT96938306 T AT 96938306T AT E240300 T1 ATE240300 T1 AT E240300T1
Authority
AT
Austria
Prior art keywords
phenylimidazoline
derivatives
producing
producing phenylimidazoline
phenylimidazoline derivatives
Prior art date
Application number
AT96938306T
Other languages
English (en)
Inventor
Rapha L Bouchet
Michel Delthil
Daniel Guilmard
Philippe Mackiewicz
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of ATE240300T1 publication Critical patent/ATE240300T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
AT96938306T 1995-11-16 1996-11-14 Verfahren zur herstellung von phenylimidazolin- derivaten ATE240300T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9513589A FR2741346B1 (fr) 1995-11-16 1995-11-16 Nouveau procede de preparation de derives phenylimidazolidine
PCT/FR1996/001794 WO1997018197A1 (fr) 1995-11-16 1996-11-14 Nouveau procede de preparation de derives phenylimidazolidine

Publications (1)

Publication Number Publication Date
ATE240300T1 true ATE240300T1 (de) 2003-05-15

Family

ID=9484624

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96938306T ATE240300T1 (de) 1995-11-16 1996-11-14 Verfahren zur herstellung von phenylimidazolin- derivaten

Country Status (29)

Country Link
US (1) US6107488A (de)
EP (1) EP0877738B1 (de)
JP (1) JP2000500150A (de)
KR (1) KR100466991B1 (de)
CN (1) CN1131219C (de)
AR (1) AR004965A1 (de)
AT (1) ATE240300T1 (de)
AU (1) AU718832B2 (de)
BR (1) BR9611573A (de)
CA (1) CA2235335A1 (de)
CU (1) CU22890A3 (de)
CZ (1) CZ144498A3 (de)
DE (1) DE69628203T2 (de)
DK (1) DK0877738T3 (de)
EA (1) EA002658B1 (de)
ES (1) ES2193271T3 (de)
FR (1) FR2741346B1 (de)
HU (1) HUP9904034A3 (de)
IL (1) IL124382A0 (de)
MX (1) MX9803730A (de)
NO (1) NO316514B1 (de)
PL (1) PL189697B1 (de)
PT (1) PT877738E (de)
SI (1) SI0877738T1 (de)
TR (1) TR199800865T2 (de)
TW (1) TW404942B (de)
UA (1) UA67720C2 (de)
WO (1) WO1997018197A1 (de)
ZA (1) ZA969442B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE602004031881D1 (de) * 2003-12-19 2011-04-28 Univ California Verfahren und materialien zur beurteilung von prostatakrebstherapien
US7718684B2 (en) * 2004-02-24 2010-05-18 The Regents Of The University Of California Methods and materials for assessing prostate cancer therapies and compounds
US7709517B2 (en) * 2005-05-13 2010-05-04 The Regents Of The University Of California Diarylhydantoin compounds
EP2656842B1 (de) 2006-03-27 2016-08-10 The Regents of The University of California Androgenrezeptor-modulator zur behandlung von prostatakrebs und androgenrezeptor-assoziierte erkrankungen
WO2007127010A2 (en) * 2006-03-29 2007-11-08 The Regents Of The University Of California Diarylthiohydantoin compounds
CA2966280A1 (en) 2007-10-26 2009-04-30 The Regents Of The University Of California Diarylhydantoin compounds
US20120238533A1 (en) 2009-09-11 2012-09-20 Bayer Pharma Aktiengesellschaft (Heteroarylmethyl) Thiohydantoins as anticancer drugs
KR101390985B1 (ko) 2009-09-15 2014-05-02 밀란 그룹 코폴리머, 상기 코폴리머를 포함하는 폴리머성 입자 및 네거티브형 감방사선성 평판 인쇄판용 감방사선성 코팅 조성물의 코폴리머성 결합제
HUE037389T2 (hu) 2010-02-16 2018-08-28 Aragon Pharmaceuticals Inc Androgén receptor modulátorok és alkalmazásaik
WO2011006265A2 (en) 2010-09-14 2011-01-20 Mylan Group Copolymers for near-infrared radiation-sensitive coating compositions for positive-working thermal lithographic printing plates
ES2836424T3 (es) 2012-09-26 2021-06-25 Aragon Pharmaceuticals Inc Antiandrógenos para tratar el cáncer de próstata no metastásico y resistente a la castración
CA3105575A1 (en) 2013-01-15 2014-07-24 Aragon Pharmaceuticals, Inc. Androgen receptor modulator and uses thereof
TWI726969B (zh) 2016-01-11 2021-05-11 比利時商健生藥品公司 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物
UA129105C2 (uk) 2017-10-16 2025-01-15 Арагон Фармасьютикалз, Інк. Антиандрогени для лікування неметастатичного резистентного до кастрації раку передміхурової залози
CN108218784A (zh) * 2018-01-16 2018-06-29 吴江信凯医药科技有限公司 一种尼鲁米特的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4916937B1 (de) * 1970-01-21 1974-04-25
JPS5136332B1 (de) * 1970-12-09 1976-10-07
CH544491A (de) * 1971-03-16 1973-11-30 Ciba Geigy Ag Herbizides Mittel
MC1220A1 (fr) * 1977-10-28 1979-07-20 Hoffmann La Roche Nouveaux derives d'imidazolidine
JPS57197268A (en) * 1981-05-29 1982-12-03 Sumitomo Chem Co Ltd Substituted phenylhydantoin derivative, its preparation, and herbicide containing the same as active ingredient
JPS62298562A (ja) * 1986-06-17 1987-12-25 Nippon Kayaku Co Ltd ブロモアニリン類の製造法
FR2656302B1 (fr) * 1989-12-22 1992-05-07 Roussel Uclaf Nouveau procede de preparation de l'anandron et derives de l'anandron.
US5411981A (en) * 1991-01-09 1995-05-02 Roussel Uclaf Phenylimidazolidines having antiandrogenic activity
FR2694290B1 (fr) * 1992-07-08 1994-09-02 Roussel Uclaf Nouvelles phénylimidazolidines éventuellement substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.

Also Published As

Publication number Publication date
EP0877738B1 (de) 2003-05-14
EA199800378A1 (ru) 1998-10-29
NO982237D0 (no) 1998-05-15
CU22890A3 (es) 2004-01-23
PL189697B1 (pl) 2005-09-30
KR19990067639A (ko) 1999-08-25
DK0877738T3 (da) 2003-09-08
JP2000500150A (ja) 2000-01-11
HUP9904034A3 (en) 2001-08-28
AR004965A1 (es) 1999-04-07
SI0877738T1 (en) 2003-10-31
ES2193271T3 (es) 2003-11-01
PL326491A1 (en) 1998-09-28
NO982237L (no) 1998-07-10
PT877738E (pt) 2003-09-30
FR2741346A1 (fr) 1997-05-23
BR9611573A (pt) 1999-05-11
EA002658B1 (ru) 2002-08-29
CN1207732A (zh) 1999-02-10
FR2741346B1 (fr) 1997-12-19
DE69628203D1 (de) 2003-06-18
CN1131219C (zh) 2003-12-17
ZA969442B (en) 1997-11-11
CZ144498A3 (cs) 1998-09-16
CA2235335A1 (fr) 1997-05-22
UA67720C2 (en) 2004-07-15
MX9803730A (es) 1998-11-30
TW404942B (en) 2000-09-11
NO316514B1 (no) 2004-02-02
IL124382A0 (en) 1998-12-06
HUP9904034A2 (hu) 2000-05-28
KR100466991B1 (ko) 2005-04-06
EP0877738A1 (de) 1998-11-18
AU718832B2 (en) 2000-04-20
TR199800865T2 (xx) 1998-08-21
WO1997018197A1 (fr) 1997-05-22
DE69628203T2 (de) 2004-02-05
AU7577396A (en) 1997-06-05
US6107488A (en) 2000-08-22

Similar Documents

Publication Publication Date Title
ATE243211T1 (de) Verfahren zur herstellung von dihalogenazolopyrimidinen
DE69525373D1 (de) Verfahren zur herstellung von alumosilikatderivaten
DE59603155D1 (de) Verfahren zur herstellung von hydrotalciten
DE59604922D1 (de) Verfahren zur herstellung von polyalkoholen
DE69602331D1 (de) Verfahren zur herstellung von polyolefin
DE69604277D1 (de) Verfahren zur herstellung von nootkaton
DE69814862D1 (de) Verfahren zur herstellung von pyridinderivaten
DE69519379D1 (de) Verfahren zur herstellung von trifluorethylene
ATE187727T1 (de) Verfahren zur herstellung von imidazo- benzodiazepin-derivaten
ATE267812T1 (de) Verfahren zur herstellung von n-substituierten 3- hydroxypyrazolen
ATE229021T1 (de) Verfahren zur herstellung von imidazochinazolinon-derivaten
DE59601604D1 (de) Verfahren zur herstellung von n-aryl- und n-hetarylhydroxylaminen
ATE240300T1 (de) Verfahren zur herstellung von phenylimidazolin- derivaten
ATE303134T1 (de) Verfahren zur herstellung von flavano-lignan- zubereitungen
ATE309230T1 (de) Verfahren zur herstellung von 2- chlorthiazolderivaten
DE69813869D1 (de) Verfahren zur herstellung von thiazolidindion-derivaten
DE59601895D1 (de) Verfahren zur herstellung von butyrolactonen
ATE203046T1 (de) Verfahren zur herstellung von pigmenten
ATE181554T1 (de) Verfahren zur herstellung von n- phosphonomethylglyzin
ATE207900T1 (de) Verfahren zur herstellung von ropivacainehydrochlorid-monohydrat
DE69616322D1 (de) Verfahren zur herstellung von 3-isochromanonen
DE69808068D1 (de) Verfahren zur herstellung von indolderivaten
DE69601993D1 (de) Verfahren zur herstellung von doxorubicin
ATE219056T1 (de) Verfahren zur herstellung von alpha- bromolactamderivaten
DE69615836D1 (de) Verfahren zur herstellung von boroxyd

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification

Ref document number: 0877738

Country of ref document: EP

REN Ceased due to non-payment of the annual fee