KR100741257B1 - Ｎｍｄａ, 5ｈｔ₃ 및 신경원 세포의 니코틴작용성 수용체길항물질로서 아미노시클로헥산의 아자비시클로,아자트리시클로 및 아자스피로시클로 유도체 - Google Patents

Ｎｍｄａ, 5ｈｔ₃ 및 신경원 세포의 니코틴작용성 수용체길항물질로서 아미노시클로헥산의 아자비시클로,아자트리시클로 및 아자스피로시클로 유도체 Download PDF

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KR100741257B1
KR100741257B1 KR1020047011982A KR20047011982A KR100741257B1 KR 100741257 B1 KR100741257 B1 KR 100741257B1 KR 1020047011982 A KR1020047011982 A KR 1020047011982A KR 20047011982 A KR20047011982 A KR 20047011982A KR 100741257 B1 KR100741257 B1 KR 100741257B1
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disease
disorders
azabicyclo
drug
hydrochlorides
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KR20040091005A (ko
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파르존스크리스토퍼그라암라파엘
헨리히마르쿠스
단시츠보이치에흐
칼빈쉬이바르스
카우스발레르얀스
지르겐존스아이가르스
골트마르쿠스
바네제브스막심스
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메르츠 파마 게엠베하 운트 코. 카가아
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KR1020047011982A 2002-03-21 2003-03-21 Ｎｍｄａ, 5ｈｔ₃ 및 신경원 세포의 니코틴작용성 수용체길항물질로서 아미노시클로헥산의 아자비시클로,아자트리시클로 및 아자스피로시클로 유도체 Expired - Fee Related KR100741257B1 (ko)

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Application Number Priority Date Filing Date Title
US36638602P 2002-03-21 2002-03-21
US?60/366,386? 2002-03-21
PCT/GB2003/001236 WO2003080046A1 (en) 2002-03-21 2003-03-21 Azabicyclic, azatricyclic and azaspirocyclic derivatives of aminocyclohexane nmda, 5ht3, and neuronal nicotinic receptor antagoni sts

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KR20040091005A KR20040091005A (ko) 2004-10-27
KR100741257B1 true KR100741257B1 (ko) 2007-07-19

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US (4) US7022729B2 (https=)
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CN (1) CN1638762A (https=)
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ES2483126T3 (es) 2004-06-17 2014-08-05 Merz Pharma Gmbh & Co. Kgaa Formulaciones de formas de dosificación de neramexano
US20060205822A1 (en) * 2004-12-22 2006-09-14 Forest Laboratories, Inc. 1-Aminocyclohexane derivatives for the treatment of multiple sclerosis, emotional lability and pseudobulbar affect
EP2111858A1 (en) 2008-04-25 2009-10-28 EPFL Ecole Polytechnique Fédérale de Lausanne Novel treatment for alzheimer's disease
US20090275597A1 (en) * 2008-05-02 2009-11-05 Forest Laboratories Holdings Limited Methods of treating cns disorders
PE20130775A1 (es) * 2010-05-27 2013-07-21 Targacept Inc Antagonistas no competitivos de receptores nicotinicos
RU2014122338A (ru) * 2011-11-03 2015-12-10 Таргасепт, Инк. Неконкурентные модуляторы никотиновых рецепторов
JP6095122B2 (ja) * 2012-01-25 2017-03-15 国立大学法人東北大学 脳機能改善剤
PE20151727A1 (es) 2013-03-14 2015-12-17 Boehringer Ingelheim Int Acido 2-aza-biciclo[2.2.1]heptano-3-carboxilico (bencil-ciano-metil)-amidas sustituidas inhibidores de catepsina c
KR102510588B1 (ko) 2014-09-12 2023-03-17 베링거 인겔하임 인터내셔날 게엠베하 카텝신 c의 스피로사이클릭 억제제

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JPH0578560A (ja) * 1991-09-18 1993-03-30 Toyobo Co Ltd 難燃性ポリエステル樹脂組成物

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