CN1638762A - 作为nmda、5ht3和神经元烟碱性受体拮抗剂的氨基环己烷的氮杂二环、氮杂三环和氮杂螺环衍生物 - Google Patents

作为nmda、5ht3和神经元烟碱性受体拮抗剂的氨基环己烷的氮杂二环、氮杂三环和氮杂螺环衍生物 Download PDF

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Publication number
CN1638762A
CN1638762A CNA038044900A CN03804490A CN1638762A CN 1638762 A CN1638762 A CN 1638762A CN A038044900 A CNA038044900 A CN A038044900A CN 03804490 A CN03804490 A CN 03804490A CN 1638762 A CN1638762 A CN 1638762A
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Prior art keywords
disease
hydrochlorate
azabicyclic
octane
nmda
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Pending
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CNA038044900A
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English (en)
Chinese (zh)
Inventor
C·G·R·帕森斯
M·翰里驰
W·达尼兹
I·卡尔温施
V·考斯
A·吉尔根森斯
M·勾德
M·瓦尼耶弗斯
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Merz Pharma GmbH and Co KGaA
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Merz Pharma GmbH and Co KGaA
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Publication of CN1638762A publication Critical patent/CN1638762A/zh
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  • Immunology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CNA038044900A 2002-03-21 2003-03-21 作为nmda、5ht3和神经元烟碱性受体拮抗剂的氨基环己烷的氮杂二环、氮杂三环和氮杂螺环衍生物 Pending CN1638762A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36638602P 2002-03-21 2002-03-21
US60/366,386 2002-03-21

Publications (1)

Publication Number Publication Date
CN1638762A true CN1638762A (zh) 2005-07-13

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CNA038044900A Pending CN1638762A (zh) 2002-03-21 2003-03-21 作为nmda、5ht3和神经元烟碱性受体拮抗剂的氨基环己烷的氮杂二环、氮杂三环和氮杂螺环衍生物

Country Status (19)

Country Link
US (4) US7022729B2 (https=)
EP (1) EP1485086A1 (https=)
JP (1) JP4262606B2 (https=)
KR (1) KR100741257B1 (https=)
CN (1) CN1638762A (https=)
AR (1) AR039008A1 (https=)
AU (1) AU2003216855B2 (https=)
CA (1) CA2474637A1 (https=)
CO (1) CO5611104A2 (https=)
EA (1) EA007098B1 (https=)
GE (1) GEP20063954B (https=)
IL (1) IL164041A0 (https=)
MX (1) MXPA04007755A (https=)
NO (1) NO20044481L (https=)
PL (1) PL372701A1 (https=)
TW (1) TW200306189A (https=)
UA (1) UA77778C2 (https=)
WO (1) WO2003080046A1 (https=)
ZA (1) ZA200406940B (https=)

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ES2483126T3 (es) 2004-06-17 2014-08-05 Merz Pharma Gmbh & Co. Kgaa Formulaciones de formas de dosificación de neramexano
US20060205822A1 (en) * 2004-12-22 2006-09-14 Forest Laboratories, Inc. 1-Aminocyclohexane derivatives for the treatment of multiple sclerosis, emotional lability and pseudobulbar affect
EP2111858A1 (en) 2008-04-25 2009-10-28 EPFL Ecole Polytechnique Fédérale de Lausanne Novel treatment for alzheimer's disease
US20090275597A1 (en) * 2008-05-02 2009-11-05 Forest Laboratories Holdings Limited Methods of treating cns disorders
PE20130775A1 (es) * 2010-05-27 2013-07-21 Targacept Inc Antagonistas no competitivos de receptores nicotinicos
RU2014122338A (ru) * 2011-11-03 2015-12-10 Таргасепт, Инк. Неконкурентные модуляторы никотиновых рецепторов
JP6095122B2 (ja) * 2012-01-25 2017-03-15 国立大学法人東北大学 脳機能改善剤
PE20151727A1 (es) 2013-03-14 2015-12-17 Boehringer Ingelheim Int Acido 2-aza-biciclo[2.2.1]heptano-3-carboxilico (bencil-ciano-metil)-amidas sustituidas inhibidores de catepsina c
KR102510588B1 (ko) 2014-09-12 2023-03-17 베링거 인겔하임 인터내셔날 게엠베하 카텝신 c의 스피로사이클릭 억제제

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