KR100196969B1 - 축합 디아제피논, 이의 제조방법 및 이를 함유하는 약제학적 조성물 - Google Patents

축합 디아제피논, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Download PDF

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Publication number
KR100196969B1
KR100196969B1 KR1019920006036A KR920006036A KR100196969B1 KR 100196969 B1 KR100196969 B1 KR 100196969B1 KR 1019920006036 A KR1019920006036 A KR 1019920006036A KR 920006036 A KR920006036 A KR 920006036A KR 100196969 B1 KR100196969 B1 KR 100196969B1
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KR
South Korea
Prior art keywords
dihydro
acetyl
piperidinyl
pyrido
ethylamino
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Expired - Fee Related
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KR1019920006036A
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English (en)
Korean (ko)
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KR920019792A (ko
Inventor
에베르라인 볼프강
밈 게르하르트
엔겔 볼프하르트
루돌프 클라우스
두즈 헨리
찌글러 하랄트
엔쩨로트 미카엘
Original Assignee
라이펜 메르. 밀네스
닥터.칼토매게엠베하
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Publication of KR920019792A publication Critical patent/KR920019792A/ko
Application granted granted Critical
Publication of KR100196969B1 publication Critical patent/KR100196969B1/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
KR1019920006036A 1991-04-12 1992-04-11 축합 디아제피논, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Expired - Fee Related KR100196969B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DEP4112014.0 1991-04-12
DE4112014A DE4112014A1 (de) 1991-04-12 1991-04-12 Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende mittel zur behandlung von erkrankungen des zentralnervensystems und zur foerderung der cerebralen durchblutung

Publications (2)

Publication Number Publication Date
KR920019792A KR920019792A (ko) 1992-11-20
KR100196969B1 true KR100196969B1 (ko) 1999-06-15

Family

ID=6429483

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019920006036A Expired - Fee Related KR100196969B1 (ko) 1991-04-12 1992-04-11 축합 디아제피논, 이의 제조방법 및 이를 함유하는 약제학적 조성물

Country Status (28)

Country Link
US (1) US5641772A (enExample)
EP (1) EP0508370B1 (enExample)
JP (1) JPH0597845A (enExample)
KR (1) KR100196969B1 (enExample)
AT (1) ATE140004T1 (enExample)
AU (1) AU653802B2 (enExample)
CA (1) CA2065800A1 (enExample)
CZ (1) CZ283399B6 (enExample)
DE (2) DE4112014A1 (enExample)
DK (1) DK0508370T3 (enExample)
ES (1) ES2090396T3 (enExample)
FI (1) FI97470C (enExample)
GR (1) GR3020860T3 (enExample)
HR (1) HRP940753A2 (enExample)
HU (2) HUT61301A (enExample)
IE (1) IE921147A1 (enExample)
IL (1) IL101560A (enExample)
MX (1) MX9201675A (enExample)
NO (1) NO180303C (enExample)
NZ (1) NZ242305A (enExample)
PL (1) PL169745B1 (enExample)
RU (1) RU2081870C1 (enExample)
SG (1) SG48793A1 (enExample)
SI (1) SI9210325A (enExample)
SK (1) SK279466B6 (enExample)
TW (1) TW205551B (enExample)
YU (1) YU48645B (enExample)
ZA (1) ZA922617B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102478480B1 (ko) 2021-11-17 2022-12-19 주식회사 지농 통신 데이터 사용량을 최소화한 스마트팜 제어 및 동작확인 장치
KR20240109659A (ko) 2023-01-04 2024-07-12 주식회사 다온정보기술 스마트기기를 이용한 스마트팜 제어시스템

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4332168A1 (de) * 1993-02-22 1995-03-23 Thomae Gmbh Dr K Cyclische Derivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
ATE221067T1 (de) * 1993-04-05 2002-08-15 Pharmaceutical Discovery Corp Pyrido(2,3-b)(1,4)benzodiazepinone als m2- rezeptorligand zur behandlung neurologischer störungen
AU3754495A (en) * 1994-10-31 1996-05-23 Yamanouchi Pharmaceutical Co., Ltd. Novel benzodiazepinone derivative and medicinal composition thereof
US5573780A (en) * 1995-08-04 1996-11-12 Apotex Usa Inc. Stable solid formulation of enalapril salt and process for preparation thereof
RU2194707C2 (ru) * 2000-04-04 2002-12-20 Научно-исследовательский институт фармакологии РАМН 2-(2'-ГИДРОКСИ-2'-ЗАМЕЩЕННЫЕ)ЭТИЛ-1,2,3,4-ТЕТРАГИДРОПИРРОЛО[1,2-a]ПИРАЗИНЫ ИЛИ ИХ ФУМАРАТЫ, ОБЛАДАЮЩИЕ АНТИАРИТМИЧЕСКОЙ И ПРОТИВОИШЕМИЧЕСКОЙ АКТИВНОСТЬЮ
US20070105835A1 (en) * 2005-11-07 2007-05-10 Kazantsev Aleksey G Compositions and methods for modulating poly(ADP-ribose) polymerase activity
RU2010103105A (ru) * 2007-07-02 2011-08-10 Ац Иммуне С.А. (Ch) Пирензепин и его производные в качестве анти-амилоидных агентов

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3409237A1 (de) * 1984-03-14 1985-09-19 Dr. Karl Thomae Gmbh, 7950 Biberach Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3735895A1 (de) * 1987-10-23 1989-05-03 Thomae Gmbh Dr K Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3919076A1 (de) * 1989-06-10 1990-12-13 Thomae Gmbh Dr K Mittel zur behandlung von erkrankungen des zentralnervensystems und zur foerderung der cerebralen durchblutung

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102478480B1 (ko) 2021-11-17 2022-12-19 주식회사 지농 통신 데이터 사용량을 최소화한 스마트팜 제어 및 동작확인 장치
KR20240109659A (ko) 2023-01-04 2024-07-12 주식회사 다온정보기술 스마트기기를 이용한 스마트팜 제어시스템

Also Published As

Publication number Publication date
MX9201675A (es) 1992-10-01
PL294184A1 (en) 1993-05-04
RU2081870C1 (ru) 1997-06-20
EP0508370A1 (de) 1992-10-14
CZ111192A3 (en) 1993-04-14
IL101560A0 (en) 1992-12-30
AU653802B2 (en) 1994-10-13
SI9210325A (en) 1995-04-30
SK111192A3 (en) 1995-04-12
KR920019792A (ko) 1992-11-20
NO180303B (no) 1996-12-16
NO921447L (no) 1992-10-13
HUT61301A (en) 1992-12-28
ES2090396T3 (es) 1996-10-16
YU32592A (sh) 1998-09-18
PL169745B1 (pl) 1996-08-30
FI921589A7 (fi) 1992-10-13
FI97470B (fi) 1996-09-13
IL101560A (en) 1996-03-31
NO921447D0 (no) 1992-04-10
ATE140004T1 (de) 1996-07-15
CA2065800A1 (en) 1992-10-13
YU48645B (sh) 1999-06-15
NZ242305A (en) 1994-09-27
NO180303C (no) 1997-03-26
DE59206679D1 (de) 1996-08-08
HRP940753A2 (en) 1997-08-31
FI97470C (fi) 1996-12-27
US5641772A (en) 1997-06-24
FI921589A0 (fi) 1992-04-10
TW205551B (enExample) 1993-05-11
CZ283399B6 (cs) 1998-04-15
DK0508370T3 (da) 1996-11-04
EP0508370B1 (de) 1996-07-03
HU9201247D0 (en) 1992-07-28
SK279466B6 (sk) 1998-11-04
DE4112014A1 (de) 1992-10-15
JPH0597845A (ja) 1993-04-20
IE921147A1 (en) 1992-10-21
SG48793A1 (en) 1998-05-18
HU211156A9 (en) 1995-10-30
AU1481492A (en) 1992-10-15
ZA922617B (en) 1993-10-11
GR3020860T3 (en) 1996-11-30

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