JP5964756B2 - 選択的アンドロゲン受容体モジュレーター - Google Patents

選択的アンドロゲン受容体モジュレーター Download PDF

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JP5964756B2
JP5964756B2 JP2012552115A JP2012552115A JP5964756B2 JP 5964756 B2 JP5964756 B2 JP 5964756B2 JP 2012552115 A JP2012552115 A JP 2012552115A JP 2012552115 A JP2012552115 A JP 2012552115A JP 5964756 B2 JP5964756 B2 JP 5964756B2
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tetrahydro
dichloro
trifluoromethyl
carbazol
mmol
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JP2013518902A (ja
JP2013518902A5 (https=
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ミラー，クリス，ピー．
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ラジウス ヘルス，インコーポレイテッド
ラジウス ヘルス，インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
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  • Medicinal Chemistry (AREA)
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  • Urology & Nephrology (AREA)
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  • Obesity (AREA)
  • Rheumatology (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pain & Pain Management (AREA)
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JP2012552115A 2010-02-04 2011-02-04 選択的アンドロゲン受容体モジュレーター Expired - Fee Related JP5964756B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30149210P 2010-02-04 2010-02-04
US61/301,492 2010-02-04
PCT/US2011/023768 WO2011097496A1 (en) 2010-02-04 2011-02-04 Selective androgen receptor modulators

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JP2016035296A Division JP2016138118A (ja) 2010-02-04 2016-02-26 選択的アンドロゲン受容体モジュレーター

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JP2013518902A JP2013518902A (ja) 2013-05-23
JP2013518902A5 JP2013518902A5 (https=) 2015-05-28
JP5964756B2 true JP5964756B2 (ja) 2016-08-03

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JP2012552115A Expired - Fee Related JP5964756B2 (ja) 2010-02-04 2011-02-04 選択的アンドロゲン受容体モジュレーター
JP2016035296A Pending JP2016138118A (ja) 2010-02-04 2016-02-26 選択的アンドロゲン受容体モジュレーター

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US (3) US8987319B2 (https=)
EP (1) EP2531029B1 (https=)
JP (2) JP5964756B2 (https=)
AU (1) AU2011212813B2 (https=)
BR (1) BR112012019551A2 (https=)
CA (1) CA2788907A1 (https=)
MX (1) MX338831B (https=)
WO (1) WO2011097496A1 (https=)

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EP4464384A3 (en) 2007-08-17 2025-01-08 Purdue Research Foundation Psma binding ligand-linker conjugates and methods for using
MX338831B (es) 2010-02-04 2016-05-03 Radius Health Inc Moduladores selectivos de receptores de androgenos.
US9951324B2 (en) 2010-02-25 2018-04-24 Purdue Research Foundation PSMA binding ligand-linker conjugates and methods for using
EP2568806B1 (en) 2010-05-12 2016-05-11 Radius Health, Inc. Therapeutic regimens
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