BR112012019551A2 - moduladores seletivos do receptor de androgênio. - Google Patents

moduladores seletivos do receptor de androgênio.

Info

Publication number
BR112012019551A2
BR112012019551A2 BR112012019551A BR112012019551A BR112012019551A2 BR 112012019551 A2 BR112012019551 A2 BR 112012019551A2 BR 112012019551 A BR112012019551 A BR 112012019551A BR 112012019551 A BR112012019551 A BR 112012019551A BR 112012019551 A2 BR112012019551 A2 BR 112012019551A2
Authority
BR
Brazil
Prior art keywords
androgen receptor
iia
iii
formula
methods
Prior art date
Application number
BR112012019551A
Other languages
English (en)
Portuguese (pt)
Inventor
Chris P Miller
Original Assignee
Radius Health Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Radius Health Inc filed Critical Radius Health Inc
Publication of BR112012019551A2 publication Critical patent/BR112012019551A2/pt

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
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  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
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  • Endocrinology (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
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BR112012019551A 2010-02-04 2011-02-04 moduladores seletivos do receptor de androgênio. BR112012019551A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30149210P 2010-02-04 2010-02-04
PCT/US2011/023768 WO2011097496A1 (en) 2010-02-04 2011-02-04 Selective androgen receptor modulators

Publications (1)

Publication Number Publication Date
BR112012019551A2 true BR112012019551A2 (pt) 2016-08-09

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Application Number Title Priority Date Filing Date
BR112012019551A BR112012019551A2 (pt) 2010-02-04 2011-02-04 moduladores seletivos do receptor de androgênio.

Country Status (8)

Country Link
US (3) US8987319B2 (https=)
EP (1) EP2531029B1 (https=)
JP (2) JP5964756B2 (https=)
AU (1) AU2011212813B2 (https=)
BR (1) BR112012019551A2 (https=)
CA (1) CA2788907A1 (https=)
MX (1) MX338831B (https=)
WO (1) WO2011097496A1 (https=)

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MX338831B (es) 2010-02-04 2016-05-03 Radius Health Inc Moduladores selectivos de receptores de androgenos.
US9951324B2 (en) 2010-02-25 2018-04-24 Purdue Research Foundation PSMA binding ligand-linker conjugates and methods for using
EP2568806B1 (en) 2010-05-12 2016-05-11 Radius Health, Inc. Therapeutic regimens
US9133182B2 (en) 2010-09-28 2015-09-15 Radius Health, Inc. Selective androgen receptor modulators
CN103172643B (zh) * 2011-12-26 2016-03-02 中国医学科学院药物研究所 黄皮咔唑生物碱及其制备方法和其药物组合物与用途
BR112015011118B1 (pt) 2012-11-15 2022-12-13 Endocyte, Inc Conjugado; composição farmacêutica; e uso de um conjugado
LT4095130T (lt) 2013-10-18 2024-04-25 Novartis Ag Žymėti prostatos specifinio membranos antigeno (psma) inhibitoriai, jų naudojimas kaip vizualizavimo medžiagų ir farmacinių medžiagų prostatos vėžiui gydyti
BR112016010927A2 (pt) 2013-11-14 2017-08-08 Endocyte Inc Conjugado de fórmula
US9682960B2 (en) 2013-12-19 2017-06-20 Endorecherche, Inc. Non-steroidal antiandrogens and selective androgen receptor modulators with a pyridyl moiety
FI3834824T3 (fi) 2014-03-28 2025-12-05 Univ Duke Estrogeenireseptoripositiivisen rintasyövän hoito selektiivisellä estrogeenireseptorin modulaattorilla
US9421264B2 (en) 2014-03-28 2016-08-23 Duke University Method of treating cancer using selective estrogen receptor modulators
US10188759B2 (en) 2015-01-07 2019-01-29 Endocyte, Inc. Conjugates for imaging
JP6757037B2 (ja) * 2016-02-15 2020-09-16 学校法人近畿大学 ストレス評価方法
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