AU2011212813B2 - Selective androgen receptor modulators - Google Patents

Selective androgen receptor modulators Download PDF

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Publication number
AU2011212813B2
AU2011212813B2 AU2011212813A AU2011212813A AU2011212813B2 AU 2011212813 B2 AU2011212813 B2 AU 2011212813B2 AU 2011212813 A AU2011212813 A AU 2011212813A AU 2011212813 A AU2011212813 A AU 2011212813A AU 2011212813 B2 AU2011212813 B2 AU 2011212813B2
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tetrahydro
compound
dichloro
carbazol
trifluoromethyl
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AU2011212813A
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AU2011212813A1 (en
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Chris P. Miller
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Radius Health Inc
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Radius Health Inc
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    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
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AU2011212813A 2010-02-04 2011-02-04 Selective androgen receptor modulators Ceased AU2011212813B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30149210P 2010-02-04 2010-02-04
US61/301,492 2010-02-04
PCT/US2011/023768 WO2011097496A1 (en) 2010-02-04 2011-02-04 Selective androgen receptor modulators

Publications (2)

Publication Number Publication Date
AU2011212813A1 AU2011212813A1 (en) 2012-09-06
AU2011212813B2 true AU2011212813B2 (en) 2014-10-23

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AU2011212813A Ceased AU2011212813B2 (en) 2010-02-04 2011-02-04 Selective androgen receptor modulators

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US (3) US8987319B2 (https=)
EP (1) EP2531029B1 (https=)
JP (2) JP5964756B2 (https=)
AU (1) AU2011212813B2 (https=)
BR (1) BR112012019551A2 (https=)
CA (1) CA2788907A1 (https=)
MX (1) MX338831B (https=)
WO (1) WO2011097496A1 (https=)

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US9951324B2 (en) 2010-02-25 2018-04-24 Purdue Research Foundation PSMA binding ligand-linker conjugates and methods for using
EP2568806B1 (en) 2010-05-12 2016-05-11 Radius Health, Inc. Therapeutic regimens
US9133182B2 (en) 2010-09-28 2015-09-15 Radius Health, Inc. Selective androgen receptor modulators
CN103172643B (zh) * 2011-12-26 2016-03-02 中国医学科学院药物研究所 黄皮咔唑生物碱及其制备方法和其药物组合物与用途
BR112015011118B1 (pt) 2012-11-15 2022-12-13 Endocyte, Inc Conjugado; composição farmacêutica; e uso de um conjugado
LT4095130T (lt) 2013-10-18 2024-04-25 Novartis Ag Žymėti prostatos specifinio membranos antigeno (psma) inhibitoriai, jų naudojimas kaip vizualizavimo medžiagų ir farmacinių medžiagų prostatos vėžiui gydyti
BR112016010927A2 (pt) 2013-11-14 2017-08-08 Endocyte Inc Conjugado de fórmula
US9682960B2 (en) 2013-12-19 2017-06-20 Endorecherche, Inc. Non-steroidal antiandrogens and selective androgen receptor modulators with a pyridyl moiety
FI3834824T3 (fi) 2014-03-28 2025-12-05 Univ Duke Estrogeenireseptoripositiivisen rintasyövän hoito selektiivisellä estrogeenireseptorin modulaattorilla
US9421264B2 (en) 2014-03-28 2016-08-23 Duke University Method of treating cancer using selective estrogen receptor modulators
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