JP2693559B2 - テトラヒドロイミダゾ[1,4]ベンゾジアゼピン―2―オン類 - Google Patents
テトラヒドロイミダゾ[1,4]ベンゾジアゼピン―2―オン類Info
- Publication number
- JP2693559B2 JP2693559B2 JP1059859A JP5985989A JP2693559B2 JP 2693559 B2 JP2693559 B2 JP 2693559B2 JP 1059859 A JP1059859 A JP 1059859A JP 5985989 A JP5985989 A JP 5985989A JP 2693559 B2 JP2693559 B2 JP 2693559B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- hydrogen
- alkyl
- compound
- parts
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Virology (AREA)
- Oncology (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB888806449A GB8806449D0 (en) | 1988-03-18 | 1988-03-18 | Antiviral hexahydroimiazo(1 4)benzodiazepin-2-ones |
GB8806449 | 1988-03-18 |
Publications (2)
Publication Number | Publication Date |
---|---|
JPH01275582A JPH01275582A (ja) | 1989-11-06 |
JP2693559B2 true JP2693559B2 (ja) | 1997-12-24 |
Family
ID=10633662
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP1059859A Expired - Lifetime JP2693559B2 (ja) | 1988-03-18 | 1989-03-14 | テトラヒドロイミダゾ[1,4]ベンゾジアゼピン―2―オン類 |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP0336466B1 (zh) |
JP (1) | JP2693559B2 (zh) |
KR (1) | KR0133073B1 (zh) |
CN (1) | CN1031058C (zh) |
AT (1) | ATE84035T1 (zh) |
AU (2) | AU617435B2 (zh) |
BG (1) | BG51251A3 (zh) |
CA (1) | CA1310964C (zh) |
DE (1) | DE68904102T2 (zh) |
DK (1) | DK130989A (zh) |
ES (1) | ES2053946T3 (zh) |
FI (1) | FI89800C (zh) |
GB (1) | GB8806449D0 (zh) |
GR (1) | GR3006728T3 (zh) |
HU (2) | HU206873B (zh) |
IE (1) | IE63108B1 (zh) |
IL (1) | IL89633A (zh) |
JO (1) | JO1589B1 (zh) |
MY (1) | MY104942A (zh) |
NO (1) | NO167737C (zh) |
NZ (1) | NZ228216A (zh) |
PH (1) | PH27044A (zh) |
PT (1) | PT90034B (zh) |
SU (1) | SU1748647A3 (zh) |
TN (1) | TNSN89039A1 (zh) |
ZA (1) | ZA892062B (zh) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5270464A (en) * | 1989-03-14 | 1993-12-14 | Janssen Pharmaceutica N.V. | Anti-HIV-1 tetrahydroimidazo[1,4]benzodiazepin-2-(thi) ones |
IL93136A (en) * | 1989-02-23 | 1995-01-24 | Janssen Pharmaceutica Nv | History of tetrahydroimidazo [1,4] benzodiazepine-2-thione, their preparation and pharmaceutical preparations containing them |
NZ235137A (en) * | 1989-09-13 | 1992-02-25 | Janssen Pharmaceutica Nv | Tetrahydroimidazo(1,4)benzodiazepine derivatives, preparation and pharmaceutical compositions thereof |
US5164376A (en) * | 1989-10-30 | 1992-11-17 | Hoffmann-Laroche Inc. | Method for treating retroviral infections with aryl-(2-pyrryl) keytone compound |
EP0436245A1 (en) * | 1989-12-27 | 1991-07-10 | Duphar International Research B.V | Substituted 3,4-annelated benzimidazol-2(1H)-ones |
US5141735A (en) * | 1990-06-18 | 1992-08-25 | Hoffman-La Roche, Inc. | Substituted amino-benzodiazepines having anitviral activity |
NZ238664A (en) * | 1990-07-06 | 1992-12-23 | Janssen Pharmaceutica Nv | Substituted tetrahydroimidazo(1,4)benzodiazepin-2-(thi)ones and pharmaceutical anti-viral compositions |
GB9018601D0 (en) * | 1990-08-24 | 1990-10-10 | Fujisawa Pharmaceutical Co | Tricyclic compounds |
DE4036552C1 (zh) * | 1990-11-16 | 1992-02-06 | Boehringer Mannheim Gmbh, 6800 Mannheim, De | |
GB9109557D0 (en) | 1991-05-02 | 1991-06-26 | Wellcome Found | Chemical compounds |
ES2138624T3 (es) * | 1992-05-13 | 2000-01-16 | Wellcome Found | Combinaciones terapeuticas. |
US6177435B1 (en) | 1992-05-13 | 2001-01-23 | Glaxo Wellcome Inc. | Therapeutic combinations |
KR101589314B1 (ko) | 2007-08-20 | 2016-01-28 | 에보텍 인터내셔널 게엠베하 | 수면 장애의 치료 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2534257A1 (fr) * | 1982-10-12 | 1984-04-13 | Roussel Uclaf | Nouveaux derives de la 6-amino 7-hydroxy 4,5,6,7-tetrahydro-imidazo/4,5,1-j-k/ /1/ benzazepin-2(1h)-one, leurs sels, application a titre de medicaments, compositions les renfermant et un intermediaire |
IL93136A (en) * | 1989-02-23 | 1995-01-24 | Janssen Pharmaceutica Nv | History of tetrahydroimidazo [1,4] benzodiazepine-2-thione, their preparation and pharmaceutical preparations containing them |
-
1988
- 1988-03-18 GB GB888806449A patent/GB8806449D0/en active Pending
-
1989
- 1989-02-10 MY MYPI89000163A patent/MY104942A/en unknown
- 1989-03-03 NZ NZ228216A patent/NZ228216A/xx unknown
- 1989-03-08 ES ES89200575T patent/ES2053946T3/es not_active Expired - Lifetime
- 1989-03-08 DE DE8989200575T patent/DE68904102T2/de not_active Expired - Fee Related
- 1989-03-08 EP EP89200575A patent/EP0336466B1/en not_active Expired - Lifetime
- 1989-03-08 AT AT89200575T patent/ATE84035T1/de not_active IP Right Cessation
- 1989-03-13 JO JO19891589A patent/JO1589B1/en active
- 1989-03-14 AU AU31310/89A patent/AU617435B2/en not_active Ceased
- 1989-03-14 JP JP1059859A patent/JP2693559B2/ja not_active Expired - Lifetime
- 1989-03-16 CA CA000593935A patent/CA1310964C/en not_active Expired - Fee Related
- 1989-03-16 IL IL8963389A patent/IL89633A/en not_active IP Right Cessation
- 1989-03-16 IE IE85189A patent/IE63108B1/en not_active IP Right Cessation
- 1989-03-16 HU HU911782A patent/HU206873B/hu not_active IP Right Cessation
- 1989-03-16 HU HU891240A patent/HU203757B/hu not_active IP Right Cessation
- 1989-03-16 BG BG087682A patent/BG51251A3/xx unknown
- 1989-03-17 ZA ZA892062A patent/ZA892062B/xx unknown
- 1989-03-17 PT PT90034A patent/PT90034B/pt not_active IP Right Cessation
- 1989-03-17 DK DK130989A patent/DK130989A/da not_active Application Discontinuation
- 1989-03-17 PH PH38339A patent/PH27044A/en unknown
- 1989-03-17 NO NO891176A patent/NO167737C/no unknown
- 1989-03-17 SU SU894613664A patent/SU1748647A3/ru active
- 1989-03-17 FI FI891279A patent/FI89800C/fi not_active IP Right Cessation
- 1989-03-18 KR KR89003388A patent/KR0133073B1/ko not_active IP Right Cessation
- 1989-03-18 CN CN89101474A patent/CN1031058C/zh not_active Expired - Fee Related
- 1989-03-19 TN TNTNSN89039A patent/TNSN89039A1/fr unknown
-
1991
- 1991-09-02 AU AU83602/91A patent/AU630575B2/en not_active Ceased
-
1992
- 1992-12-31 GR GR920403099T patent/GR3006728T3/el unknown
Also Published As
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