JP2019517996A5 - - Google Patents

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Publication number
JP2019517996A5
JP2019517996A5 JP2018550733A JP2018550733A JP2019517996A5 JP 2019517996 A5 JP2019517996 A5 JP 2019517996A5 JP 2018550733 A JP2018550733 A JP 2018550733A JP 2018550733 A JP2018550733 A JP 2018550733A JP 2019517996 A5 JP2019517996 A5 JP 2019517996A5
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JP
Japan
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methyl
pyrazolo
pyridin
tetrahydropyran
group
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JP2018550733A
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Japanese (ja)
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JP7093306B2 (ja
JP2019517996A (ja
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Priority claimed from PCT/EP2017/058332 external-priority patent/WO2017178350A1/en
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Publication of JP2019517996A5 publication Critical patent/JP2019517996A5/ja
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JP2018550733A 2016-04-12 2017-04-07 ＰＤＥ１阻害剤としての１，５－ジヒドロ－４Ｈ－ピラゾロ［３，４－ｄ］ピリミジン－４－オン及び１，５－ジヒドロ－４Ｈ－ピラゾロ［４，３－ｃ］ピリジン－４－オン Expired - Fee Related JP7093306B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA201600221 2016-04-12
DKPA201600221 2016-04-12
PCT/EP2017/058332 WO2017178350A1 (en) 2016-04-12 2017-04-07 1,5-dihydro-4h-pyrazolo[3,4-d]pyrimidin-4-ones and 1,5-dihydro-4h-pyrazolo[4,3-c]pyridin-4-ones as pde1 inhibitors

Publications (3)

Publication Number Publication Date
JP2019517996A JP2019517996A (ja) 2019-06-27
JP2019517996A5 true JP2019517996A5 (enExample) 2020-05-07
JP7093306B2 JP7093306B2 (ja) 2022-06-29

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JP2018550733A Expired - Fee Related JP7093306B2 (ja) 2016-04-12 2017-04-07 ＰＤＥ１阻害剤としての１，５－ジヒドロ－４Ｈ－ピラゾロ［３，４－ｄ］ピリミジン－４－オン及び１，５－ジヒドロ－４Ｈ－ピラゾロ［４，３－ｃ］ピリジン－４－オン

Country Status (43)

Country Link
US (3) US20170291901A1 (enExample)
EP (1) EP3442975B1 (enExample)
JP (1) JP7093306B2 (enExample)
KR (1) KR20180133413A (enExample)
CN (1) CN109071549B (enExample)
AR (1) AR108109A1 (enExample)
AU (1) AU2017250431B2 (enExample)
BR (1) BR112017026278A2 (enExample)
CA (1) CA3020053A1 (enExample)
CL (1) CL2018002881A1 (enExample)
CO (1) CO2018010323A2 (enExample)
CR (1) CR20180470A (enExample)
CY (1) CY1123269T1 (enExample)
DK (1) DK3442975T3 (enExample)
DO (1) DOP2018000201A (enExample)
EA (1) EA035197B1 (enExample)
EC (1) ECSP18074641A (enExample)
ES (1) ES2814289T3 (enExample)
GE (2) GEAP201914901A (enExample)
HR (1) HRP20201331T1 (enExample)
HU (1) HUE050320T2 (enExample)
IL (1) IL262257B (enExample)
LT (1) LT3442975T (enExample)
MA (1) MA44656B1 (enExample)
ME (1) ME03820B (enExample)
MX (1) MX374251B (enExample)
MY (1) MY194722A (enExample)
NI (1) NI201800092A (enExample)
PE (1) PE20181853A1 (enExample)
PH (1) PH12018502168A1 (enExample)
PL (1) PL3442975T3 (enExample)
PT (1) PT3442975T (enExample)
RS (1) RS60714B1 (enExample)
RU (1) RU2018133391A (enExample)
SG (1) SG11201808221QA (enExample)
SI (1) SI3442975T1 (enExample)
SM (1) SMT202000446T1 (enExample)
SV (1) SV2018005753A (enExample)
TN (1) TN2018000321A1 (enExample)
TW (1) TWI729109B (enExample)
UA (1) UA121925C2 (enExample)
WO (1) WO2017178350A1 (enExample)
ZA (1) ZA201806407B (enExample)

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JO3627B1 (ar) 2015-04-30 2020-08-27 H Lundbeck As إيميدازو بيرازينونات على هيئة مثبطات pde1
TWI729109B (zh) 2016-04-12 2021-06-01 丹麥商Ｈ 朗德貝克公司 作爲PDE1抑制劑的1,5-二氫-4H-吡唑并[3,4-d]嘧啶-4-酮和1,5-二氫-4H-吡唑并[4,3-c]吡啶-4-酮
EP3529250B1 (en) 2016-10-18 2023-12-06 H. Lundbeck A/S Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as pde1 inhibitors
BR112018013084A2 (pt) 2016-10-28 2018-12-11 H Lundbeck As tratamentos de combinação compreendendo a administração de imidazopirazinonas
SG11201903770UA (en) 2016-10-28 2019-05-30 H Lundbeck As Combination treatments comprising imidazopyrazinones for the treatment of psychiatric and/or cognitive disorders
KR102590848B1 (ko) 2016-12-28 2023-10-19 다트 뉴로사이언스, 엘엘씨 Pde2 억제제로서 치환된 피라졸로피리미디논 화합물
ES2902365T3 (es) * 2017-11-27 2022-03-28 Dart Neuroscience Llc Compuestos de furanopirimidina sustituidos como inhibidores de PDE1
KR20210013214A (ko) 2018-05-25 2021-02-03 인트라-셀룰라 써래피스, 인코퍼레이티드. 유기 화합물
WO2020210614A1 (en) 2019-04-12 2020-10-15 Intra-Cellular Therapies, Inc. Organic compounds
CN115304607B (zh) * 2022-07-06 2023-06-27 华南农业大学 吡唑并嘧啶衍生物的制备方法

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JO3627B1 (ar) 2015-04-30 2020-08-27 H Lundbeck As إيميدازو بيرازينونات على هيئة مثبطات pde1
AR107456A1 (es) 2016-02-12 2018-05-02 Lilly Co Eli Inhibidor de pde1
TWI729109B (zh) 2016-04-12 2021-06-01 丹麥商Ｈ 朗德貝克公司 作爲PDE1抑制劑的1,5-二氫-4H-吡唑并[3,4-d]嘧啶-4-酮和1,5-二氫-4H-吡唑并[4,3-c]吡啶-4-酮
JP2018076285A (ja) 2016-09-14 2018-05-17 大日本住友製薬株式会社 二環性イミダゾロ誘導体を含む医薬
EP3529250B1 (en) 2016-10-18 2023-12-06 H. Lundbeck A/S Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as pde1 inhibitors
SG11201903770UA (en) 2016-10-28 2019-05-30 H Lundbeck As Combination treatments comprising imidazopyrazinones for the treatment of psychiatric and/or cognitive disorders
BR112018013084A2 (pt) 2016-10-28 2018-12-11 H Lundbeck As tratamentos de combinação compreendendo a administração de imidazopirazinonas

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