JP2019513746A5 - - Google Patents
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- JP2019513746A5 JP2019513746A5 JP2018552788A JP2018552788A JP2019513746A5 JP 2019513746 A5 JP2019513746 A5 JP 2019513746A5 JP 2018552788 A JP2018552788 A JP 2018552788A JP 2018552788 A JP2018552788 A JP 2018552788A JP 2019513746 A5 JP2019513746 A5 JP 2019513746A5
- Authority
- JP
- Japan
- Prior art keywords
- dione
- oxoisoindoline
- piperidine
- amino
- dioxopiperidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 C*(C)(C)c1c[n](C)cn1 Chemical compound C*(C)(C)c1c[n](C)cn1 0.000 description 5
- CFPJFKUXYOFKCX-SREVYHEPSA-N CC(/N=N\N(C)C)=C Chemical compound CC(/N=N\N(C)C)=C CFPJFKUXYOFKCX-SREVYHEPSA-N 0.000 description 1
- XNGFRIKTXZKULT-UHFFFAOYSA-N CC1=NCN(C)N=C1 Chemical compound CC1=NCN(C)N=C1 XNGFRIKTXZKULT-UHFFFAOYSA-N 0.000 description 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021210079A JP2022050469A (ja) | 2016-04-06 | 2021-12-24 | リガンド依存性の標的タンパク質分解のための単官能性中間体 |
Applications Claiming Priority (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662318974P | 2016-04-06 | 2016-04-06 | |
| US62/318,974 | 2016-04-06 | ||
| US201662321499P | 2016-04-12 | 2016-04-12 | |
| US62/321,499 | 2016-04-12 | ||
| US201662393935P | 2016-09-13 | 2016-09-13 | |
| US201662393888P | 2016-09-13 | 2016-09-13 | |
| US201662393874P | 2016-09-13 | 2016-09-13 | |
| US62/393,935 | 2016-09-13 | ||
| US62/393,888 | 2016-09-13 | ||
| US62/393,874 | 2016-09-13 | ||
| US201662409571P | 2016-10-18 | 2016-10-18 | |
| US201662409592P | 2016-10-18 | 2016-10-18 | |
| US62/409,571 | 2016-10-18 | ||
| US62/409,592 | 2016-10-18 | ||
| PCT/US2017/026275 WO2017176958A1 (en) | 2016-04-06 | 2017-04-06 | Monofunctional intermediates for ligand-dependent target protein degradation |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021210079A Division JP2022050469A (ja) | 2016-04-06 | 2021-12-24 | リガンド依存性の標的タンパク質分解のための単官能性中間体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019513746A JP2019513746A (ja) | 2019-05-30 |
| JP2019513746A5 true JP2019513746A5 (https=) | 2020-05-14 |
| JP7001614B2 JP7001614B2 (ja) | 2022-02-03 |
Family
ID=58549317
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018552788A Expired - Fee Related JP7001614B2 (ja) | 2016-04-06 | 2017-04-06 | リガンド依存性の標的タンパク質分解のための単官能性中間体 |
| JP2021210079A Withdrawn JP2022050469A (ja) | 2016-04-06 | 2021-12-24 | リガンド依存性の標的タンパク質分解のための単官能性中間体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021210079A Withdrawn JP2022050469A (ja) | 2016-04-06 | 2021-12-24 | リガンド依存性の標的タンパク質分解のための単官能性中間体 |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US10759808B2 (https=) |
| EP (1) | EP3440082A1 (https=) |
| JP (2) | JP7001614B2 (https=) |
| CN (1) | CN109311900A (https=) |
| AU (2) | AU2017246453A1 (https=) |
| CA (1) | CA3020281A1 (https=) |
| WO (1) | WO2017176958A1 (https=) |
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-
2017
- 2017-04-06 US US16/091,544 patent/US10759808B2/en active Active
- 2017-04-06 JP JP2018552788A patent/JP7001614B2/ja not_active Expired - Fee Related
- 2017-04-06 CN CN201780035311.3A patent/CN109311900A/zh active Pending
- 2017-04-06 AU AU2017246453A patent/AU2017246453A1/en not_active Abandoned
- 2017-04-06 CA CA3020281A patent/CA3020281A1/en active Pending
- 2017-04-06 WO PCT/US2017/026275 patent/WO2017176958A1/en not_active Ceased
- 2017-04-06 EP EP17718291.2A patent/EP3440082A1/en not_active Withdrawn
-
2020
- 2020-08-31 US US17/007,191 patent/US20210002289A1/en not_active Abandoned
-
2021
- 2021-09-15 AU AU2021232732A patent/AU2021232732A1/en not_active Abandoned
- 2021-12-24 JP JP2021210079A patent/JP2022050469A/ja not_active Withdrawn
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