JP2017522340A5 - - Google Patents

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JP2017522340A5
JP2017522340A5 JP2017504775A JP2017504775A JP2017522340A5 JP 2017522340 A5 JP2017522340 A5 JP 2017522340A5 JP 2017504775 A JP2017504775 A JP 2017504775A JP 2017504775 A JP2017504775 A JP 2017504775A JP 2017522340 A5 JP2017522340 A5 JP 2017522340A5
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alkyl
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disorders
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hydrogen
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JP6662846B2 (ja
JP2017522340A (ja
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Priority claimed from PCT/EP2015/067530 external-priority patent/WO2016016380A1/en
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JP2017504775A 2014-08-01 2015-07-30 ６，７−ジヒドロピラゾロ［１，５−ａ］ピラジン−４（５Ｈ）−オン化合物およびＭＧＬＵＲ２受容体の負のアロステリック調節因子としてのそれらの使用 Expired - Fee Related JP6662846B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14179598 2014-08-01
EP14179598.9 2014-08-01
PCT/EP2015/067530 WO2016016380A1 (en) 2014-08-01 2015-07-30 6,7-DIHYDROPYRAZOLO[1,5-α]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS

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JP2017522340A JP2017522340A (ja) 2017-08-10
JP2017522340A5 true JP2017522340A5 (enExample) 2018-08-23
JP6662846B2 JP6662846B2 (ja) 2020-03-11

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JP2017504775A Expired - Fee Related JP6662846B2 (ja) 2014-08-01 2015-07-30 ６，７−ジヒドロピラゾロ［１，５−ａ］ピラジン−４（５Ｈ）−オン化合物およびＭＧＬＵＲ２受容体の負のアロステリック調節因子としてのそれらの使用

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US (3) US10005786B2 (enExample)
EP (1) EP3177623B1 (enExample)
JP (1) JP6662846B2 (enExample)
KR (1) KR102531689B1 (enExample)
CN (1) CN106573936B (enExample)
AR (1) AR101392A1 (enExample)
AU (1) AU2015295298B2 (enExample)
BR (1) BR112017001726A2 (enExample)
CA (1) CA2954093C (enExample)
CL (1) CL2017000192A1 (enExample)
CY (1) CY1121649T1 (enExample)
DK (1) DK3177623T3 (enExample)
EA (1) EA031087B1 (enExample)
ES (1) ES2708215T3 (enExample)
HR (1) HRP20181997T1 (enExample)
HU (1) HUE042871T2 (enExample)
IL (1) IL250298A0 (enExample)
JO (1) JOP20150179B1 (enExample)
LT (1) LT3177623T (enExample)
MA (1) MA39582B1 (enExample)
ME (1) ME03320B (enExample)
MX (1) MX376289B (enExample)
NZ (1) NZ728122A (enExample)
PH (1) PH12017500161B1 (enExample)
PL (1) PL3177623T3 (enExample)
PT (1) PT3177623T (enExample)
RS (1) RS58279B1 (enExample)
SG (1) SG11201700638YA (enExample)
SI (1) SI3177623T1 (enExample)
SM (1) SMT201900038T1 (enExample)
TR (1) TR201901074T4 (enExample)
TW (1) TWI696624B (enExample)
WO (1) WO2016016380A1 (enExample)
ZA (1) ZA201700759B (enExample)

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JP6861154B2 (ja) 2014-12-03 2021-04-21 ヤンセン ファーマシューティカ エヌ．ベー． 放射標識されたｍＧｌｕＲ２ ＰＥＴリガンド
EP3227295B1 (en) 2014-12-03 2019-02-20 Janssen Pharmaceutica NV 6,7-dihydropyrazolo[1,5- ]pyrazin-4(5h)-one compounds and their use as negative allosteric modulators of mglu2 receptors
CA3003962A1 (en) 2015-12-18 2017-06-22 Janssen Pharmaceutica Nv Radiolabelled mglur2/3 pet ligands
PL3389727T3 (pl) 2015-12-18 2021-02-08 Janssen Pharmaceutica Nv RADIOZNAKOWANE LIGANDY mGluR2/3 DO PET

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