JP2015512433A5 - - Google Patents

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Publication number
JP2015512433A5
JP2015512433A5 JP2015503848A JP2015503848A JP2015512433A5 JP 2015512433 A5 JP2015512433 A5 JP 2015512433A5 JP 2015503848 A JP2015503848 A JP 2015503848A JP 2015503848 A JP2015503848 A JP 2015503848A JP 2015512433 A5 JP2015512433 A5 JP 2015512433A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
weight
disintegrant
diluent
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JP2015503848A
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English (en)
Japanese (ja)
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JP6320990B2 (ja
JP2015512433A (ja
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Priority claimed from PCT/EP2013/056867 external-priority patent/WO2013149987A1/en
Publication of JP2015512433A publication Critical patent/JP2015512433A/ja
Publication of JP2015512433A5 publication Critical patent/JP2015512433A5/ja
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Publication of JP6320990B2 publication Critical patent/JP6320990B2/ja
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JP2015503848A 2012-04-04 2013-04-02 Ｃｃｒ３アンタゴニストを含む医薬製剤 Active JP6320990B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12163078.4 2012-04-04
EP12163078 2012-04-04
PCT/EP2013/056867 WO2013149987A1 (en) 2012-04-04 2013-04-02 Pharmaceutical formulations comprising ccr3 antagonists

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2018072309A Division JP6700332B2 (ja) 2012-04-04 2018-04-04 Ｃｃｒ３アンタゴニストを含む医薬製剤

Publications (3)

Publication Number Publication Date
JP2015512433A JP2015512433A (ja) 2015-04-27
JP2015512433A5 true JP2015512433A5 (enExample) 2016-06-02
JP6320990B2 JP6320990B2 (ja) 2018-05-09

Family

ID=49292482

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2015503848A Active JP6320990B2 (ja) 2012-04-04 2013-04-02 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2018072309A Active JP6700332B2 (ja) 2012-04-04 2018-04-04 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2020080024A Pending JP2020143080A (ja) 2012-04-04 2020-04-30 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2022026735A Pending JP2022081524A (ja) 2012-04-04 2022-02-24 Ｃｃｒ３アンタゴニストを含む医薬製剤

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP2018072309A Active JP6700332B2 (ja) 2012-04-04 2018-04-04 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2020080024A Pending JP2020143080A (ja) 2012-04-04 2020-04-30 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2022026735A Pending JP2022081524A (ja) 2012-04-04 2022-02-24 Ｃｃｒ３アンタゴニストを含む医薬製剤

Country Status (31)

Country Link
US (3) US10213421B2 (enExample)
EP (3) EP3524230B1 (enExample)
JP (4) JP6320990B2 (enExample)
KR (2) KR102338465B1 (enExample)
CN (1) CN104203213A (enExample)
AR (1) AR090596A1 (enExample)
AU (1) AU2013245028B2 (enExample)
BR (1) BR112014024479A8 (enExample)
CA (1) CA2869058C (enExample)
CL (1) CL2014002524A1 (enExample)
CY (1) CY1121137T1 (enExample)
DK (2) DK3524230T3 (enExample)
EA (1) EA027627B1 (enExample)
ES (3) ES3044310T3 (enExample)
HR (1) HRP20190069T1 (enExample)
HU (2) HUE056943T2 (enExample)
IL (1) IL234299A (enExample)
IN (1) IN2014DN07082A (enExample)
LT (1) LT2833864T (enExample)
MX (1) MX358307B (enExample)
NZ (1) NZ628993A (enExample)
PH (1) PH12014502241A1 (enExample)
PL (2) PL2833864T3 (enExample)
PT (2) PT2833864T (enExample)
RS (1) RS58360B1 (enExample)
SI (1) SI2833864T1 (enExample)
SM (1) SMT201900121T1 (enExample)
TR (1) TR201821285T4 (enExample)
TW (1) TW201400115A (enExample)
UY (1) UY34730A (enExample)
WO (1) WO2013149987A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
US11382907B2 (en) * 2017-04-05 2022-07-12 Alkahest, Inc. Methods and compositions for treating aging-associated impairments using CCR3-inhibitors
SG11201909207VA (en) 2017-04-05 2019-11-28 Alkahest Inc Methods and compositions for treating retina-associated disease using ccr3-inhibitors
WO2019075351A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. METHODS AND COMPOSITIONS FOR TREATING PRURIT, XEROSIS AND ASSOCIATED DISEASE USING CCR3 INHIBITORS
MY198220A (en) 2018-05-15 2023-08-14 Alkahest Inc Treatment Of Aging-Associated Disease With Modulators Of Leukotriene A4 Hydrolase
AU2019346456A1 (en) * 2018-09-26 2021-04-15 Alkahest, Inc. Methods and compositions for treating aging-associated impairments using CCR3-inhibitors
KR20230056017A (ko) 2020-08-27 2023-04-26 에이지씨 가부시키가이샤 무알칼리 유리 및 유리판
WO2023076679A1 (en) 2021-11-01 2023-05-04 Alkahest, Inc. Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases

Family Cites Families (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7907121L (sv) 1979-08-27 1981-02-28 Astra Laekemedel Ab Ftalimidinderivat
US4992277A (en) 1989-08-25 1991-02-12 Schering Corporation Immediate release diltiazem formulation
JP2807577B2 (ja) 1990-06-15 1998-10-08 エーザイ株式会社 環状アミド誘導体
IL116539A (en) * 1995-01-06 2002-02-10 Noven Pharma Preparations given through the skin of unstable anti-acid drugs
WO1998050019A1 (en) * 1997-05-09 1998-11-12 Sage Pharmaceuticals, Inc. Stable oral pharmaceutical dosage forms
CA2318088A1 (en) 1998-01-21 1999-07-29 Yoshisuke Nakasato Chemokine receptor antagonists and methods of use therefor
JP2002501898A (ja) 1998-02-02 2002-01-22 メルク エンド カムパニー インコーポレーテッド ケモカイン受容体活性の環状アミン調節剤
US6140349A (en) 1998-02-02 2000-10-31 Merck & Co., Inc. Cyclic amine modulators of chemokine receptor activity
SE9802973D0 (sv) 1998-09-03 1998-09-03 Astra Ab Immediate release tablet
EP2305257A1 (en) * 2002-07-08 2011-04-06 ChemGenex Pharmaceuticals, Inc. Amonafide salts and compositions comprising same
JP4792392B2 (ja) 2003-09-11 2011-10-12 コーナーストーン セラピューティクス インコーポレイテッド Ｈｍｇｂ１に対するモノクローナル抗体
WO2005040129A2 (en) 2003-10-24 2005-05-06 F. Hoffmann-La Roche Ag Ccr3 receptor antagonists
NZ547314A (en) 2003-11-17 2010-02-26 Boehringer Ingelheim Int Novel piperidine-substituted indoles- or hetero-derivatives thereof and their use as modulators of chemokine receptor (CCR-3)
ATE428422T1 (de) 2004-02-05 2009-05-15 Schering Corp Piperidin-derivate als ccr3-antagonisten
JP2006137718A (ja) 2004-11-12 2006-06-01 Astellas Pharma Inc インドール若しくはインダゾール誘導体
US8030003B2 (en) 2004-12-07 2011-10-04 Children's Hospital Medical Center Diagnosis of eosinophilic esophagitis based on presence of an elevated level of eotaxin-3
DOP2006000051A (es) 2005-02-24 2006-08-31 Lilly Co Eli Inhibidores de vegf-r2 y métodos
JP3701964B1 (ja) 2005-03-08 2005-10-05 アステラス製薬株式会社 キヌクリジン誘導体の新規な塩
EP1994019B1 (en) 2005-04-30 2011-11-02 Boehringer Ingelheim International GmbH Novel piperidin - substituted indoles and their use as ccr-3 modulators
NL2000323C2 (nl) * 2005-12-20 2007-11-20 Pfizer Ltd Pyrimidine-derivaten.
US20090124636A1 (en) 2006-04-12 2009-05-14 Pfizer Inc. Chemical compounds
US8148403B2 (en) 2006-10-27 2012-04-03 Boehringer Ingelheim International Gmbh Substituted piperidyl-propane-thiols
US8153660B2 (en) 2006-10-27 2012-04-10 Boehringer Ingelheim International Gmbh Piperidyl-propane-thiol CCR3 modulators
GB0701992D0 (en) 2007-02-02 2007-03-14 7Tm Pharma As Grehlin Receptor Modulators
US8008092B2 (en) 2007-10-09 2011-08-30 University Of Kentucky Research Foundation CCR3 inhibition for ocular angiogenesis and macular degeneration
EP2222649A2 (en) 2007-10-24 2010-09-01 Generics (UK) Limited Novel crystalline forms
TW201000446A (en) 2008-05-30 2010-01-01 Astrazeneca Ab New compounds useful in pain therapy
WO2010052727A1 (en) * 2008-11-04 2010-05-14 Ideal Cures Private Limited High performance film coating compositions
US8278302B2 (en) * 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
KR20120070629A (ko) * 2009-04-22 2012-06-29 액시킨 파마수티컬스 인코포레이티드 2,5-이치환 아릴설폰아마이드 ｃｃｒ3 길항제
EP2749554B1 (en) 2009-04-22 2017-12-20 SMA Therapeutics, Inc. 2,5-disubstituted arylsulfonamide CCR3 antagonists
WO2011083402A2 (en) * 2010-01-11 2011-07-14 Muneera Mohamed Shafee Immediate release compositions of acid labile drugs
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US20130261153A1 (en) 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists

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