JP2015512433A5 - - Google Patents
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- JP2015512433A5 JP2015512433A5 JP2015503848A JP2015503848A JP2015512433A5 JP 2015512433 A5 JP2015512433 A5 JP 2015512433A5 JP 2015503848 A JP2015503848 A JP 2015503848A JP 2015503848 A JP2015503848 A JP 2015503848A JP 2015512433 A5 JP2015512433 A5 JP 2015512433A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- composition according
- weight
- disintegrant
- diluent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12163078.4 | 2012-04-04 | ||
| EP12163078 | 2012-04-04 | ||
| PCT/EP2013/056867 WO2013149987A1 (en) | 2012-04-04 | 2013-04-02 | Pharmaceutical formulations comprising ccr3 antagonists |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018072309A Division JP6700332B2 (ja) | 2012-04-04 | 2018-04-04 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015512433A JP2015512433A (ja) | 2015-04-27 |
| JP2015512433A5 true JP2015512433A5 (enExample) | 2016-06-02 |
| JP6320990B2 JP6320990B2 (ja) | 2018-05-09 |
Family
ID=49292482
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015503848A Active JP6320990B2 (ja) | 2012-04-04 | 2013-04-02 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
| JP2018072309A Active JP6700332B2 (ja) | 2012-04-04 | 2018-04-04 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
| JP2020080024A Pending JP2020143080A (ja) | 2012-04-04 | 2020-04-30 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
| JP2022026735A Pending JP2022081524A (ja) | 2012-04-04 | 2022-02-24 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018072309A Active JP6700332B2 (ja) | 2012-04-04 | 2018-04-04 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
| JP2020080024A Pending JP2020143080A (ja) | 2012-04-04 | 2020-04-30 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
| JP2022026735A Pending JP2022081524A (ja) | 2012-04-04 | 2022-02-24 | Ｃｃｒ３アンタゴニストを含む医薬製剤 |
Country Status (31)
| Country | Link |
|---|---|
| US (3) | US10213421B2 (enExample) |
| EP (3) | EP2833864B1 (enExample) |
| JP (4) | JP6320990B2 (enExample) |
| KR (2) | KR102338465B1 (enExample) |
| CN (1) | CN104203213A (enExample) |
| AR (1) | AR090596A1 (enExample) |
| AU (1) | AU2013245028B2 (enExample) |
| BR (1) | BR112014024479A8 (enExample) |
| CA (1) | CA2869058C (enExample) |
| CL (1) | CL2014002524A1 (enExample) |
| CY (1) | CY1121137T1 (enExample) |
| DK (2) | DK3524230T3 (enExample) |
| EA (1) | EA027627B1 (enExample) |
| ES (3) | ES3044310T3 (enExample) |
| HR (1) | HRP20190069T1 (enExample) |
| HU (2) | HUE041519T2 (enExample) |
| IL (1) | IL234299A (enExample) |
| IN (1) | IN2014DN07082A (enExample) |
| LT (1) | LT2833864T (enExample) |
| MX (1) | MX358307B (enExample) |
| NZ (1) | NZ628993A (enExample) |
| PH (1) | PH12014502241A1 (enExample) |
| PL (2) | PL3524230T3 (enExample) |
| PT (2) | PT2833864T (enExample) |
| RS (1) | RS58360B1 (enExample) |
| SI (1) | SI2833864T1 (enExample) |
| SM (1) | SMT201900121T1 (enExample) |
| TR (1) | TR201821285T4 (enExample) |
| TW (1) | TW201400115A (enExample) |
| UY (1) | UY34730A (enExample) |
| WO (1) | WO2013149987A1 (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8278302B2 (en) | 2009-04-08 | 2012-10-02 | Boehringer Ingelheim International Gmbh | Substituted piperidines as CCR3 antagonists |
| UA109290C2 (uk) | 2010-10-07 | 2015-08-10 | Спільні кристали і солі інгібіторів ccr3 | |
| AR090566A1 (es) | 2012-04-02 | 2014-11-19 | Boehringer Ingelheim Int | Proceso para la produccion de inhibidores de crr |
| US20130261153A1 (en) * | 2012-04-03 | 2013-10-03 | Boehringer Ingelheim International Gmbh | Use of ccr3-inhibitors |
| US10213421B2 (en) * | 2012-04-04 | 2019-02-26 | Alkahest, Inc. | Pharmaceutical formulations comprising CCR3 antagonists |
| NZ757769A (en) * | 2017-04-05 | 2025-10-31 | Alkahest Inc | Methods and compositions for treating retina-associated disease using ccr3-inhibitors |
| WO2018187503A1 (en) * | 2017-04-05 | 2018-10-11 | Alkahest, Inc. | Methods and compositions for treating aging-associated impairments using ccr3-inhibitors |
| JP2020536929A (ja) * | 2017-10-13 | 2020-12-17 | アルカヘスト，インコーポレイテッド | Ｃｃｒ３阻害剤を用いた、そう痒症、乾皮症、及び関連疾患を治療するための方法及び組成物 |
| AU2019271122A1 (en) | 2018-05-15 | 2020-11-12 | Alkahest, Inc. | Treatment of aging-associated disease with modulators of leukotriene A4 hydrolase |
| CA3111433A1 (en) * | 2018-09-26 | 2020-04-02 | Alkahest, Inc. | Methods and compositions for treating aging-associated impairments using ccr3-inhibitors |
| JPWO2022045226A1 (enExample) | 2020-08-27 | 2022-03-03 | ||
| US11957671B2 (en) | 2021-11-01 | 2024-04-16 | Alkahest, Inc. | Benzodioxane modulators of leukotriene A4 hydrolase (LTA4H) for prevention and treatment of aging-associated diseases |
Family Cites Families (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7907121L (sv) | 1979-08-27 | 1981-02-28 | Astra Laekemedel Ab | Ftalimidinderivat |
| US4992277A (en) | 1989-08-25 | 1991-02-12 | Schering Corporation | Immediate release diltiazem formulation |
| JP2807577B2 (ja) | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
| IL116539A (en) * | 1995-01-06 | 2002-02-10 | Noven Pharma | Preparations given through the skin of unstable anti-acid drugs |
| TW550090B (en) * | 1997-05-09 | 2003-09-01 | Sage Pharmaceuticals Inc | Stable oral pharmaceutical dosage forms for acid-unstable drug |
| EP1047675A1 (en) | 1998-01-21 | 2000-11-02 | Millennium Pharmaceuticals, Inc. | Chemokine receptor antagonists and methods of use therefor |
| JP2002501898A (ja) | 1998-02-02 | 2002-01-22 | メルク エンド カムパニー インコーポレーテッド | ケモカイン受容体活性の環状アミン調節剤 |
| US6140349A (en) | 1998-02-02 | 2000-10-31 | Merck & Co., Inc. | Cyclic amine modulators of chemokine receptor activity |
| SE9802973D0 (sv) | 1998-09-03 | 1998-09-03 | Astra Ab | Immediate release tablet |
| EP1539150A4 (en) * | 2002-07-08 | 2006-10-11 | Chemgenex Pharmaceuticals Inc | SYNTHESIS OF NAPHTHALIMIDES, INCLUDING AMONAFIDS, AND PHARMACEUTICAL PREPARATIONS CONTAINING SAME |
| CA2538763C (en) | 2003-09-11 | 2015-05-05 | Critical Therapeutics, Inc. | Monoclonal antibodies against hmgb1 |
| KR20060061393A (ko) | 2003-10-24 | 2006-06-07 | 에프. 호프만-라 로슈 아게 | Ｃｃｒ3 수용체 길항제 |
| BRPI0416665A (pt) | 2003-11-17 | 2007-01-16 | Boehringer Ingelheim Int | indóis substituìdos com piperidina ou heteroderivados dos mesmos |
| ES2324224T3 (es) | 2004-02-05 | 2009-08-03 | Schering Corporation | Derivados de piperidina que se pueden utilizar como antagonistas ccr3. |
| JP2006137718A (ja) | 2004-11-12 | 2006-06-01 | Astellas Pharma Inc | インドール若しくはインダゾール誘導体 |
| WO2006083390A2 (en) | 2004-12-07 | 2006-08-10 | Children's Hospital Medical Center | Eotaxin-3 in eosinophilic esophagitis |
| DOP2006000051A (es) | 2005-02-24 | 2006-08-31 | Lilly Co Eli | Inhibidores de vegf-r2 y métodos |
| JP3701964B1 (ja) | 2005-03-08 | 2005-10-05 | アステラス製薬株式会社 | キヌクリジン誘導体の新規な塩 |
| JP5080450B2 (ja) | 2005-04-30 | 2012-11-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 新規なピペリジン置換インドール |
| NL2000323C2 (nl) * | 2005-12-20 | 2007-11-20 | Pfizer Ltd | Pyrimidine-derivaten. |
| EP2059515A2 (en) | 2006-04-12 | 2009-05-20 | Pfizer Limited | Pyrrolidine derivatives as modulators of chemokine ccr5 receptors |
| WO2008049875A1 (en) | 2006-10-27 | 2008-05-02 | Boehringer Ingelheim International Gmbh | Novel substituted piperidyl-propane-thiols |
| ATE537166T1 (de) | 2006-10-27 | 2011-12-15 | Boehringer Ingelheim Int | Piperidylpropanthiole als ccr3-modulatoren |
| GB0701992D0 (en) | 2007-02-02 | 2007-03-14 | 7Tm Pharma As | Grehlin Receptor Modulators |
| US8008092B2 (en) | 2007-10-09 | 2011-08-30 | University Of Kentucky Research Foundation | CCR3 inhibition for ocular angiogenesis and macular degeneration |
| JP2011500780A (ja) | 2007-10-24 | 2011-01-06 | ジェネリクス・（ユーケー）・リミテッド | 新規結晶形 |
| TW201000446A (en) | 2008-05-30 | 2010-01-01 | Astrazeneca Ab | New compounds useful in pain therapy |
| WO2010052727A1 (en) * | 2008-11-04 | 2010-05-14 | Ideal Cures Private Limited | High performance film coating compositions |
| US8278302B2 (en) * | 2009-04-08 | 2012-10-02 | Boehringer Ingelheim International Gmbh | Substituted piperidines as CCR3 antagonists |
| AR078120A1 (es) * | 2009-04-22 | 2011-10-19 | Axikin Pharmaceuticals Inc | Antagonistas de ccr3 de arilsulfonamida 2,5-disustituida y composiciones farmaceuticas |
| TWI510469B (zh) | 2009-04-22 | 2015-12-01 | Axikin Pharmaceuticals Inc | ２，５－雙取代芳基磺醯胺ｃｃｒ３拮抗劑 |
| WO2011083402A2 (en) * | 2010-01-11 | 2011-07-14 | Muneera Mohamed Shafee | Immediate release compositions of acid labile drugs |
| UA109290C2 (uk) | 2010-10-07 | 2015-08-10 | Спільні кристали і солі інгібіторів ccr3 | |
| AR090566A1 (es) | 2012-04-02 | 2014-11-19 | Boehringer Ingelheim Int | Proceso para la produccion de inhibidores de crr |
| US20130261153A1 (en) | 2012-04-03 | 2013-10-03 | Boehringer Ingelheim International Gmbh | Use of ccr3-inhibitors |
| US10213421B2 (en) * | 2012-04-04 | 2019-02-26 | Alkahest, Inc. | Pharmaceutical formulations comprising CCR3 antagonists |
-
2013
- 2013-03-27 US US13/851,538 patent/US10213421B2/en active Active
- 2013-04-02 ES ES21190323T patent/ES3044310T3/es active Active
- 2013-04-02 ES ES13714618T patent/ES2715844T3/es active Active
- 2013-04-02 NZ NZ628993A patent/NZ628993A/en unknown
- 2013-04-02 ES ES18213458T patent/ES2898179T3/es active Active
- 2013-04-02 PL PL18213458T patent/PL3524230T3/pl unknown
- 2013-04-02 EP EP13714618.9A patent/EP2833864B1/en active Active
- 2013-04-02 IN IN7082DEN2014 patent/IN2014DN07082A/en unknown
- 2013-04-02 DK DK18213458.5T patent/DK3524230T3/da active
- 2013-04-02 EA EA201401082A patent/EA027627B1/ru not_active IP Right Cessation
- 2013-04-02 HU HUE13714618A patent/HUE041519T2/hu unknown
- 2013-04-02 AU AU2013245028A patent/AU2013245028B2/en active Active
- 2013-04-02 TR TR2018/21285T patent/TR201821285T4/tr unknown
- 2013-04-02 KR KR1020207021307A patent/KR102338465B1/ko active Active
- 2013-04-02 RS RS20190050A patent/RS58360B1/sr unknown
- 2013-04-02 CN CN201380016781.7A patent/CN104203213A/zh active Pending
- 2013-04-02 JP JP2015503848A patent/JP6320990B2/ja active Active
- 2013-04-02 LT LTEP13714618.9T patent/LT2833864T/lt unknown
- 2013-04-02 PT PT13714618T patent/PT2833864T/pt unknown
- 2013-04-02 CA CA2869058A patent/CA2869058C/en active Active
- 2013-04-02 DK DK13714618.9T patent/DK2833864T3/en active
- 2013-04-02 MX MX2014011787A patent/MX358307B/es active IP Right Grant
- 2013-04-02 HR HRP20190069TT patent/HRP20190069T1/hr unknown
- 2013-04-02 PL PL13714618T patent/PL2833864T3/pl unknown
- 2013-04-02 HU HUE18213458A patent/HUE056943T2/hu unknown
- 2013-04-02 BR BR112014024479A patent/BR112014024479A8/pt not_active Application Discontinuation
- 2013-04-02 SI SI201331330T patent/SI2833864T1/sl unknown
- 2013-04-02 KR KR1020147027802A patent/KR102138709B1/ko active Active
- 2013-04-02 EP EP18213458.5A patent/EP3524230B1/en active Active
- 2013-04-02 WO PCT/EP2013/056867 patent/WO2013149987A1/en not_active Ceased
- 2013-04-02 SM SM20190121T patent/SMT201900121T1/it unknown
- 2013-04-02 PT PT182134585T patent/PT3524230T/pt unknown
- 2013-04-02 EP EP21190323.2A patent/EP3970693B1/en active Active
- 2013-04-03 TW TW102112244A patent/TW201400115A/zh unknown
- 2013-04-03 AR ARP130101093A patent/AR090596A1/es unknown
- 2013-04-04 UY UY0001034730A patent/UY34730A/es unknown
-
2014
- 2014-08-26 IL IL234299A patent/IL234299A/en active IP Right Grant
- 2014-09-24 CL CL2014002524A patent/CL2014002524A1/es unknown
- 2014-10-03 PH PH12014502241A patent/PH12014502241A1/en unknown
-
2018
- 2018-04-04 JP JP2018072309A patent/JP6700332B2/ja active Active
- 2018-12-28 US US16/235,905 patent/US20190151300A1/en not_active Abandoned
-
2019
- 2019-01-17 CY CY20191100062T patent/CY1121137T1/el unknown
-
2020
- 2020-04-29 US US16/861,473 patent/US11612596B2/en active Active
- 2020-04-30 JP JP2020080024A patent/JP2020143080A/ja active Pending
-
2022
- 2022-02-24 JP JP2022026735A patent/JP2022081524A/ja active Pending
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