JP2015512433A5 - - Google Patents

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Publication number
JP2015512433A5
JP2015512433A5 JP2015503848A JP2015503848A JP2015512433A5 JP 2015512433 A5 JP2015512433 A5 JP 2015512433A5 JP 2015503848 A JP2015503848 A JP 2015503848A JP 2015503848 A JP2015503848 A JP 2015503848A JP 2015512433 A5 JP2015512433 A5 JP 2015512433A5
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Japan
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pharmaceutical composition
composition according
weight
disintegrant
diluent
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JP2015503848A
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English (en)
Japanese (ja)
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JP2015512433A (ja
JP6320990B2 (ja
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Priority claimed from PCT/EP2013/056867 external-priority patent/WO2013149987A1/en
Publication of JP2015512433A publication Critical patent/JP2015512433A/ja
Publication of JP2015512433A5 publication Critical patent/JP2015512433A5/ja
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Publication of JP6320990B2 publication Critical patent/JP6320990B2/ja
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JP2015503848A 2012-04-04 2013-04-02 Ｃｃｒ３アンタゴニストを含む医薬製剤 Active JP6320990B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12163078.4 2012-04-04
EP12163078 2012-04-04
PCT/EP2013/056867 WO2013149987A1 (en) 2012-04-04 2013-04-02 Pharmaceutical formulations comprising ccr3 antagonists

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2018072309A Division JP6700332B2 (ja) 2012-04-04 2018-04-04 Ｃｃｒ３アンタゴニストを含む医薬製剤

Publications (3)

Publication Number Publication Date
JP2015512433A JP2015512433A (ja) 2015-04-27
JP2015512433A5 true JP2015512433A5 (enExample) 2016-06-02
JP6320990B2 JP6320990B2 (ja) 2018-05-09

Family

ID=49292482

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2015503848A Active JP6320990B2 (ja) 2012-04-04 2013-04-02 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2018072309A Active JP6700332B2 (ja) 2012-04-04 2018-04-04 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2020080024A Pending JP2020143080A (ja) 2012-04-04 2020-04-30 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2022026735A Pending JP2022081524A (ja) 2012-04-04 2022-02-24 Ｃｃｒ３アンタゴニストを含む医薬製剤

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP2018072309A Active JP6700332B2 (ja) 2012-04-04 2018-04-04 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2020080024A Pending JP2020143080A (ja) 2012-04-04 2020-04-30 Ｃｃｒ３アンタゴニストを含む医薬製剤
JP2022026735A Pending JP2022081524A (ja) 2012-04-04 2022-02-24 Ｃｃｒ３アンタゴニストを含む医薬製剤

Country Status (31)

Country Link
US (3) US10213421B2 (enExample)
EP (3) EP2833864B1 (enExample)
JP (4) JP6320990B2 (enExample)
KR (2) KR102338465B1 (enExample)
CN (1) CN104203213A (enExample)
AR (1) AR090596A1 (enExample)
AU (1) AU2013245028B2 (enExample)
BR (1) BR112014024479A8 (enExample)
CA (1) CA2869058C (enExample)
CL (1) CL2014002524A1 (enExample)
CY (1) CY1121137T1 (enExample)
DK (2) DK2833864T3 (enExample)
EA (1) EA027627B1 (enExample)
ES (3) ES3044310T3 (enExample)
HR (1) HRP20190069T1 (enExample)
HU (2) HUE056943T2 (enExample)
IL (1) IL234299A (enExample)
IN (1) IN2014DN07082A (enExample)
LT (1) LT2833864T (enExample)
MX (1) MX358307B (enExample)
NZ (1) NZ628993A (enExample)
PH (1) PH12014502241A1 (enExample)
PL (2) PL3524230T3 (enExample)
PT (2) PT3524230T (enExample)
RS (1) RS58360B1 (enExample)
SI (1) SI2833864T1 (enExample)
SM (1) SMT201900121T1 (enExample)
TR (1) TR201821285T4 (enExample)
TW (1) TW201400115A (enExample)
UY (1) UY34730A (enExample)
WO (1) WO2013149987A1 (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
MY199462A (en) * 2017-04-05 2023-10-30 Alkahest Inc Methods and compositions for treating retina-associated disease using ccr3-inhibitors
CN110636844A (zh) 2017-04-05 2019-12-31 万能溶剂有限公司 使用ccr3-抑制剂治疗衰老相关损伤的方法及组合物
CN111343983A (zh) * 2017-10-13 2020-06-26 万能溶剂有限公司 使用ccr3抑制剂治疗瘙痒、干燥症和相关疾病的方法和组合物
MY198220A (en) 2018-05-15 2023-08-14 Alkahest Inc Treatment Of Aging-Associated Disease With Modulators Of Leukotriene A4 Hydrolase
KR20210065950A (ko) * 2018-09-26 2021-06-04 알카헤스트 인코포레이티드 Ccr3-억제제를 사용한 노화 관련 장애 치료를 위한 방법 및 조성물
US20230312697A1 (en) 2020-06-11 2023-10-05 Alkahest Inc. Methods of improving retina-associated disease outcome using ccr3-inhibitors
KR20230056017A (ko) 2020-08-27 2023-04-26 에이지씨 가부시키가이샤 무알칼리 유리 및 유리판
AU2022376563A1 (en) 2021-11-01 2023-12-07 Alkahest, Inc. Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases

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CA2318088A1 (en) 1998-01-21 1999-07-29 Yoshisuke Nakasato Chemokine receptor antagonists and methods of use therefor
US6140349A (en) 1998-02-02 2000-10-31 Merck & Co., Inc. Cyclic amine modulators of chemokine receptor activity
JP2002501898A (ja) 1998-02-02 2002-01-22 メルク エンド カムパニー インコーポレーテッド ケモカイン受容体活性の環状アミン調節剤
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RU2382037C2 (ru) 2003-11-17 2010-02-20 Бёрингер Ингельхайм Интернациональ Гмбх Новые пиперидинзамещенные индолы или их гетеропроизводные
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EP2079725B1 (en) 2006-10-27 2011-12-14 Boehringer Ingelheim International GmbH Piperidyl-propane-thiol ccr3 modulators
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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
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MX2011011080A (es) 2009-04-22 2012-02-23 Axikin Pharmaceuticals Inc Antagonistas de ccr3 de arilsulfonamida 2, 5-disustituida.
EP2523654A4 (en) * 2010-01-11 2014-08-06 Mohamed Shafee Muneera IMMEDIATE RELEASE COMPOSITIONS OF MEDICAMENTS LABILES ACIDES
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists

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