IN2014DN07082A - - Google Patents

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Publication number
IN2014DN07082A
IN2014DN07082A IN7082DEN2014A IN2014DN07082A IN 2014DN07082 A IN2014DN07082 A IN 2014DN07082A IN 7082DEN2014 A IN7082DEN2014 A IN 7082DEN2014A IN 2014DN07082 A IN2014DN07082 A IN 2014DN07082A
Authority
IN
India
Prior art keywords
alkyl
dibenzoyltartrate
haloalkyl
cycloalkyl
chloride
Prior art date
Application number
Other languages
English (en)
Inventor
Alfred Fetscher
Jochen Matthias Scher
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014DN07082(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of IN2014DN07082A publication Critical patent/IN2014DN07082A/en

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Classifications

    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
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Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IN7082DEN2014 2012-04-04 2013-04-02 IN2014DN07082A (enExample)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04
PCT/EP2013/056867 WO2013149987A1 (en) 2012-04-04 2013-04-02 Pharmaceutical formulations comprising ccr3 antagonists

Publications (1)

Publication Number Publication Date
IN2014DN07082A true IN2014DN07082A (enExample) 2015-04-10

Family

ID=49292482

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7082DEN2014 IN2014DN07082A (enExample) 2012-04-04 2013-04-02

Country Status (31)

Country Link
US (3) US10213421B2 (enExample)
EP (3) EP3970693B1 (enExample)
JP (4) JP6320990B2 (enExample)
KR (2) KR102338465B1 (enExample)
CN (1) CN104203213A (enExample)
AR (1) AR090596A1 (enExample)
AU (1) AU2013245028B2 (enExample)
BR (1) BR112014024479A8 (enExample)
CA (1) CA2869058C (enExample)
CL (1) CL2014002524A1 (enExample)
CY (1) CY1121137T1 (enExample)
DK (2) DK2833864T3 (enExample)
EA (1) EA027627B1 (enExample)
ES (3) ES3044310T3 (enExample)
HR (1) HRP20190069T1 (enExample)
HU (2) HUE056943T2 (enExample)
IL (1) IL234299A (enExample)
IN (1) IN2014DN07082A (enExample)
LT (1) LT2833864T (enExample)
MX (1) MX358307B (enExample)
NZ (1) NZ628993A (enExample)
PH (1) PH12014502241A1 (enExample)
PL (2) PL3524230T3 (enExample)
PT (2) PT3524230T (enExample)
RS (1) RS58360B1 (enExample)
SI (1) SI2833864T1 (enExample)
SM (1) SMT201900121T1 (enExample)
TR (1) TR201821285T4 (enExample)
TW (1) TW201400115A (enExample)
UY (1) UY34730A (enExample)
WO (1) WO2013149987A1 (enExample)

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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
US11382907B2 (en) * 2017-04-05 2022-07-12 Alkahest, Inc. Methods and compositions for treating aging-associated impairments using CCR3-inhibitors
EA201992356A1 (ru) * 2017-04-05 2020-03-23 Алкахест Инк. Способ и композиция для лечения заболевания, связанного с сетчаткой глаза, с использованием ингибитора ccr3
CA3076017A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. Methods and compositions for treating pruritus, xerosis, and associated disease using ccr3-inhibitors
US11426399B2 (en) 2018-05-15 2022-08-30 Alkahest, Inc. Treatment of aging-associated disease with modulators of leukotriene A4 hydrolase
EP3856195A4 (en) * 2018-09-26 2022-06-22 Alkahest, Inc. METHODS AND COMPOSITIONS FOR TREATMENT OF AGING-RELATED DISORDERS USING CCR3 INHIBITORS
US12692301B2 (en) 2020-06-11 2026-07-28 Alkahest Inc. Methods of improving retina-associated disease outcome using CCR3-inhibitors
WO2022045226A1 (ja) 2020-08-27 2022-03-03 Ａｇｃ株式会社 無アルカリガラスおよびガラス板
CA3221177A1 (en) 2021-11-01 2023-05-04 Meghan Kerrisk Campbell Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases

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