HUE041519T2 - CCR3 antagonistákat tartalmazó gyógyászati készítmények - Google Patents

CCR3 antagonistákat tartalmazó gyógyászati készítmények

Info

Publication number
HUE041519T2
HUE041519T2 HUE13714618A HUE13714618A HUE041519T2 HU E041519 T2 HUE041519 T2 HU E041519T2 HU E13714618 A HUE13714618 A HU E13714618A HU E13714618 A HUE13714618 A HU E13714618A HU E041519 T2 HUE041519 T2 HU E041519T2
Authority
HU
Hungary
Prior art keywords
pharmaceutical formulations
ccr3 antagonists
ccr3
antagonists
formulations
Prior art date
Application number
HUE13714618A
Other languages
English (en)
Hungarian (hu)
Inventor
Alfred Fetscher
Jochen Matthias Scher
Original Assignee
Alkahest Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUE041519(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alkahest Inc filed Critical Alkahest Inc
Publication of HUE041519T2 publication Critical patent/HUE041519T2/hu

Links

Classifications

    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
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    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
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    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
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    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Otolaryngology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HUE13714618A 2012-04-04 2013-04-02 CCR3 antagonistákat tartalmazó gyógyászati készítmények HUE041519T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04

Publications (1)

Publication Number Publication Date
HUE041519T2 true HUE041519T2 (hu) 2019-05-28

Family

ID=49292482

Family Applications (2)

Application Number Title Priority Date Filing Date
HUE18213458A HUE056943T2 (hu) 2012-04-04 2013-04-02 CCR3 antagonistákat tartalmazó gyógyászati készítmények
HUE13714618A HUE041519T2 (hu) 2012-04-04 2013-04-02 CCR3 antagonistákat tartalmazó gyógyászati készítmények

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HUE18213458A HUE056943T2 (hu) 2012-04-04 2013-04-02 CCR3 antagonistákat tartalmazó gyógyászati készítmények

Country Status (31)

Country Link
US (3) US10213421B2 (enExample)
EP (3) EP2833864B1 (enExample)
JP (4) JP6320990B2 (enExample)
KR (2) KR102138709B1 (enExample)
CN (1) CN104203213A (enExample)
AR (1) AR090596A1 (enExample)
AU (1) AU2013245028B2 (enExample)
BR (1) BR112014024479A8 (enExample)
CA (1) CA2869058C (enExample)
CL (1) CL2014002524A1 (enExample)
CY (1) CY1121137T1 (enExample)
DK (2) DK2833864T3 (enExample)
EA (1) EA027627B1 (enExample)
ES (3) ES2898179T3 (enExample)
HR (1) HRP20190069T1 (enExample)
HU (2) HUE056943T2 (enExample)
IL (1) IL234299A (enExample)
IN (1) IN2014DN07082A (enExample)
LT (1) LT2833864T (enExample)
MX (1) MX358307B (enExample)
NZ (1) NZ628993A (enExample)
PH (1) PH12014502241A1 (enExample)
PL (2) PL3524230T3 (enExample)
PT (2) PT2833864T (enExample)
RS (1) RS58360B1 (enExample)
SI (1) SI2833864T1 (enExample)
SM (1) SMT201900121T1 (enExample)
TR (1) TR201821285T4 (enExample)
TW (1) TW201400115A (enExample)
UY (1) UY34730A (enExample)
WO (1) WO2013149987A1 (enExample)

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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
AU2018250214B2 (en) * 2017-04-05 2021-09-16 Alkahest, Inc. Methods and compositions for treating aging-associated impairments using CCR3-inhibitors
ES3046717T3 (en) 2017-04-05 2025-12-02 Alkahest Inc Compounds and pharmaceutical compositions for use in treating retina-associated disease using ccr3-inhibitors
EP3694514A4 (en) * 2017-10-13 2021-07-07 Alkahest, Inc. METHODS AND COMPOSITIONS FOR TREATING PRURITUS, XEROSIS AND ASSOCIATED ILLNESS USING CCR3 INHIBITORS
JP2021529156A (ja) 2018-05-15 2021-10-28 アルカヘスト,インコーポレイテッド ロイコトリエンa4ヒドロラーゼの調節剤を用いた老化関連疾患の治療
BR112021004938A2 (pt) * 2018-09-26 2021-06-01 Alkahest, Inc. métodos e composições para tratamento de danos associados com o envelhecimento usando inibidores de ccr3
EP4206153A4 (en) 2020-08-27 2024-05-15 Agc Inc. ALKALI-FREE GLASS AND PLATE GLASS
JP2024542963A (ja) 2021-11-01 2024-11-19 アルカヘスト,インコーポレイテッド 加齢関連疾患の予防及び治療のためのロイコトリエンa4加水分解酵素(lta4h)のベンゾジオキサン調節剤

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BRPI0415767A (pt) 2003-10-24 2006-12-26 Hoffmann La Roche antagonistas de receptor de ccr-3
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