JP2015503609A5 - - Google Patents

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Publication number
JP2015503609A5
JP2015503609A5 JP2014551714A JP2014551714A JP2015503609A5 JP 2015503609 A5 JP2015503609 A5 JP 2015503609A5 JP 2014551714 A JP2014551714 A JP 2014551714A JP 2014551714 A JP2014551714 A JP 2014551714A JP 2015503609 A5 JP2015503609 A5 JP 2015503609A5
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JP
Japan
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alkyl
optionally substituted
alkoxy
halogen
aryl
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JP2014551714A
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Japanese (ja)
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JP2015503609A (ja
JP6073923B2 (ja
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Priority claimed from PCT/IB2013/050271 external-priority patent/WO2013105057A1/en
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Publication of JP2015503609A5 publication Critical patent/JP2015503609A5/ja
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Publication of JP6073923B2 publication Critical patent/JP6073923B2/ja
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JP2014551714A 2012-01-13 2013-01-11 肺動脈高血圧症（ｐａｈ）および関連障害の治療のためのｉｐ受容体アゴニストとしての縮合ピロール Expired - Fee Related JP6073923B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261586546P 2012-01-13 2012-01-13
US61/586,546 2012-01-13
PCT/IB2013/050271 WO2013105057A1 (en) 2012-01-13 2013-01-11 Fused pyrroles as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders

Publications (3)

Publication Number Publication Date
JP2015503609A JP2015503609A (ja) 2015-02-02
JP2015503609A5 true JP2015503609A5 (enExample) 2016-02-18
JP6073923B2 JP6073923B2 (ja) 2017-02-01

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JP2014551714A Expired - Fee Related JP6073923B2 (ja) 2012-01-13 2013-01-11 肺動脈高血圧症（ｐａｈ）および関連障害の治療のためのｉｐ受容体アゴニストとしての縮合ピロール

Country Status (9)

Country Link
US (2) US8937069B2 (enExample)
EP (1) EP2802589B1 (enExample)
JP (1) JP6073923B2 (enExample)
CN (1) CN104053659B (enExample)
AR (1) AR089698A1 (enExample)
ES (1) ES2565826T3 (enExample)
TW (1) TW201335160A (enExample)
UY (1) UY34572A (enExample)
WO (1) WO2013105057A1 (enExample)

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ES2637719T3 (es) 2013-02-13 2017-10-16 Novartis Ag Compuestos heterocíclicos agonistas del receptor IP
UA119247C2 (uk) 2013-09-06 2019-05-27 РОЙВЕНТ САЙЕНСИЗ ҐмбГ Спіроциклічні сполуки як інгібітори триптофангідроксилази
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BR112013000946B1 (pt) 2010-07-14 2020-09-08 Novartis Ag Compostos heterocíclicos agonistas de receptor de ip, seus usos, composição e combinação farmacêuticas
US9174985B2 (en) 2012-01-13 2015-11-03 Novartis Ag Salts of 7-(2,3-di-p-tolyl-7,8-dihydropyrido[2,3-b]pyrazin-5(6H)-yl)heptanoic acid as IP receptor agonists
EP2802582A1 (en) 2012-01-13 2014-11-19 Novartis AG Fused dihydropyrido [2,3 -b]pyrazines as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders
EP2802583A1 (en) 2012-01-13 2014-11-19 Novartis AG Fused piperidines as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders
US9115129B2 (en) 2012-01-13 2015-08-25 Novartis Ag Substituted pyrido[2,3-B]pyrazines as IP receptor agonists
WO2013105058A1 (en) 2012-01-13 2013-07-18 Novartis Ag 7,8- dihydropyrido [3, 4 - b] pyrazines as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders
AR089698A1 (es) 2012-01-13 2014-09-10 Novartis Ag Compuestos heterociclicos antagonistas del receptor ip

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