MXPA05009688A - Derivados de naftiridina como agentes antibacterianos. - Google Patents

Derivados de naftiridina como agentes antibacterianos.

Info

Publication number
MXPA05009688A
MXPA05009688A MXPA05009688A MXPA05009688A MXPA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A
Authority
MX
Mexico
Prior art keywords
antibacterial agents
naphthyridine derivatives
compounds
prodrugs
salts
Prior art date
Application number
MXPA05009688A
Other languages
English (en)
Inventor
Zhang Tianyuan
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Priority claimed from US10/387,318 external-priority patent/US8163769B2/en
Publication of MXPA05009688A publication Critical patent/MXPA05009688A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Se describen agentes antibacterianos que tienen la formula (I) y sus sales, profarmacos y las sales de sus profarmacos; proceso para preparar los compuestos, e intermediarios usados en los procesos; composiciones que contienen los compuestos y metodos de profilaxis y tratamiento de infecciones bacterianas, utilizando los compuestos.
MXPA05009688A 2003-03-12 2003-03-12 Derivados de naftiridina como agentes antibacterianos. MXPA05009688A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/387,318 US8163769B2 (en) 2002-03-12 2003-03-12 Antibacterial compounds
PCT/US2003/007689 WO2004083207A1 (en) 2003-03-12 2003-03-12 Naphthyridine derivatives as antibacterial agents

Publications (1)

Publication Number Publication Date
MXPA05009688A true MXPA05009688A (es) 2005-12-05

Family

ID=33029637

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05009688A MXPA05009688A (es) 2003-03-12 2003-03-12 Derivados de naftiridina como agentes antibacterianos.

Country Status (5)

Country Link
EP (1) EP1631570A1 (es)
JP (1) JP2006514964A (es)
CA (1) CA2518443A1 (es)
MX (1) MXPA05009688A (es)
WO (1) WO2004083207A1 (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005026165A1 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Quinolone antibacterial agents
CA2629461C (en) * 2005-11-10 2016-01-12 Anita Melikian Substituted quinolones and methods of use
WO2008046135A1 (en) 2006-10-16 2008-04-24 Bionomics Limited Novel anxiolytic compounds
US10954231B2 (en) 2006-10-16 2021-03-23 Bionomics Limited Anxiolytic compounds
EP1972338A1 (en) 2007-03-19 2008-09-24 Technische Universität Carolo-Wilhelmina zu Braunschweig Anti-infective agents
FR2928150A1 (fr) * 2008-02-29 2009-09-04 Vetoquinol Sa Sa Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens
TW201028378A (en) * 2008-11-26 2010-08-01 Abbott Lab Novel substituted octahydrocyclopenta[c]pyrrol-4-amines as calcium channel blockers
CN102140098A (zh) * 2010-01-29 2011-08-03 南京医科大学 7-(2-取代-3-氨基-1-四氢吡咯[3,4-c]吡唑基)喹啉羧酸衍生物及其制备方法和在抗菌抗结核上的应用
ES2622519T3 (es) 2010-07-14 2017-07-06 Novartis Ag Componentes heterocíclicos agonistas del receptor IP
CN103502219A (zh) 2011-03-02 2014-01-08 生态学有限公司 作为治疗剂的新型小分子
JP6055817B2 (ja) 2011-05-12 2016-12-27 バイオノミックス リミテッド ナフチリジンの調製方法
AR089698A1 (es) 2012-01-13 2014-09-10 Novartis Ag Compuestos heterociclicos antagonistas del receptor ip
GB201206384D0 (en) * 2012-04-11 2012-05-23 Redx Pharma Ltd Antibacterial drug derivatives
JP2016507582A (ja) 2013-02-13 2016-03-10 ノバルティス アーゲー Ip受容体アゴニスト複素環式化合物
CA3061877A1 (en) 2017-03-24 2019-10-29 Wakunaga Pharmaceutical Co., Ltd. Novel pyridone carboxylic acid derivative or salt thereof

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3873554A (en) * 1973-03-06 1975-03-25 Sterling Drug Inc Preparation of 1-alkyl-1,4-dihydro-7-substituted-4-oxo-1,8-naphthyridine-3-carboxylic acids via the 3-carboxaldehyde analogs
US3857851A (en) * 1973-03-06 1974-12-31 Sterling Drug Inc 1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxaldehydes
JPS5925391A (ja) * 1982-07-30 1984-02-09 Dainippon Pharmaceut Co Ltd ピリジルナフチリジン誘導体およびその塩
US4954507A (en) * 1986-10-08 1990-09-04 Bristol-Myers Company 1-tertiary-alkyl-substituted naphthyridine carboxylic acid antibacterial agents
DE3816119A1 (de) * 1988-05-11 1989-11-23 Bayer Ag 7-substituierte chinolon- und naphthyridoncarbonsaeure-derivate
JPH04502317A (ja) * 1988-12-06 1992-04-23 ジ・アップジョン・カンパニー 抗菌性キノロン化合物
US5137892A (en) * 1990-12-12 1992-08-11 Abbott Laboratories Quinoline, naphthyridine and pyridobenzoxazine derivatives
DE4435479A1 (de) * 1994-10-04 1996-04-11 Bayer Ag Chinolon- und Naphthyridoncarbonsäure-Derivate
AR030537A1 (es) * 1999-11-05 2003-08-27 Abbott Lab Acidos quinolincarboxilicos y naftiridincarboxilico antibacterianos
SE9904108D0 (sv) * 1999-11-15 1999-11-15 New Pharma Research Ab Nya föreningar
US6964966B2 (en) * 2001-04-25 2005-11-15 Wockhardt Limited Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments

Also Published As

Publication number Publication date
CA2518443A1 (en) 2004-09-30
JP2006514964A (ja) 2006-05-18
WO2004083207A1 (en) 2004-09-30
EP1631570A1 (en) 2006-03-08

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Legal Events

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