MXPA05009688A - Derivados de naftiridina como agentes antibacterianos. - Google Patents
Derivados de naftiridina como agentes antibacterianos.Info
- Publication number
- MXPA05009688A MXPA05009688A MXPA05009688A MXPA05009688A MXPA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A MX PA05009688 A MXPA05009688 A MX PA05009688A
- Authority
- MX
- Mexico
- Prior art keywords
- antibacterial agents
- naphthyridine derivatives
- compounds
- prodrugs
- salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Se describen agentes antibacterianos que tienen la formula (I) y sus sales, profarmacos y las sales de sus profarmacos; proceso para preparar los compuestos, e intermediarios usados en los procesos; composiciones que contienen los compuestos y metodos de profilaxis y tratamiento de infecciones bacterianas, utilizando los compuestos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/387,318 US8163769B2 (en) | 2002-03-12 | 2003-03-12 | Antibacterial compounds |
PCT/US2003/007689 WO2004083207A1 (en) | 2003-03-12 | 2003-03-12 | Naphthyridine derivatives as antibacterial agents |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA05009688A true MXPA05009688A (es) | 2005-12-05 |
Family
ID=33029637
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA05009688A MXPA05009688A (es) | 2003-03-12 | 2003-03-12 | Derivados de naftiridina como agentes antibacterianos. |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP1631570A1 (es) |
JP (1) | JP2006514964A (es) |
CA (1) | CA2518443A1 (es) |
MX (1) | MXPA05009688A (es) |
WO (1) | WO2004083207A1 (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2005026165A1 (en) * | 2003-09-12 | 2005-03-24 | Warner-Lambert Company Llc | Quinolone antibacterial agents |
CA2629461C (en) * | 2005-11-10 | 2016-01-12 | Anita Melikian | Substituted quinolones and methods of use |
WO2008046135A1 (en) | 2006-10-16 | 2008-04-24 | Bionomics Limited | Novel anxiolytic compounds |
US10954231B2 (en) | 2006-10-16 | 2021-03-23 | Bionomics Limited | Anxiolytic compounds |
EP1972338A1 (en) | 2007-03-19 | 2008-09-24 | Technische Universität Carolo-Wilhelmina zu Braunschweig | Anti-infective agents |
FR2928150A1 (fr) * | 2008-02-29 | 2009-09-04 | Vetoquinol Sa Sa | Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens |
TW201028378A (en) * | 2008-11-26 | 2010-08-01 | Abbott Lab | Novel substituted octahydrocyclopenta[c]pyrrol-4-amines as calcium channel blockers |
CN102140098A (zh) * | 2010-01-29 | 2011-08-03 | 南京医科大学 | 7-(2-取代-3-氨基-1-四氢吡咯[3,4-c]吡唑基)喹啉羧酸衍生物及其制备方法和在抗菌抗结核上的应用 |
ES2622519T3 (es) | 2010-07-14 | 2017-07-06 | Novartis Ag | Componentes heterocíclicos agonistas del receptor IP |
CN103502219A (zh) | 2011-03-02 | 2014-01-08 | 生态学有限公司 | 作为治疗剂的新型小分子 |
JP6055817B2 (ja) | 2011-05-12 | 2016-12-27 | バイオノミックス リミテッド | ナフチリジンの調製方法 |
AR089698A1 (es) | 2012-01-13 | 2014-09-10 | Novartis Ag | Compuestos heterociclicos antagonistas del receptor ip |
GB201206384D0 (en) * | 2012-04-11 | 2012-05-23 | Redx Pharma Ltd | Antibacterial drug derivatives |
JP2016507582A (ja) | 2013-02-13 | 2016-03-10 | ノバルティス アーゲー | Ip受容体アゴニスト複素環式化合物 |
CA3061877A1 (en) | 2017-03-24 | 2019-10-29 | Wakunaga Pharmaceutical Co., Ltd. | Novel pyridone carboxylic acid derivative or salt thereof |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3873554A (en) * | 1973-03-06 | 1975-03-25 | Sterling Drug Inc | Preparation of 1-alkyl-1,4-dihydro-7-substituted-4-oxo-1,8-naphthyridine-3-carboxylic acids via the 3-carboxaldehyde analogs |
US3857851A (en) * | 1973-03-06 | 1974-12-31 | Sterling Drug Inc | 1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxaldehydes |
JPS5925391A (ja) * | 1982-07-30 | 1984-02-09 | Dainippon Pharmaceut Co Ltd | ピリジルナフチリジン誘導体およびその塩 |
US4954507A (en) * | 1986-10-08 | 1990-09-04 | Bristol-Myers Company | 1-tertiary-alkyl-substituted naphthyridine carboxylic acid antibacterial agents |
DE3816119A1 (de) * | 1988-05-11 | 1989-11-23 | Bayer Ag | 7-substituierte chinolon- und naphthyridoncarbonsaeure-derivate |
JPH04502317A (ja) * | 1988-12-06 | 1992-04-23 | ジ・アップジョン・カンパニー | 抗菌性キノロン化合物 |
US5137892A (en) * | 1990-12-12 | 1992-08-11 | Abbott Laboratories | Quinoline, naphthyridine and pyridobenzoxazine derivatives |
DE4435479A1 (de) * | 1994-10-04 | 1996-04-11 | Bayer Ag | Chinolon- und Naphthyridoncarbonsäure-Derivate |
AR030537A1 (es) * | 1999-11-05 | 2003-08-27 | Abbott Lab | Acidos quinolincarboxilicos y naftiridincarboxilico antibacterianos |
SE9904108D0 (sv) * | 1999-11-15 | 1999-11-15 | New Pharma Research Ab | Nya föreningar |
US6964966B2 (en) * | 2001-04-25 | 2005-11-15 | Wockhardt Limited | Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
-
2003
- 2003-03-12 MX MXPA05009688A patent/MXPA05009688A/es not_active Application Discontinuation
- 2003-03-12 JP JP2004569641A patent/JP2006514964A/ja active Pending
- 2003-03-12 EP EP03723732A patent/EP1631570A1/en not_active Withdrawn
- 2003-03-12 WO PCT/US2003/007689 patent/WO2004083207A1/en active Application Filing
- 2003-03-12 CA CA002518443A patent/CA2518443A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2518443A1 (en) | 2004-09-30 |
JP2006514964A (ja) | 2006-05-18 |
WO2004083207A1 (en) | 2004-09-30 |
EP1631570A1 (en) | 2006-03-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |