SE9904108D0 - Nya föreningar - Google Patents
Nya föreningarInfo
- Publication number
- SE9904108D0 SE9904108D0 SE9904108A SE9904108A SE9904108D0 SE 9904108 D0 SE9904108 D0 SE 9904108D0 SE 9904108 A SE9904108 A SE 9904108A SE 9904108 A SE9904108 A SE 9904108A SE 9904108 D0 SE9904108 D0 SE 9904108D0
- Authority
- SE
- Sweden
- Prior art keywords
- sub
- new compounds
- treatment
- antibacterial
- antiparasitic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Priority Applications (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE9904108A SE9904108D0 (sv) | 1999-11-15 | 1999-11-15 | Nya föreningar |
US10/111,898 US6967205B1 (en) | 1999-11-15 | 2000-11-13 | Compounds with antibacterial and antiparasitic properties |
JP2001538897A JP2003514812A (ja) | 1999-11-15 | 2000-11-13 | 抗菌性および抗寄生虫性を有する化合物 |
AT00980176T ATE398117T1 (de) | 1999-11-15 | 2000-11-13 | Verbindungen mit antibakteriellen und antiparasitischen eigenschaften |
EP00980176A EP1230235B1 (en) | 1999-11-15 | 2000-11-13 | Compounds with antibacterial and antiparasitic properties |
AU17472/01A AU1747201A (en) | 1999-11-15 | 2000-11-13 | Compounds with antibacterial and antiparasitic properties |
PCT/SE2000/002217 WO2001036408A1 (en) | 1999-11-15 | 2000-11-13 | Compounds with antibacterial and antiparasitic properties |
DE60039183T DE60039183D1 (de) | 1999-11-15 | 2000-11-13 | Verbindungen mit antibakteriellen und antiparasitischen eigenschaften |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE9904108A SE9904108D0 (sv) | 1999-11-15 | 1999-11-15 | Nya föreningar |
Publications (1)
Publication Number | Publication Date |
---|---|
SE9904108D0 true SE9904108D0 (sv) | 1999-11-15 |
Family
ID=20417705
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE9904108A SE9904108D0 (sv) | 1999-11-15 | 1999-11-15 | Nya föreningar |
Country Status (8)
Country | Link |
---|---|
US (1) | US6967205B1 (sv) |
EP (1) | EP1230235B1 (sv) |
JP (1) | JP2003514812A (sv) |
AT (1) | ATE398117T1 (sv) |
AU (1) | AU1747201A (sv) |
DE (1) | DE60039183D1 (sv) |
SE (1) | SE9904108D0 (sv) |
WO (1) | WO2001036408A1 (sv) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8163769B2 (en) | 2002-03-12 | 2012-04-24 | Abbott Laboratories | Antibacterial compounds |
GB0215775D0 (en) * | 2002-07-06 | 2002-08-14 | Astex Technology Ltd | Pharmaceutical compounds |
EP1559321A1 (en) * | 2002-10-11 | 2005-08-03 | Meiji Seika Kaisha Ltd. | Mixed compositions for controlling parasitic insects |
CA2518443A1 (en) * | 2003-03-12 | 2004-09-30 | Abbott Laboratories | Naphthyridine derivatives as antibacterial agents |
PT1666477E (pt) | 2003-09-10 | 2013-08-28 | Kyorin Seiyaku Kk | Derivado de 7-(4-substituído-3-ciclopropilaminometil-1- pirrolidinil) quinolonecarboxílico |
US20050124625A1 (en) * | 2003-10-21 | 2005-06-09 | Salvati Mark E. | Piperazine derivatives and their use as modulators of nuclear hormone receptor function |
US7498341B2 (en) * | 2004-01-31 | 2009-03-03 | Sanofi Aventis Deutschland Gmbh | Heterocyclically substituted 7-amino-4-quinolone-3-carboxylic acid derivatives, process for their preparation and their use as medicaments |
WO2005097752A1 (en) * | 2004-03-31 | 2005-10-20 | Bayer Pharmaceuticals Corporation | Quinolone carboxylic acid derivatives for treatment of hyperproliferative conditions |
AU2006326540A1 (en) | 2005-12-14 | 2007-06-21 | Amgen Inc. | Diaza heterocyclic sulfonamide derivatives and their uses |
PT2383271E (pt) * | 2006-03-13 | 2013-10-10 | Kyorin Seiyaku Kk | Aminoquinolonas como inibidores de gsk-3 |
EP2149571A4 (en) * | 2007-05-24 | 2010-09-01 | Kyorin Seiyaku Kk | MUTILINE DERIVATIVE WITH A RINGED, HETEROCYCLIC AND AROMATIC CARBOXYLIC ACID STRUCTURE IN A SUBSTITUTE AT POSITION 14 |
US7902227B2 (en) | 2007-07-27 | 2011-03-08 | Janssen Pharmaceutica Nv. | C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents |
US8389514B2 (en) * | 2007-09-11 | 2013-03-05 | Kyorin Pharmaceutical Co., Ltd. | Cyanoaminoquinolones and tetrazoloaminoquinolones as GSK-3 inhibitors |
CN101855229A (zh) | 2007-09-12 | 2010-10-06 | 埃迪威克斯生物科学公司 | 作为gsk-3抑制剂的螺环状氨基喹诺酮 |
WO2009090548A2 (en) * | 2008-01-17 | 2009-07-23 | Glenmark Pharmaceuticals, S.A. | 3-azabicyclo [3.1.0] hexane derivatives as vanilloid receptor ligands |
FR2928150A1 (fr) * | 2008-02-29 | 2009-09-04 | Vetoquinol Sa Sa | Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens |
US8071591B2 (en) | 2009-03-11 | 2011-12-06 | Kyorin Pharmaceutical Co., Ltd. | 7-cycloalkylaminoquinolones as GSK-3 inhibitors |
CN102030737B (zh) * | 2010-10-29 | 2014-03-26 | 重庆巴仕迪动物药业有限公司 | 克林沙星氨基衍生物及其应用 |
WO2013142628A2 (en) * | 2012-03-20 | 2013-09-26 | Fred Hutchinson Cancer Research Center | Antibiotic compounds and compositions, and methods for identification thereof |
NZ630199A (en) * | 2012-08-03 | 2016-12-23 | Gilead Sciences Inc | Process and intermediates for preparing integrase inhibitors |
EP3221295B1 (en) * | 2014-11-17 | 2021-04-14 | Nirogy Therapeutics, Inc. | Monocarboxylate transport modulators and uses thereof |
JP2018528260A (ja) * | 2015-07-28 | 2018-09-27 | ビオーム バイオサイエンシズ プライベート リミティド | 抗菌性治療薬及び予防薬 |
DE102017218119A1 (de) * | 2017-10-11 | 2019-04-11 | Christian-Albrechts-Universität Zu Kiel | In der Umwelt abbaubare Chinolon-Antibiotika mit Hemiaminal-Struktureinheit |
CN108484577B (zh) * | 2018-03-05 | 2021-03-30 | 复旦大学 | 一种嘧啶-喹诺酮类杂合物及其制备方法和用途 |
CN111087409B (zh) * | 2018-10-24 | 2021-06-08 | 江阴安博生物医药有限公司 | 一种喹诺酮类化合物及其制备方法和应用 |
JP7324846B2 (ja) * | 2018-12-18 | 2023-08-10 | エランコ・ティアゲゾンタイト・アーゲー | 二環式誘導体 |
CN109942546B (zh) * | 2019-04-16 | 2022-04-08 | 西南大学 | 喹诺酮嘧啶类化合物及其制备方法和应用 |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1598915A (en) * | 1977-09-20 | 1981-09-23 | Bellon Labor Sa Roger | 1,4-dihydro-quinoline-3-carboxylic acid derivatives process for their preparation and composition containing them |
GB2093018B (en) * | 1979-08-22 | 1984-09-12 | Kyorin Seiyaku Kk | 6,8-difluoro-quinoline carboxylic acid derivatives |
JPS5630964A (en) | 1979-08-22 | 1981-03-28 | Kyorin Pharmaceut Co Ltd | Novel substituted quinolinecarboxylic acid and its preparation |
JPS5746986A (en) * | 1980-09-02 | 1982-03-17 | Dai Ichi Seiyaku Co Ltd | Pyrido(1,2,3-de)(1,4)benzoxazine derivative |
DE3142854A1 (de) | 1981-10-29 | 1983-05-11 | Bayer Ag, 5090 Leverkusen | 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7-piperazino-chinolin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
DE3033157A1 (de) | 1980-09-03 | 1982-04-01 | Bayer Ag, 5090 Leverkusen | 7-amino-1-cyclopropyl-4-oxo-1,4-dihydro-naphthyridin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
NZ208470A (en) | 1983-07-18 | 1988-06-30 | Abbott Lab | 6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives and antibacterial compositions containing such |
AU553415B2 (en) * | 1983-09-19 | 1986-07-17 | Abbott Japan Co., Ltd. | 6-fluoro-1-4-dihydro-4-oxo-7-substituted piperazinyl- quinoline-3-carboxylic acids |
DE3577089D1 (de) | 1984-01-26 | 1990-05-17 | Abbott Lab | Antibakterielle chinolinderivate. |
IT1173374B (it) * | 1984-02-24 | 1987-06-24 | Mediolanum Farmaceutici Srl | Derivati pirido-benzotiazinici ad elevata attivita' antimicrobica |
DE3608745A1 (de) * | 1985-07-24 | 1987-01-29 | Bayer Ag | Bakterizide zubereitungen zur anwendung auf dem gebiet der veterinaermedizin |
DE3632222A1 (de) * | 1986-09-23 | 1988-04-07 | Bayer Ag | Topisch anwendbare zubereitungen von gyrase-inhibitoren |
DE3637649A1 (de) * | 1986-10-13 | 1988-04-14 | Uwe Dr Spohr | Verwendung von 4-chinolon-derivaten zur bekaempfung von protozoen und helminthen |
DE3639465A1 (de) * | 1986-11-18 | 1988-05-19 | Hoechst Ag | Optisch aktive gyrasehemmer, ihre herstellung und verwendung als antibiotika |
MY104139A (en) * | 1988-08-09 | 1994-02-28 | Daiichi Seiyaku Co | Antimicrobial agent for animals |
US5225413A (en) * | 1988-09-16 | 1993-07-06 | Bayer-Aktiengesellschaft | pH-neutral aqueous solutions of quinolone-carboxylic acids |
US5164402A (en) | 1989-08-16 | 1992-11-17 | Pfizer Inc | Azabicyclo quinolone and naphthyridinone carboxylic acids |
US5266569A (en) * | 1989-08-16 | 1993-11-30 | Pfizer Inc. | Azatricyclo carboxylic acids useful as anti-bacterial agents |
FR2674854B1 (fr) * | 1991-04-04 | 1995-03-03 | Bouchara | Nouvelles quinolones leur procede de preparation et les compositions pharmaceutiques en refermant. |
US5395936A (en) * | 1993-06-04 | 1995-03-07 | Manzo; Ruben H. | 7-(4-[4-aminophenyl)sulphonyl]-1-piperazinyl fluorquinolonic derivatives and synthesis |
EP0676199B1 (en) * | 1994-04-07 | 1998-09-02 | Pfizer Inc. | Use of trovafloxacin or derivatives thereof for the manufacture of a medicament for the treatment of H. pylori infections |
DE19519822A1 (de) * | 1995-05-31 | 1996-12-05 | Bayer Ag | Neue antibakterielle Mittel |
-
1999
- 1999-11-15 SE SE9904108A patent/SE9904108D0/sv unknown
-
2000
- 2000-11-13 DE DE60039183T patent/DE60039183D1/de not_active Expired - Fee Related
- 2000-11-13 EP EP00980176A patent/EP1230235B1/en not_active Expired - Lifetime
- 2000-11-13 US US10/111,898 patent/US6967205B1/en not_active Expired - Fee Related
- 2000-11-13 AU AU17472/01A patent/AU1747201A/en not_active Abandoned
- 2000-11-13 AT AT00980176T patent/ATE398117T1/de not_active IP Right Cessation
- 2000-11-13 JP JP2001538897A patent/JP2003514812A/ja active Pending
- 2000-11-13 WO PCT/SE2000/002217 patent/WO2001036408A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
JP2003514812A (ja) | 2003-04-22 |
AU1747201A (en) | 2001-05-30 |
DE60039183D1 (de) | 2008-07-24 |
WO2001036408A1 (en) | 2001-05-25 |
ATE398117T1 (de) | 2008-07-15 |
EP1230235B1 (en) | 2008-06-11 |
US6967205B1 (en) | 2005-11-22 |
EP1230235A1 (en) | 2002-08-14 |
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