JP2011519854A5 - - Google Patents

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Publication number
JP2011519854A5
JP2011519854A5 JP2011507529A JP2011507529A JP2011519854A5 JP 2011519854 A5 JP2011519854 A5 JP 2011519854A5 JP 2011507529 A JP2011507529 A JP 2011507529A JP 2011507529 A JP2011507529 A JP 2011507529A JP 2011519854 A5 JP2011519854 A5 JP 2011519854A5
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fluoro
acceptable salt
hydrogen
optionally substituted
compound
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JP2011507529A
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JP5658139B2 (ja
JP2011519854A (ja
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Priority claimed from PCT/US2009/040589 external-priority patent/WO2009134617A1/en
Publication of JP2011519854A publication Critical patent/JP2011519854A/ja
Publication of JP2011519854A5 publication Critical patent/JP2011519854A5/ja
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Publication of JP5658139B2 publication Critical patent/JP5658139B2/ja
Expired - Fee Related legal-status Critical Current
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JP2011507529A 2008-05-02 2009-04-15 Bace阻害剤 Expired - Fee Related JP5658139B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4988108P 2008-05-02 2008-05-02
US61/049,881 2008-05-02
PCT/US2009/040589 WO2009134617A1 (en) 2008-05-02 2009-04-15 Aminodihydrothiazine derivatives as bace inhibitors for the treatment of alzheimer's disease

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014208277A Division JP2015051980A (ja) 2008-05-02 2014-10-09 Bace阻害剤

Publications (3)

Publication Number Publication Date
JP2011519854A JP2011519854A (ja) 2011-07-14
JP2011519854A5 true JP2011519854A5 (enExample) 2012-06-07
JP5658139B2 JP5658139B2 (ja) 2015-01-21

Family

ID=40839645

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011507529A Expired - Fee Related JP5658139B2 (ja) 2008-05-02 2009-04-15 Bace阻害剤
JP2014208277A Pending JP2015051980A (ja) 2008-05-02 2014-10-09 Bace阻害剤
JP2016211189A Withdrawn JP2017048212A (ja) 2008-05-02 2016-10-28 Bace阻害剤

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014208277A Pending JP2015051980A (ja) 2008-05-02 2014-10-09 Bace阻害剤
JP2016211189A Withdrawn JP2017048212A (ja) 2008-05-02 2016-10-28 Bace阻害剤

Country Status (32)

Country Link
US (1) US7648983B2 (enExample)
EP (1) EP2297120B1 (enExample)
JP (3) JP5658139B2 (enExample)
KR (1) KR101253835B1 (enExample)
CN (1) CN102015667B (enExample)
AR (1) AR071187A1 (enExample)
AU (1) AU2009241515B2 (enExample)
CA (1) CA2723207C (enExample)
CL (1) CL2009000860A1 (enExample)
CO (1) CO6311079A2 (enExample)
CR (1) CR11776A (enExample)
DK (1) DK2297120T3 (enExample)
DO (1) DOP2010000328A (enExample)
EA (1) EA016955B1 (enExample)
EC (1) ECSP10010582A (enExample)
ES (1) ES2549087T3 (enExample)
HR (1) HRP20150941T1 (enExample)
HU (1) HUE025520T2 (enExample)
IL (1) IL208350A (enExample)
MA (1) MA32351B1 (enExample)
MX (1) MX2010011972A (enExample)
NZ (1) NZ588300A (enExample)
PE (1) PE20091816A1 (enExample)
PL (1) PL2297120T3 (enExample)
PT (1) PT2297120E (enExample)
RS (1) RS54260B1 (enExample)
SI (1) SI2297120T1 (enExample)
SV (1) SV2010003718A (enExample)
TW (1) TWI431004B (enExample)
UA (1) UA102251C2 (enExample)
WO (1) WO2009134617A1 (enExample)
ZA (1) ZA201006868B (enExample)

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CN103596939A (zh) * 2011-04-13 2014-02-19 默沙东公司 作为bace抑制剂的5-取代的亚氨基噻嗪类及其单和二氧化物、组合物及其应用
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