HRP20150941T1 - Derivati aminodihidrotiazina kao inhibitori bace u lijeäśenju alzheimerove bolesti - Google Patents

Derivati aminodihidrotiazina kao inhibitori bace u lijeäśenju alzheimerove bolesti Download PDF

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Publication number
HRP20150941T1
HRP20150941T1 HRP20150941TT HRP20150941T HRP20150941T1 HR P20150941 T1 HRP20150941 T1 HR P20150941T1 HR P20150941T T HRP20150941T T HR P20150941TT HR P20150941 T HRP20150941 T HR P20150941T HR P20150941 T1 HRP20150941 T1 HR P20150941T1
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Croatia
Prior art keywords
fluorine
pharmaceutically acceptable
compound according
hydrogen
acceptable salt
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HRP20150941TT
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English (en)
Croatian (hr)
Inventor
James Edmund Audia
Dustin James Mergott
Scott Martin Sheehan
Brian Morgan Watson
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Eli Lilly & Company
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40839645&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20150941(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eli Lilly & Company filed Critical Eli Lilly & Company
Publication of HRP20150941T1 publication Critical patent/HRP20150941T1/hr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
    • C07D279/06—1,3-Thiazines; Hydrogenated 1,3-thiazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HRP20150941TT 2008-05-02 2009-04-15 Derivati aminodihidrotiazina kao inhibitori bace u lijeäśenju alzheimerove bolesti HRP20150941T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4988108P 2008-05-02 2008-05-02
EP09739419.1A EP2297120B1 (en) 2008-05-02 2009-04-15 Aminodihydrothiazine derivatives as bace inhibitors for the treatment of alzheimer's disease
PCT/US2009/040589 WO2009134617A1 (en) 2008-05-02 2009-04-15 Aminodihydrothiazine derivatives as bace inhibitors for the treatment of alzheimer's disease

Publications (1)

Publication Number Publication Date
HRP20150941T1 true HRP20150941T1 (hr) 2015-10-09

Family

ID=40839645

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20150941TT HRP20150941T1 (hr) 2008-05-02 2009-04-15 Derivati aminodihidrotiazina kao inhibitori bace u lijeäśenju alzheimerove bolesti

Country Status (32)

Country Link
US (1) US7648983B2 (enExample)
EP (1) EP2297120B1 (enExample)
JP (3) JP5658139B2 (enExample)
KR (1) KR101253835B1 (enExample)
CN (1) CN102015667B (enExample)
AR (1) AR071187A1 (enExample)
AU (1) AU2009241515B2 (enExample)
CA (1) CA2723207C (enExample)
CL (1) CL2009000860A1 (enExample)
CO (1) CO6311079A2 (enExample)
CR (1) CR11776A (enExample)
DK (1) DK2297120T3 (enExample)
DO (1) DOP2010000328A (enExample)
EA (1) EA016955B1 (enExample)
EC (1) ECSP10010582A (enExample)
ES (1) ES2549087T3 (enExample)
HR (1) HRP20150941T1 (enExample)
HU (1) HUE025520T2 (enExample)
IL (1) IL208350A (enExample)
MA (1) MA32351B1 (enExample)
MX (1) MX2010011972A (enExample)
NZ (1) NZ588300A (enExample)
PE (1) PE20091816A1 (enExample)
PL (1) PL2297120T3 (enExample)
PT (1) PT2297120E (enExample)
RS (1) RS54260B1 (enExample)
SI (1) SI2297120T1 (enExample)
SV (1) SV2010003718A (enExample)
TW (1) TWI431004B (enExample)
UA (1) UA102251C2 (enExample)
WO (1) WO2009134617A1 (enExample)
ZA (1) ZA201006868B (enExample)

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