PT2297120E - Derivados de aminodi-hidrotiazina como inibidores da bace para o tratamento da doença de alzheimer - Google Patents

Derivados de aminodi-hidrotiazina como inibidores da bace para o tratamento da doença de alzheimer Download PDF

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Publication number
PT2297120E
PT2297120E PT97394191T PT09739419T PT2297120E PT 2297120 E PT2297120 E PT 2297120E PT 97394191 T PT97394191 T PT 97394191T PT 09739419 T PT09739419 T PT 09739419T PT 2297120 E PT2297120 E PT 2297120E
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PT
Portugal
Prior art keywords
alzheimer
disease
treatment
bace inhibitors
aminodihydrothiazine derivatives
Prior art date
Application number
PT97394191T
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English (en)
Inventor
James Edmund Audia
Dustin James Mergott
Scott Martin Sheehan
Brian Morgan Watson
Original Assignee
Lilly Co Eli
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40839645&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2297120(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT2297120E publication Critical patent/PT2297120E/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
    • C07D279/06—1,3-Thiazines; Hydrogenated 1,3-thiazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
PT97394191T 2008-05-02 2009-04-15 Derivados de aminodi-hidrotiazina como inibidores da bace para o tratamento da doença de alzheimer PT2297120E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4988108P 2008-05-02 2008-05-02

Publications (1)

Publication Number Publication Date
PT2297120E true PT2297120E (pt) 2015-10-26

Family

ID=40839645

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97394191T PT2297120E (pt) 2008-05-02 2009-04-15 Derivados de aminodi-hidrotiazina como inibidores da bace para o tratamento da doença de alzheimer

Country Status (32)

Country Link
US (1) US7648983B2 (pt)
EP (1) EP2297120B1 (pt)
JP (3) JP5658139B2 (pt)
KR (1) KR101253835B1 (pt)
CN (1) CN102015667B (pt)
AR (1) AR071187A1 (pt)
AU (1) AU2009241515B2 (pt)
CA (1) CA2723207C (pt)
CL (1) CL2009000860A1 (pt)
CO (1) CO6311079A2 (pt)
CR (1) CR11776A (pt)
DK (1) DK2297120T3 (pt)
DO (1) DOP2010000328A (pt)
EA (1) EA016955B1 (pt)
EC (1) ECSP10010582A (pt)
ES (1) ES2549087T3 (pt)
HR (1) HRP20150941T1 (pt)
HU (1) HUE025520T2 (pt)
IL (1) IL208350A (pt)
MA (1) MA32351B1 (pt)
MX (1) MX2010011972A (pt)
NZ (1) NZ588300A (pt)
PE (1) PE20091816A1 (pt)
PL (1) PL2297120T3 (pt)
PT (1) PT2297120E (pt)
RS (1) RS54260B1 (pt)
SI (1) SI2297120T1 (pt)
SV (1) SV2010003718A (pt)
TW (1) TWI431004B (pt)
UA (1) UA102251C2 (pt)
WO (1) WO2009134617A1 (pt)
ZA (1) ZA201006868B (pt)

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Publication number Publication date
US7648983B2 (en) 2010-01-19
DK2297120T3 (en) 2015-10-12
UA102251C2 (ru) 2013-06-25
HRP20150941T1 (hr) 2015-10-09
ECSP10010582A (es) 2010-11-30
SV2010003718A (es) 2011-02-14
JP2015051980A (ja) 2015-03-19
NZ588300A (en) 2012-07-27
CN102015667A (zh) 2011-04-13
HUE025520T2 (en) 2016-02-29
CO6311079A2 (es) 2011-08-22
EA016955B1 (ru) 2012-08-30
TW200946522A (en) 2009-11-16
WO2009134617A1 (en) 2009-11-05
DOP2010000328A (es) 2010-11-15
JP5658139B2 (ja) 2015-01-21
MX2010011972A (es) 2010-11-25
KR20100125475A (ko) 2010-11-30
TWI431004B (zh) 2014-03-21
EA201071264A1 (ru) 2011-04-29
EP2297120B1 (en) 2015-08-19
RS54260B1 (en) 2016-02-29
IL208350A0 (en) 2010-12-30
PE20091816A1 (es) 2009-11-25
CR11776A (es) 2011-01-28
CA2723207C (en) 2016-07-12
KR101253835B1 (ko) 2013-04-15
IL208350A (en) 2014-05-28
ES2549087T3 (es) 2015-10-22
JP2011519854A (ja) 2011-07-14
SI2297120T1 (sl) 2015-11-30
ZA201006868B (en) 2012-03-28
EP2297120A1 (en) 2011-03-23
PL2297120T3 (pl) 2016-01-29
AR071187A1 (es) 2010-06-02
AU2009241515B2 (en) 2012-04-19
CL2009000860A1 (es) 2010-05-07
CA2723207A1 (en) 2009-11-05
JP2017048212A (ja) 2017-03-09
MA32351B1 (fr) 2011-06-01
AU2009241515A1 (en) 2009-11-05
CN102015667B (zh) 2013-06-12
US20090275566A1 (en) 2009-11-05

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