JP2014526510A5 - - Google Patents
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- JP2014526510A5 JP2014526510A5 JP2014530787A JP2014530787A JP2014526510A5 JP 2014526510 A5 JP2014526510 A5 JP 2014526510A5 JP 2014530787 A JP2014530787 A JP 2014530787A JP 2014530787 A JP2014530787 A JP 2014530787A JP 2014526510 A5 JP2014526510 A5 JP 2014526510A5
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- alkyl
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- cancer
- disease
- pyridyl
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161534601P | 2011-09-14 | 2011-09-14 | |
| US61/534,601 | 2011-09-14 | ||
| US201261624646P | 2012-04-16 | 2012-04-16 | |
| US61/624,646 | 2012-04-16 | ||
| PCT/US2012/055172 WO2013040215A1 (en) | 2011-09-14 | 2012-09-13 | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016202360A Division JP6457459B2 (ja) | 2011-09-14 | 2016-10-14 | インダゾール−３−カルボキサミドおよびＷＮＴ／β−カテニンシグナル伝達経路阻害剤としてのそれらの使用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2014526510A JP2014526510A (ja) | 2014-10-06 |
| JP2014526510A5 true JP2014526510A5 (OSRAM) | 2016-12-01 |
Family
ID=47883736
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014530787A Pending JP2014526510A (ja) | 2011-09-14 | 2012-09-13 | インダゾール−３−カルボキサミドおよびＷＮＴ／β−カテニンシグナル伝達経路阻害剤としてのそれらの使用 |
| JP2016202360A Active JP6457459B2 (ja) | 2011-09-14 | 2016-10-14 | インダゾール−３−カルボキサミドおよびＷＮＴ／β−カテニンシグナル伝達経路阻害剤としてのそれらの使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016202360A Active JP6457459B2 (ja) | 2011-09-14 | 2016-10-14 | インダゾール−３−カルボキサミドおよびＷＮＴ／β−カテニンシグナル伝達経路阻害剤としてのそれらの使用 |
Country Status (32)
| Country | Link |
|---|---|
| US (6) | US9221793B2 (OSRAM) |
| EP (2) | EP3473099A1 (OSRAM) |
| JP (2) | JP2014526510A (OSRAM) |
| KR (1) | KR102010611B1 (OSRAM) |
| CN (2) | CN109705097B (OSRAM) |
| AU (2) | AU2012308570B2 (OSRAM) |
| BR (1) | BR112014006127A2 (OSRAM) |
| CA (1) | CA2848659C (OSRAM) |
| CL (1) | CL2014000642A1 (OSRAM) |
| CO (1) | CO6940416A2 (OSRAM) |
| CY (1) | CY1122795T1 (OSRAM) |
| DK (1) | DK2755483T3 (OSRAM) |
| ES (1) | ES2711777T3 (OSRAM) |
| HR (1) | HRP20190281T1 (OSRAM) |
| HU (1) | HUE041576T2 (OSRAM) |
| IL (1) | IL231536A (OSRAM) |
| IN (1) | IN2014CN02646A (OSRAM) |
| LT (1) | LT2755483T (OSRAM) |
| ME (1) | ME03332B (OSRAM) |
| MX (3) | MX362494B (OSRAM) |
| MY (1) | MY184882A (OSRAM) |
| PE (1) | PE20141678A1 (OSRAM) |
| PH (1) | PH12014500594A1 (OSRAM) |
| PL (1) | PL2755483T3 (OSRAM) |
| PT (1) | PT2755483T (OSRAM) |
| RS (1) | RS58462B1 (OSRAM) |
| RU (1) | RU2627693C2 (OSRAM) |
| SG (3) | SG10202002005SA (OSRAM) |
| SI (1) | SI2755483T1 (OSRAM) |
| SM (1) | SMT201900098T1 (OSRAM) |
| WO (1) | WO2013040215A1 (OSRAM) |
| ZA (1) | ZA201402623B (OSRAM) |
Families Citing this family (80)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011019651A1 (en) | 2009-08-10 | 2011-02-17 | Epitherix, Llc | Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof |
| SMT201700581T1 (it) | 2009-12-21 | 2018-01-11 | Samumed Llc | 1h-pirazolo[3,4-b]piridine e loro usi terapeutici |
| US9526648B2 (en) | 2010-06-13 | 2016-12-27 | Synerz Medical, Inc. | Intragastric device for treating obesity |
| US10010439B2 (en) | 2010-06-13 | 2018-07-03 | Synerz Medical, Inc. | Intragastric device for treating obesity |
| US10420665B2 (en) | 2010-06-13 | 2019-09-24 | W. L. Gore & Associates, Inc. | Intragastric device for treating obesity |
| US8628554B2 (en) | 2010-06-13 | 2014-01-14 | Virender K. Sharma | Intragastric device for treating obesity |
| EP3473099A1 (en) | 2011-09-14 | 2019-04-24 | Samumed, LLC | Indazole-3-carboxamides and their use as wnt/b-catenin signaling pathway inhibitors |
| PH12017500997A1 (en) | 2012-04-04 | 2018-02-19 | Samumed Llc | Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof |
| NZ629282A (en) | 2012-05-04 | 2017-04-28 | Samumed Llc | 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof |
| BR112015014752B1 (pt) | 2012-12-21 | 2022-07-05 | Plexxikon, Inc | Compostos e seus uso para modulação de cinase |
| CA2897400A1 (en) | 2013-01-08 | 2014-07-17 | Samumed, Llc | 3-(benzoimidazol-2-yl)-indazole inhibitors of the wnt signaling pathway and therapeutic uses thereof |
| CA3184040A1 (en) | 2013-03-14 | 2014-10-02 | The Brigham And Women's Hospital, Inc. | Compositions and methods for epithelial stem cell expansion comprising a wnt agonist and a histone deacetylase inhibitor |
| GB201309333D0 (en) * | 2013-05-23 | 2013-07-10 | Agency Science Tech & Res | Purine diones as WNT pathway modulators |
| JP6657079B2 (ja) | 2013-10-15 | 2020-03-04 | ラドゥックス・ディヴァイシーズ・エルエルシー | 弁器具への医療用装置の固定 |
| CA2942687A1 (en) | 2014-03-20 | 2015-09-24 | Samumed, Llc | 5-substituted indazole-3-carboxamides and preparation and use thereof |
| WO2016037016A1 (en) | 2014-09-03 | 2016-03-10 | The Brigham And Women's Hospital, Inc. | Compositions, systems, and methods for generating inner ear hair cells for treatment of hearing loss |
| WO2016040181A1 (en) | 2014-09-08 | 2016-03-17 | Samumed, Llc | 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof |
| WO2016040182A1 (en) | 2014-09-08 | 2016-03-17 | Samumed, Llc | 2-(1h-indazol-3-yl)-1h-imidazo[4,5-c]pyridine and therapeutic uses thereof |
| WO2016040193A1 (en) | 2014-09-08 | 2016-03-17 | Samumed, Llc | 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof |
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