JP2013529637A5 - - Google Patents

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Publication number
JP2013529637A5
JP2013529637A5 JP2013516636A JP2013516636A JP2013529637A5 JP 2013529637 A5 JP2013529637 A5 JP 2013529637A5 JP 2013516636 A JP2013516636 A JP 2013516636A JP 2013516636 A JP2013516636 A JP 2013516636A JP 2013529637 A5 JP2013529637 A5 JP 2013529637A5
Authority
JP
Japan
Prior art keywords
solid dispersion
phenoxymethyl
tetrazol
thiazol
pyrimidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2013516636A
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English (en)
Japanese (ja)
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JP2013529637A (ja
JP5847813B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/040972 external-priority patent/WO2011163090A1/en
Publication of JP2013529637A publication Critical patent/JP2013529637A/ja
Publication of JP2013529637A5 publication Critical patent/JP2013529637A5/ja
Application granted granted Critical
Publication of JP5847813B2 publication Critical patent/JP5847813B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2013516636A 2010-06-23 2011-06-17 ５−エチル−２−｛４−［４−（４−テトラゾル−１−イル−フェノキシメチル）−チアゾール−２−イル］−ピペリジン−１−イル｝−ピリミジンの組成物 Expired - Fee Related JP5847813B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35798110P 2010-06-23 2010-06-23
US61/357,981 2010-06-23
PCT/US2011/040972 WO2011163090A1 (en) 2010-06-23 2011-06-17 Compositions of 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine

Publications (3)

Publication Number Publication Date
JP2013529637A JP2013529637A (ja) 2013-07-22
JP2013529637A5 true JP2013529637A5 (enExample) 2014-08-07
JP5847813B2 JP5847813B2 (ja) 2016-01-27

Family

ID=44584703

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013516636A Expired - Fee Related JP5847813B2 (ja) 2010-06-23 2011-06-17 ５−エチル−２−｛４−［４−（４−テトラゾル−１−イル−フェノキシメチル）−チアゾール−２−イル］−ピペリジン−１−イル｝−ピリミジンの組成物

Country Status (8)

Country Link
US (2) US9241924B2 (enExample)
EP (1) EP2585048B1 (enExample)
JP (1) JP5847813B2 (enExample)
CN (2) CN103037843A (enExample)
BR (1) BR112012032248A2 (enExample)
CA (1) CA2802541A1 (enExample)
ES (1) ES2676209T3 (enExample)
WO (1) WO2011163090A1 (enExample)

Families Citing this family (12)

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JP5489997B2 (ja) 2007-07-19 2014-05-14 シマベイ セラピューティクス， インコーポレーテッド 糖尿病および代謝疾患の治療のためのＲＵＰ３またはＧＰＲｌ１９受容体のアゴニストとしてのＮ−アザ環状置換ピロール、ピラゾール、イミダゾール、トリアゾールおよびテトラゾール誘導体
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US9790182B2 (en) * 2014-06-11 2017-10-17 Bayer Cropscience Aktiengesellschaft Preparation of piperidine-4-carbothioamide
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CN116323608A (zh) 2020-05-19 2023-06-23 卡尔优普公司 Ampk活化剂
EP4172162A4 (en) 2020-06-26 2024-08-07 Kallyope, Inc. AMPK ACTIVATORS

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