JP2013529637A5 - - Google Patents

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Publication number
JP2013529637A5
JP2013529637A5 JP2013516636A JP2013516636A JP2013529637A5 JP 2013529637 A5 JP2013529637 A5 JP 2013529637A5 JP 2013516636 A JP2013516636 A JP 2013516636A JP 2013516636 A JP2013516636 A JP 2013516636A JP 2013529637 A5 JP2013529637 A5 JP 2013529637A5
Authority
JP
Japan
Prior art keywords
solid dispersion
phenoxymethyl
tetrazol
thiazol
pyrimidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2013516636A
Other languages
English (en)
Japanese (ja)
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JP5847813B2 (ja
JP2013529637A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/040972 external-priority patent/WO2011163090A1/en
Publication of JP2013529637A publication Critical patent/JP2013529637A/ja
Publication of JP2013529637A5 publication Critical patent/JP2013529637A5/ja
Application granted granted Critical
Publication of JP5847813B2 publication Critical patent/JP5847813B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2013516636A 2010-06-23 2011-06-17 ５−エチル−２−｛４−［４−（４−テトラゾル−１−イル−フェノキシメチル）−チアゾール−２−イル］−ピペリジン−１−イル｝−ピリミジンの組成物 Expired - Fee Related JP5847813B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35798110P 2010-06-23 2010-06-23
US61/357,981 2010-06-23
PCT/US2011/040972 WO2011163090A1 (en) 2010-06-23 2011-06-17 Compositions of 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine

Publications (3)

Publication Number Publication Date
JP2013529637A JP2013529637A (ja) 2013-07-22
JP2013529637A5 true JP2013529637A5 (enExample) 2014-08-07
JP5847813B2 JP5847813B2 (ja) 2016-01-27

Family

ID=44584703

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013516636A Expired - Fee Related JP5847813B2 (ja) 2010-06-23 2011-06-17 ５−エチル−２−｛４−［４−（４−テトラゾル−１−イル−フェノキシメチル）−チアゾール−２−イル］−ピペリジン−１−イル｝−ピリミジンの組成物

Country Status (8)

Country Link
US (2) US9241924B2 (enExample)
EP (1) EP2585048B1 (enExample)
JP (1) JP5847813B2 (enExample)
CN (2) CN109674753A (enExample)
BR (1) BR112012032248A2 (enExample)
CA (1) CA2802541A1 (enExample)
ES (1) ES2676209T3 (enExample)
WO (1) WO2011163090A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7638541B2 (en) 2006-12-28 2009-12-29 Metabolex Inc. 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine
AU2008279447A1 (en) 2007-07-19 2009-01-29 Metabolex, Inc. N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders
PL2280704T3 (pl) * 2008-03-31 2015-10-30 Cymabay Therapeutics Inc Związki oksymetylenoarylowe i ich zastosowania
US20110160222A1 (en) * 2008-11-26 2011-06-30 Metabolex, Inc. Modulators of glucose homeostasis for the treatment of diabetes and metabolic disorders
EP2483281B1 (en) * 2009-10-01 2014-06-04 Cymabay Therapeutics, Inc. Substituted tetrazol-1-yl-phenoxymethyl-thiazol-2-yl-piperidinyl-pyrimidine salts
BR112012032248A2 (pt) 2010-06-23 2016-09-13 Metabolex Inc composições de 5-etil-2-{4-[-4(-4-tetrazol-1-il-fenoximetil)-tiazol-2-il]-piperidin-1-il}-pirimidina
CN113209024A (zh) * 2013-12-31 2021-08-06 阿森迪亚制药有限责任公司 疏水性化合物的药物组合物
ES2753582T3 (es) * 2014-06-11 2020-04-13 Bayer Cropscience Ag Preparación de piperidin-4-carbotioamida
WO2018026890A1 (en) * 2016-08-03 2018-02-08 Cymabay Therapeutics Oxymethylene aryl compounds for treating inflammatory gastrointestinal diseases or gastrointestinal conditions
MX2022010548A (es) 2020-02-28 2022-09-23 Kallyope Inc Agonistas de gpr40.
MX2022014505A (es) 2020-05-19 2022-12-13 Kallyope Inc Activadores de la ampk.
CA3183575A1 (en) 2020-06-26 2021-12-30 Iyassu Sebhat Ampk activators

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