JP2014526508A5 - - Google Patents

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Publication number
JP2014526508A5
JP2014526508A5 JP2014530765A JP2014530765A JP2014526508A5 JP 2014526508 A5 JP2014526508 A5 JP 2014526508A5 JP 2014530765 A JP2014530765 A JP 2014530765A JP 2014530765 A JP2014530765 A JP 2014530765A JP 2014526508 A5 JP2014526508 A5 JP 2014526508A5
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JP
Japan
Prior art keywords
dosage form
oral dosage
disease
weight
dispersion
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2014530765A
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English (en)
Japanese (ja)
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JP2014526508A (ja
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Publication date
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Priority claimed from PCT/US2012/054990 external-priority patent/WO2013040120A1/en
Publication of JP2014526508A publication Critical patent/JP2014526508A/ja
Publication of JP2014526508A5 publication Critical patent/JP2014526508A5/ja
Ceased legal-status Critical Current

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JP2014530765A 2011-09-14 2012-09-13 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤 Ceased JP2014526508A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161534841P 2011-09-14 2011-09-14
US61/534,841 2011-09-14
PCT/US2012/054990 WO2013040120A1 (en) 2011-09-14 2012-09-13 Formulations of cyclopropanecarboxylic acid {2-(1s)-1-(3-ethoxy-4-methoxy-phenyl)-2-methanesulfonyl-ethyl]-3-oxo-2,3-dihydro-1h-isoindol-4-yl}-amidecelgene corporation state of incorporation:delaware

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017016400A Division JP6339251B2 (ja) 2011-09-14 2017-02-01 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤

Publications (2)

Publication Number Publication Date
JP2014526508A JP2014526508A (ja) 2014-10-06
JP2014526508A5 true JP2014526508A5 (enExample) 2015-11-05

Family

ID=46964044

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2014530765A Ceased JP2014526508A (ja) 2011-09-14 2012-09-13 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤
JP2017016400A Active JP6339251B2 (ja) 2011-09-14 2017-02-01 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤
JP2017104141A Pending JP2017178961A (ja) 2011-09-14 2017-05-26 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2017016400A Active JP6339251B2 (ja) 2011-09-14 2017-02-01 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤
JP2017104141A Pending JP2017178961A (ja) 2011-09-14 2017-05-26 シクロプロパンカルボン酸{2−[(1s)−1−(3−エトキシ−4−メトキシ−フェニル)−2−メタンスルホニル−エチル]−3−オキソ−2,3−ジヒドロ−1h−イソインドール−4−イル}−アミドの製剤

Country Status (15)

Country Link
US (1) US9884042B2 (enExample)
EP (1) EP2765993B1 (enExample)
JP (3) JP2014526508A (enExample)
KR (1) KR20140063808A (enExample)
CN (1) CN105142615A (enExample)
AU (1) AU2012308663B2 (enExample)
CA (1) CA2848493A1 (enExample)
CL (1) CL2014000623A1 (enExample)
ES (1) ES2803524T3 (enExample)
IL (1) IL231462A0 (enExample)
MX (1) MX356105B (enExample)
PH (1) PH12014500593A1 (enExample)
RU (2) RU2017121896A (enExample)
SG (1) SG11201400632YA (enExample)
WO (1) WO2013040120A1 (enExample)

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EP2764866A1 (en) 2013-02-07 2014-08-13 IP Gesellschaft für Management mbH Inhibitors of nedd8-activating enzyme
EP3089736B1 (en) * 2013-12-31 2025-07-23 Ascendia Pharmaceuticals, LLC Pharmaceutical compositions for poorly water-soluble compounds
WO2015175505A1 (en) * 2014-05-15 2015-11-19 Lundbeck Llc Tetrabenazine modified release formulation
US20170087129A1 (en) * 2014-05-16 2017-03-30 Celgene Corporation Compositions and methods for the treatment of atherosclerotic cardiovascular diseases with pde4 modulators
KR101722564B1 (ko) * 2014-09-16 2017-04-03 강원대학교산학협력단 수-난용성 약물을 포함하는 고체분산체
WO2016199927A1 (ja) * 2015-06-12 2016-12-15 日産化学工業株式会社 カルシウム塩組成物及びそれを用いたフィラグリン産生促進剤
KR20200043618A (ko) 2018-10-18 2020-04-28 주식회사유한양행 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구투여용 약학 조성물
EP4221704B1 (en) * 2020-10-01 2025-09-24 Imago Biosciences Inc. Pharmaceutical formulations for treating diseases mediated by kdm1a

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CN103391770A (zh) * 2011-01-10 2013-11-13 细胞基因公司 环丙烷羧酸{2-[(1s)-1-(3-乙氧基-4-甲氧基-苯基)-2-甲烷磺酰基-乙基]-3-氧代-2,3-二氢-1h-异吲哚-4-基}-酰胺的口服剂型
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