JP2007510621A - アミノ酸プロドラッグ - Google Patents
アミノ酸プロドラッグ Download PDFInfo
- Publication number
- JP2007510621A JP2007510621A JP2006522125A JP2006522125A JP2007510621A JP 2007510621 A JP2007510621 A JP 2007510621A JP 2006522125 A JP2006522125 A JP 2006522125A JP 2006522125 A JP2006522125 A JP 2006522125A JP 2007510621 A JP2007510621 A JP 2007510621A
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- Prior art keywords
- compound
- amino acid
- patient
- compound according
- hydroxyproline
- Prior art date
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- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
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- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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| KR (3) | KR20130081319A (https=) |
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| JP2013035863A (ja) * | 2003-07-29 | 2013-02-21 | Signature R&D Holdings Llc | アミノ酸プロドラッグ |
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| IT1294205B1 (it) * | 1997-07-23 | 1999-03-24 | Farmigea Spa | Procedimento per la solubilizzazione in acqua e in veicoli acquosi di sostanze farmacologicamente attive |
| WO2002016395A1 (en) * | 2000-08-18 | 2002-02-28 | The Board Of Trustees Of The University Of Illinois | Prodrugs of betulinic acid derivatives for the treatment of cancer and hiv |
| US20020160988A1 (en) * | 2001-02-20 | 2002-10-31 | Israel Institute For Biological Research | Compounds co-inducing cholinergic up-regulation and inflammation down-regulation and uses thereof |
| US7045543B2 (en) * | 2001-11-05 | 2006-05-16 | Enzrel Inc. | Covalent conjugates of biologically-active compounds with amino acids and amino acid derivatives for targeting to physiologically-protected sites |
| ATE396731T1 (de) * | 2003-03-25 | 2008-06-15 | Vertex Pharma | Thiazole zur verwendung als inhibitoren von protein-kinasen |
| CN101123878A (zh) * | 2003-07-29 | 2008-02-13 | 信号研发控股有限责任公司 | 氨基酸前药 |
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Cited By (11)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2013035863A (ja) * | 2003-07-29 | 2013-02-21 | Signature R&D Holdings Llc | アミノ酸プロドラッグ |
| JP2012512914A (ja) * | 2008-12-19 | 2012-06-07 | ピナクル ファーマシューティカルズ インコーポレイテッド | フェナゾピリジン化合物 |
| JP2013530966A (ja) * | 2010-06-23 | 2013-08-01 | 四川大学華西医院 | 置換フェノールを含むヒドロキシ酸エステル化合物、その製造方法及びそれを用いた中枢抑制薬 |
| JP2015507636A (ja) * | 2012-01-06 | 2015-03-12 | スピニフェクス ファーマシューティカルズ ピーティーワイ リミテッド | 複素環式化合物およびその使用方法 |
| JP2019069948A (ja) * | 2012-01-18 | 2019-05-09 | テックフィールズ ファーマ カンパニー リミテッド | 肺疾患の治療のための高浸透性プロドラッグ組成物およびその薬学的組成物 |
| JP7235487B2 (ja) | 2012-01-18 | 2023-03-08 | テックフィールズ ファーマ カンパニー リミテッド | 肺疾患の治療のための高浸透性プロドラッグ組成物およびその薬学的組成物 |
| JP2015519334A (ja) * | 2012-05-07 | 2015-07-09 | セリックスビオ プライヴェート リミテッド | 抗血小板薬のプロドラッグ |
| JP2019512502A (ja) * | 2016-03-18 | 2019-05-16 | ケアジェン カンパニー, リミテッドCaregen Co., Ltd. | フィナステリドとペプチドの結合体 |
| JP2021011507A (ja) * | 2016-03-18 | 2021-02-04 | ケアジェン カンパニー, リミテッドCaregen Co., Ltd. | フィナステリドとペプチドの結合体 |
| US11357783B2 (en) | 2016-03-18 | 2022-06-14 | Caregen Co., Ltd. | Conjugate of finasteride with peptide |
| JP2018519334A (ja) * | 2016-05-10 | 2018-07-19 | 浙江海正薬業股▲ふん▼有限公司Ｚｈｅｊｉａｎｇ Ｈｉｓｕｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌ ＣＯ．，ＬＴＤ． | 水溶性ラパマイシン誘導体 |
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| IL173382A0 (en) | 2006-06-11 |
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| ZA200600660B (en) | 2007-04-25 |
| EP1660017A4 (en) | 2011-03-09 |
| NZ601780A (en) | 2012-10-26 |
| CN101123878A (zh) | 2008-02-13 |
| NZ601772A (en) | 2012-10-26 |
| KR20130081319A (ko) | 2013-07-16 |
| JP2013035863A (ja) | 2013-02-21 |
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