JP2005524660A5 - - Google Patents

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Publication number
JP2005524660A5
JP2005524660A5 JP2003571259A JP2003571259A JP2005524660A5 JP 2005524660 A5 JP2005524660 A5 JP 2005524660A5 JP 2003571259 A JP2003571259 A JP 2003571259A JP 2003571259 A JP2003571259 A JP 2003571259A JP 2005524660 A5 JP2005524660 A5 JP 2005524660A5
Authority
JP
Japan
Prior art keywords
oxo
oxazolidinecarboxamide
methyl
dihydro
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003571259A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005524660A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2003/003125 external-priority patent/WO2003072553A1/en
Publication of JP2005524660A publication Critical patent/JP2005524660A/ja
Publication of JP2005524660A5 publication Critical patent/JP2005524660A5/ja
Pending legal-status Critical Current

Links

JP2003571259A 2002-02-25 2003-02-24 Ｎ−アリール−２−オキサゾリジノン−５−カルボキサミドおよびその誘導体ならびに抗細菌剤としてのそれらの使用 Pending JP2005524660A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35949502P 2002-02-25 2002-02-25
PCT/US2003/003125 WO2003072553A1 (en) 2002-02-25 2003-02-24 N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials

Publications (2)

Publication Number Publication Date
JP2005524660A JP2005524660A (ja) 2005-08-18
JP2005524660A5 true JP2005524660A5 (enExample) 2006-04-13

Family

ID=27766097

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003571259A Pending JP2005524660A (ja) 2002-02-25 2003-02-24 Ｎ−アリール−２−オキサゾリジノン−５−カルボキサミドおよびその誘導体ならびに抗細菌剤としてのそれらの使用

Country Status (36)

Country Link
US (1) US6919329B2 (enExample)
EP (1) EP1478629B1 (enExample)
JP (1) JP2005524660A (enExample)
KR (1) KR100613532B1 (enExample)
CN (1) CN1639135A (enExample)
AP (1) AP1902A (enExample)
AR (1) AR038536A1 (enExample)
AT (1) ATE342258T1 (enExample)
AU (1) AU2003210807A1 (enExample)
BR (1) BR0307924A (enExample)
CA (1) CA2476038A1 (enExample)
CO (1) CO5611128A2 (enExample)
CY (1) CY1105797T1 (enExample)
DE (1) DE60308998T2 (enExample)
DK (1) DK1478629T3 (enExample)
EA (1) EA007490B1 (enExample)
EC (1) ECSP045245A (enExample)
ES (1) ES2271615T3 (enExample)
GE (1) GEP20074198B (enExample)
HR (1) HRP20040717A2 (enExample)
IS (1) IS7376A (enExample)
MA (1) MA27180A1 (enExample)
MX (1) MXPA04008205A (enExample)
MY (1) MY135233A (enExample)
NO (1) NO20044062L (enExample)
NZ (1) NZ534521A (enExample)
OA (1) OA12779A (enExample)
PL (1) PL372461A1 (enExample)
PT (1) PT1478629E (enExample)
SI (1) SI1478629T1 (enExample)
TN (1) TNSN04163A1 (enExample)
TW (1) TW200305568A (enExample)
UA (1) UA80112C2 (enExample)
WO (1) WO2003072553A1 (enExample)
YU (1) YU72804A (enExample)
ZA (1) ZA200406362B (enExample)

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US8324398B2 (en) 2003-06-03 2012-12-04 Rib-X Pharmaceuticals, Inc. Process for the synthesis of biaryl oxazolidinones
EP2492264A3 (en) 2003-06-03 2012-12-19 Rib-X Pharmaceuticals, Inc. Biaryl Heterocyclic Compounds And Methods Of Making And Using The Same
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KR100854211B1 (ko) * 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
WO2005082900A2 (en) * 2004-01-28 2005-09-09 Pharmacia & Upjohn Company Llc Oxazolidinone amidoximes as antibacterial agents
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ATE496914T1 (de) 2005-06-08 2011-02-15 Rib X Pharmaceuticals Inc Verfahren zur synthese von triazolen
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WO2007004032A1 (en) * 2005-07-06 2007-01-11 Pharmacia & Upjohn Company Llc Oxazolidiones containing cyclobutane as antibacterial agents
JP2009500389A (ja) * 2005-07-06 2009-01-08 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー 抗菌剤としてのアゼチジンおよびシクロブタンを含むオキサゾリジノンカルボキサミド
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WO2007088478A1 (en) * 2006-02-01 2007-08-09 Pfizer Products Inc. Indazole oxazolidinones as antibacterial agents
CN101460495B (zh) * 2006-03-31 2013-08-14 财团法人乙卯研究所 具有杂环的化合物
JP5187901B2 (ja) * 2006-08-30 2013-04-24 塩野義製薬株式会社 ヒドラジンアミド誘導体
US8088777B2 (en) * 2006-08-30 2012-01-03 Shionogi & Co., Ltd. Urea derivative
JP5455906B2 (ja) * 2007-08-06 2014-03-26 ミクウルク ファーマシューティカルズ，インコーポレイテッド 細菌感染症治療のための抗微生物性オルト−フルオロフェニルオキサゾリジノン
EP2669283A1 (en) 2007-10-02 2013-12-04 Shionogi&Co., Ltd. Oxazolidinone derivative having 7-membered hetero ring
US9643922B2 (en) 2008-08-18 2017-05-09 Yale University MIF modulators
US9540322B2 (en) 2008-08-18 2017-01-10 Yale University MIF modulators
EP2326631A4 (en) * 2008-08-18 2012-03-21 Univ Yale MIF MODULATORS
AU2009318783A1 (en) * 2008-11-20 2011-06-23 Panacea Biotec Ltd. Novel antimicrobials
CN107082790A (zh) 2009-02-03 2017-08-22 默沙东公司 一种噁唑烷酮化合物的晶型
JP5696142B2 (ja) 2009-06-26 2015-04-08 パナセア バイオテック リミテッド 新規アザビシクロヘキサン類
JP5996532B2 (ja) 2010-07-15 2016-09-21 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 有害生物防除剤としての新規複素環式化合物
UA112897C2 (uk) 2012-05-09 2016-11-10 Байєр Фарма Акцієнгезелльшафт Біциклічно заміщені урацили та їх застосування для лікування і/або профілактики захворювань
CA2939098A1 (en) 2014-02-21 2015-08-27 Micurx Pharmaceuticals, Inc. Water-soluble o-carbonyl phosphoramidate prodrugs for therapeutic administration
JP7205529B2 (ja) * 2018-02-26 2023-01-17 住友化学株式会社 オキサゾリジノン化合物の製造方法

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