JP2007510629A5 - - Google Patents

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Publication number
JP2007510629A5
JP2007510629A5 JP2006536645A JP2006536645A JP2007510629A5 JP 2007510629 A5 JP2007510629 A5 JP 2007510629A5 JP 2006536645 A JP2006536645 A JP 2006536645A JP 2006536645 A JP2006536645 A JP 2006536645A JP 2007510629 A5 JP2007510629 A5 JP 2007510629A5
Authority
JP
Japan
Prior art keywords
alkyl
oxadiazol
aryl
ethylsulfanylmethyl
phenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006536645A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007510629A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2004/032314 external-priority patent/WO2005040157A2/en
Publication of JP2007510629A publication Critical patent/JP2007510629A/ja
Publication of JP2007510629A5 publication Critical patent/JP2007510629A5/ja
Pending legal-status Critical Current

Links

JP2006536645A 2003-10-22 2004-10-21 新規ｍｃｈ受容体アンタゴニスト Pending JP2007510629A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51344903P 2003-10-22 2003-10-22
PCT/US2004/032314 WO2005040157A2 (en) 2003-10-22 2004-10-21 Novel mch receptor antagonists

Publications (2)

Publication Number Publication Date
JP2007510629A JP2007510629A (ja) 2007-04-26
JP2007510629A5 true JP2007510629A5 (enExample) 2007-11-22

Family

ID=34520102

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006536645A Pending JP2007510629A (ja) 2003-10-22 2004-10-21 新規ｍｃｈ受容体アンタゴニスト

Country Status (5)

Country Link
US (1) US20070135485A1 (enExample)
EP (1) EP1723126A2 (enExample)
JP (1) JP2007510629A (enExample)
CA (1) CA2542220A1 (enExample)
WO (1) WO2005040157A2 (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100418965C (zh) 2003-08-15 2008-09-17 万有制药株式会社 咪唑并吡啶衍生物
TW200613272A (en) * 2004-08-13 2006-05-01 Astrazeneca Ab Isoindolone compounds and their use as metabotropic glutamate receptor potentiators
JP5031745B2 (ja) * 2005-08-12 2012-09-26 アストラゼネカ アクチボラグ 代謝型グルタミン酸受容体増強性イソインドロン
US7807706B2 (en) 2005-08-12 2010-10-05 Astrazeneca Ab Metabotropic glutamate-receptor-potentiating isoindolones
CA2626747A1 (en) * 2005-10-26 2007-05-03 Boehringer Ingelheim International Gmbh (hetero)aryl compounds with mch antagonistic activity and medicaments comprising these compounds
JP5193878B2 (ja) 2005-12-21 2013-05-08 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Ｍｃｈ−１が媒介する疾患における使用のための新規な置換ピラジノン誘導体
US8492378B2 (en) 2006-08-03 2013-07-23 Takeda Pharmaceutical Company Limited GSK-3β inhibitor
EP2102208B1 (en) 2006-12-05 2014-04-23 Janssen Pharmaceutica NV Novel substituted diaza spiro pyridinone derivatives for use in mch-1 mediated diseases
TWI417100B (zh) 2007-06-07 2013-12-01 Astrazeneca Ab 二唑衍生物及其作為代謝型麩胺酸受體增效劑-８４２之用途
US7790760B2 (en) 2008-06-06 2010-09-07 Astrazeneca Ab Metabotropic glutamate receptor isoxazole ligands and their use as potentiators 286
US8586792B2 (en) 2011-12-28 2013-11-19 Divi's Laboratories Ltd. Process for the preparation of 4-iodo-3-nitrobenzamide
SG11201407999TA (en) * 2012-06-01 2015-01-29 Univ Singapore ICMT Inhibitors
US9310374B2 (en) 2012-11-16 2016-04-12 Redwood Bioscience, Inc. Hydrazinyl-indole compounds and methods for producing a conjugate
WO2014078733A1 (en) 2012-11-16 2014-05-22 The Regents Of The University Of California Pictet-spengler ligation for protein chemical modification
ES2908470T3 (es) 2015-11-09 2022-04-29 Scherer Technologies Llc R P Conjugados de anticuerpo anti-CD22-maitansina y métodos de uso de los mismos
US12441707B2 (en) 2019-12-30 2025-10-14 Tyra Biosciences, Inc. Indazole compounds
MX2023007793A (es) 2020-12-30 2023-09-22 Tyra Biosciences Inc Compuestos de indazol como inhibidores de cinasas.
JP7728367B2 (ja) 2021-06-14 2025-08-22 スコーピオン・セラピューティクス・インコーポレイテッド がんを処置するために使用され得る尿素誘導体

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL96891A0 (en) * 1990-01-17 1992-03-29 Merck Sharp & Dohme Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them
GB9407447D0 (en) * 1994-04-14 1994-06-08 Glaxo Group Ltd Chemical compounds
AU7074496A (en) 1995-09-18 1997-04-09 Ligand Pharmaceuticals Incorporated Ppar gamma antagonists for treating obesity
AU7692996A (en) 1995-12-01 1997-06-27 Ciba-Geigy Ag Receptor antagonists
AU7692696A (en) 1995-12-01 1997-06-27 Novartis Ag Heteroaryl derivatives
AU1328197A (en) 1995-12-01 1997-06-19 Synaptic Pharmaceutical Corporation Aryl sulfonamide and sulfamide derivatives and uses thereof
AU7626496A (en) 1995-12-01 1997-06-27 Ciba-Geigy Ag Heteroaryl compounds
AU7692896A (en) 1995-12-01 1997-06-27 Novartis Ag Quinazolin-2,4-diazirines as NPY receptor antagonist
ATE236137T1 (de) 1996-02-02 2003-04-15 Merck & Co Inc Heterocyclische verbindungen als antidiabetische mittel und für die behandlung von fettleibigkeit
CA2244831A1 (en) 1996-02-02 1997-08-07 John T. Olson Method of treating diabetes and related disease states
JP2002503202A (ja) 1996-02-02 2002-01-29 メルク エンド カンパニー インコーポレーテッド 抗糖尿病薬
WO1997028149A1 (en) 1996-02-02 1997-08-07 Merck & Co., Inc. Method for raising hdl cholesterol levels
GB9606805D0 (en) 1996-03-30 1996-06-05 Glaxo Wellcome Inc Medicaments
GB9706089D0 (en) * 1997-03-24 1997-05-14 Scherer Ltd R P Pharmaceutical composition
WO2001021577A2 (en) * 1999-09-20 2001-03-29 Takeda Chemical Industries, Ltd. Melanin concentrating hormone antagonist
AUPR118000A0 (en) * 2000-11-02 2000-11-23 Amrad Operations Pty. Limited Therapeutic molecules and methods
EP2258694A1 (en) * 2001-03-16 2010-12-08 Abbott Laboratories Amines as histamine-3 receptor ligands and their therapeutic applications
WO2003087046A1 (en) * 2002-04-09 2003-10-23 7Tm Pharma A/S Novel aminotetraline compounds for use in mch receptor related disorders
CA2484233A1 (en) * 2002-05-13 2003-11-27 Eli Lilly And Company Multicyclic compounds for use as melanin concentrating hormone antagonists in the treatment of obesity and diabetes

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