JP2003012668A5 - - Google Patents

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Publication number
JP2003012668A5
JP2003012668A5 JP2002126869A JP2002126869A JP2003012668A5 JP 2003012668 A5 JP2003012668 A5 JP 2003012668A5 JP 2002126869 A JP2002126869 A JP 2002126869A JP 2002126869 A JP2002126869 A JP 2002126869A JP 2003012668 A5 JP2003012668 A5 JP 2003012668A5
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JP
Japan
Prior art keywords
group
compound according
alkyl
hydrogen atom
alkyl group
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Application number
JP2002126869A
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English (en)
Japanese (ja)
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JP3602513B2 (ja
JP2003012668A (ja
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Application filed filed Critical
Priority to JP2002126869A priority Critical patent/JP3602513B2/ja
Priority claimed from JP2002126869A external-priority patent/JP3602513B2/ja
Publication of JP2003012668A publication Critical patent/JP2003012668A/ja
Application granted granted Critical
Publication of JP3602513B2 publication Critical patent/JP3602513B2/ja
Publication of JP2003012668A5 publication Critical patent/JP2003012668A5/ja
Priority to NL300927C priority patent/NL300927I9/nl
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2002126869A 2001-04-27 2002-04-26 アゾリル基を有するキノリン誘導体およびキナゾリン誘導体 Expired - Lifetime JP3602513B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2002126869A JP3602513B2 (ja) 2001-04-27 2002-04-26 アゾリル基を有するキノリン誘導体およびキナゾリン誘導体
NL300927C NL300927I9 (nl) 2001-04-27 2018-01-31 Tivozanib of een zout, solvaat of hydraat ervan, in het bijzonder het hydrochloride-monohydraat

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2001-132775 2001-04-27
JP2001132775 2001-04-27
JP2002126869A JP3602513B2 (ja) 2001-04-27 2002-04-26 アゾリル基を有するキノリン誘導体およびキナゾリン誘導体

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2004101164A Division JP2004224800A (ja) 2001-04-27 2004-03-30 アゾリル基を有するキノリン誘導体およびキナゾリン誘導体

Publications (3)

Publication Number Publication Date
JP2003012668A JP2003012668A (ja) 2003-01-15
JP3602513B2 JP3602513B2 (ja) 2004-12-15
JP2003012668A5 true JP2003012668A5 (enExample) 2004-12-16

Family

ID=26614489

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002126869A Expired - Lifetime JP3602513B2 (ja) 2001-04-27 2002-04-26 アゾリル基を有するキノリン誘導体およびキナゾリン誘導体

Country Status (1)

Country Link
JP (1) JP3602513B2 (enExample)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8815241B2 (en) 2005-11-07 2014-08-26 Eisai R&D Management Co., Ltd. Use of combination of anti-angiogenic substance and c-kit kinase inhibitor
US8952035B2 (en) 2007-11-09 2015-02-10 Eisai R&D Management Co., Ltd. Combination of anti-angiogenic substance and anti-tumor platinum complex
US8962650B2 (en) 2011-04-18 2015-02-24 Eisai R&D Management Co., Ltd. Therapeutic agent for tumor
US8969344B2 (en) 2005-08-02 2015-03-03 Eisai R&D Management Co., Ltd. Method for assay on the effect of vascularization inhibitor
US9006256B2 (en) 2006-05-18 2015-04-14 Eisai R&D Management Co., Ltd. Antitumor agent for thyroid cancer
US9012458B2 (en) 2010-06-25 2015-04-21 Eisai R&D Management Co., Ltd. Antitumor agent using compounds having kinase inhibitory effect in combination
US9504746B2 (en) 2004-09-17 2016-11-29 Eisai R&D Management Co., Ltd. Pharmaceutical compositions of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1447405A4 (en) * 2001-10-17 2005-01-12 Kirin Brewery CHINOLIN OR CHINAZOLINE DERIVATIVES THAT PREVENT THE AUTOPHOSPHORYLATION OF RECEPTORS FOR THE FIBROBLAST GROWTH FACTOR
EP1604665B1 (en) 2003-03-10 2011-05-11 Eisai R&D Management Co., Ltd. C-kit kinase inhibitor
CN101511793B (zh) 2006-08-28 2011-08-03 卫材R&D管理有限公司 针对未分化型胃癌的抗肿瘤剂
JP5319306B2 (ja) 2007-01-29 2013-10-16 エーザイ・アール・アンド・ディー・マネジメント株式会社 未分化型胃癌治療用組成物
HUE026957T2 (en) 2009-08-19 2016-07-28 Eisai R&D Man Co Ltd A pharmaceutical composition comprising a quinoline derivative
ES2841809T3 (es) 2011-06-03 2021-07-09 Eisai R&D Man Co Ltd Biomarcadores para pronosticar y evaluar el grado de respuesta de sujetos con cáncer de tiroides y de riñón a compuestos de lenvatinib
AU2013364953A1 (en) 2012-12-21 2015-04-30 Eisai R&D Management Co., Ltd. Amorphous form of quinoline derivative, and method for producing same
CA2912219C (en) 2013-05-14 2021-11-16 Eisai R&D Management Co., Ltd. Biomarkers for predicting and assessing responsiveness of endometrial cancer subjects to lenvatinib compounds
EP4089076A1 (en) 2014-08-28 2022-11-16 Eisai R&D Management Co., Ltd. High-purity quinoline derivative and method for manufacturing same
KR102763349B1 (ko) 2015-02-25 2025-02-07 에자이 알앤드디 매니지먼트 가부시키가이샤 퀴놀린 유도체의 고미 억제 방법
AU2015384801B2 (en) 2015-03-04 2022-01-06 Eisai R&D Management Co., Ltd. Combination of a PD-1 antagonist and a VEGFR/FGFR/RET tyrosine kinase inhibitor for treating cancer
RU2729936C2 (ru) 2015-06-16 2020-08-13 Эйсай Ар Энд Ди Менеджмент Ко., Лтд. Противораковое средство
SG11201801083UA (en) 2015-08-20 2018-03-28 Eisai R&D Man Co Ltd Tumor therapeutic agent
MX382732B (es) 2016-09-13 2025-03-13 Kyowa Kirin Co Ltd Composición farmacéutica.
KR102539920B1 (ko) 2017-02-08 2023-06-05 에자이 알앤드디 매니지먼트 가부시키가이샤 종양-치료용 약제학적 조성물
SG11201910100PA (en) 2017-05-16 2019-11-28 Eisai R&D Man Co Ltd Treatment of hepatocellular carcinoma

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9504746B2 (en) 2004-09-17 2016-11-29 Eisai R&D Management Co., Ltd. Pharmaceutical compositions of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide
US8969344B2 (en) 2005-08-02 2015-03-03 Eisai R&D Management Co., Ltd. Method for assay on the effect of vascularization inhibitor
US9006240B2 (en) 2005-08-02 2015-04-14 Eisai R&D Management Co., Ltd. Method for assay on the effect of vascularization inhibitor
US8815241B2 (en) 2005-11-07 2014-08-26 Eisai R&D Management Co., Ltd. Use of combination of anti-angiogenic substance and c-kit kinase inhibitor
US9006256B2 (en) 2006-05-18 2015-04-14 Eisai R&D Management Co., Ltd. Antitumor agent for thyroid cancer
US8952035B2 (en) 2007-11-09 2015-02-10 Eisai R&D Management Co., Ltd. Combination of anti-angiogenic substance and anti-tumor platinum complex
US9012458B2 (en) 2010-06-25 2015-04-21 Eisai R&D Management Co., Ltd. Antitumor agent using compounds having kinase inhibitory effect in combination
US8962650B2 (en) 2011-04-18 2015-02-24 Eisai R&D Management Co., Ltd. Therapeutic agent for tumor

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