IN2015DN01119A - - Google Patents

Info

Publication number
IN2015DN01119A
IN2015DN01119A IN1119DEN2015A IN2015DN01119A IN 2015DN01119 A IN2015DN01119 A IN 2015DN01119A IN 1119DEN2015 A IN1119DEN2015 A IN 1119DEN2015A IN 2015DN01119 A IN2015DN01119 A IN 2015DN01119A
Authority
IN
India
Prior art keywords
compounds
disclosed
methods
intermediates
synthesis
Prior art date
Application number
Other languages
English (en)
Inventor
Ende Christopher William Am
Michael Eric Green
Douglas Scott Johnson
Gregory Wayne Kauffman
Christopher John Odonnell
Nandini Chaturbhai Patel
Martin Youngjin Pettersson
Antonia Friederike Stepan
Cory Michael Stiff
Chakrapani Subramanyam
Tuan Phong Tran
Patrick Robert Verhoest
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IN2015DN01119A publication Critical patent/IN2015DN01119A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Epidemiology (AREA)
IN1119DEN2015 2012-09-21 2013-09-06 IN2015DN01119A (en:Method)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261703969P 2012-09-21 2012-09-21
PCT/IB2013/058347 WO2014045156A1 (en) 2012-09-21 2013-09-06 Novel bicyclic pyridinones

Publications (1)

Publication Number Publication Date
IN2015DN01119A true IN2015DN01119A (en:Method) 2015-06-26

Family

ID=49585452

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1119DEN2015 IN2015DN01119A (en:Method) 2012-09-21 2013-09-06

Country Status (46)

Country Link
US (3) US8916564B2 (en:Method)
EP (1) EP2897956B1 (en:Method)
JP (1) JP5844018B2 (en:Method)
KR (1) KR101725696B1 (en:Method)
CN (1) CN104662021B (en:Method)
AP (1) AP2015008277A0 (en:Method)
AR (1) AR092628A1 (en:Method)
AU (1) AU2013319845B2 (en:Method)
BR (1) BR112015006436A2 (en:Method)
CA (1) CA2882386C (en:Method)
CL (1) CL2015000717A1 (en:Method)
CR (1) CR20150053A (en:Method)
CU (1) CU20150021A7 (en:Method)
CY (1) CY1118662T1 (en:Method)
DK (1) DK2897956T3 (en:Method)
DO (1) DOP2015000069A (en:Method)
EA (1) EA026668B1 (en:Method)
EC (1) ECSP15015594A (en:Method)
ES (1) ES2609987T3 (en:Method)
GE (1) GEP201706659B (en:Method)
GT (1) GT201500069A (en:Method)
HR (1) HRP20161558T1 (en:Method)
HU (1) HUE031248T2 (en:Method)
IL (1) IL237163A (en:Method)
IN (1) IN2015DN01119A (en:Method)
LT (1) LT2897956T (en:Method)
MA (1) MA37886B1 (en:Method)
MD (1) MD4583B1 (en:Method)
ME (1) ME02571B (en:Method)
MX (1) MX360599B (en:Method)
MY (1) MY181891A (en:Method)
NI (1) NI201500038A (en:Method)
NZ (1) NZ704863A (en:Method)
PE (1) PE20150686A1 (en:Method)
PH (1) PH12015500376B1 (en:Method)
PL (1) PL2897956T3 (en:Method)
PT (1) PT2897956T (en:Method)
RS (1) RS55426B1 (en:Method)
SG (1) SG11201501074WA (en:Method)
SI (1) SI2897956T1 (en:Method)
TN (1) TN2015000084A1 (en:Method)
TW (1) TWI500616B (en:Method)
UA (1) UA110688C2 (en:Method)
UY (1) UY35039A (en:Method)
WO (1) WO2014045156A1 (en:Method)
ZA (1) ZA201501195B (en:Method)

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KR102171710B1 (ko) 2013-01-17 2020-10-30 얀센 파마슈티카 엔.브이. 감마 세크레타제 조절 인자로서의 신규 치환 피리도-피페라지논 유도체
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KR20190098998A (ko) 2016-12-16 2019-08-23 파이프라인 테라퓨틱스, 아이엔씨. 달팽이관 시냅스질환의 치료 방법
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CN113402490B (zh) * 2021-03-29 2023-01-03 白银京宇新药业有限公司 一种1,2,6,7-四氢-8H-茚并[5,4-b]呋喃-8-酮的制备方法
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