IL245844A0 - Converted benzamides and methods of using them - Google Patents
Converted benzamides and methods of using themInfo
- Publication number
- IL245844A0 IL245844A0 IL245844A IL24584416A IL245844A0 IL 245844 A0 IL245844 A0 IL 245844A0 IL 245844 A IL245844 A IL 245844A IL 24584416 A IL24584416 A IL 24584416A IL 245844 A0 IL245844 A0 IL 245844A0
- Authority
- IL
- Israel
- Prior art keywords
- methods
- substituted benzamides
- benzamides
- substituted
- Prior art date
Links
- 229940054066 benzamide antipsychotics Drugs 0.000 title 1
- 150000003936 benzamides Chemical class 0.000 title 1
Classifications
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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| WO2013177224A1 (en) * | 2012-05-22 | 2013-11-28 | Genentech, Inc. | N-substituted benzamides and their use in the treatment of pain |
| BR112015000187A2 (pt) | 2012-07-06 | 2017-06-27 | Genentech Inc | benzamidas substituídas com n e métodos de uso das mesmas |
| BR112015022488A2 (pt) | 2013-03-14 | 2017-07-18 | Genentech Inc | triazolopiridinas substituídas e métodos de uso das mesmas |
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| JP6383418B2 (ja) | 2013-11-27 | 2018-08-29 | ジェネンテック, インコーポレイテッド | 置換ベンズアミド及びその使用方法 |
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| CN107428683B (zh) * | 2015-02-04 | 2020-06-02 | 上海海雁医药科技有限公司 | 杂环取代的n-磺酰基苯甲酰胺衍生物、其制法与医药上的用途 |
| CR20170591A (es) | 2015-05-22 | 2018-05-07 | Genentech Inc | Benzamidas sustituidas y métodos para utilizarlas |
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| PE20181003A1 (es) | 2015-09-28 | 2018-06-26 | Genentech Inc | Compuestos terapeuticos y sus metodos de uso |
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| WO2017091592A1 (en) * | 2015-11-25 | 2017-06-01 | Genentech, Inc. | Substituted benzamides useful as sodium channel blockers |
| WO2017095723A1 (en) * | 2015-11-30 | 2017-06-08 | Merck Sharp & Dohme Corp. | Aryl acylsulfonamides as blt1 antagonists |
| EA201891313A1 (ru) | 2015-12-18 | 2018-11-30 | Мерк Шарп И Доум Корп. | Замещенные гидроксиалкиламинами и гидроксициклоалкиламинами соединения диаминарилсульфонамидов с избирательной активностью в потенциалзависимых натриевых каналах |
| CN108430969B (zh) * | 2016-02-03 | 2020-06-02 | 上海海雁医药科技有限公司 | 杂环取代的n-磺酰基苯甲酰胺衍生物、其制法与医药上的用途 |
| EP3436432B1 (en) | 2016-03-30 | 2021-01-27 | Genentech, Inc. | Substituted benzamides and methods of use thereof |
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| TN2019000290A1 (en) | 2017-03-20 | 2021-05-07 | Forma Therapeutics Inc | Pyrrolopyrrole compositions as pyruvate kinase (pkr) activators |
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| WO2019019851A1 (zh) * | 2017-07-24 | 2019-01-31 | 上海海雁医药科技有限公司 | 钠离子通道抑制剂及其药学上可接受的盐和多晶型物及其应用 |
| WO2019045035A1 (en) | 2017-08-31 | 2019-03-07 | Raqualia Pharma Inc. | BIARYLOXY DERIVATIVES AS TTX-S BLOCKERS |
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| WO2019165290A1 (en) | 2018-02-26 | 2019-08-29 | Genentech, Inc. | Pyridine-sulfonamide compounds and their use against pain and related conditions |
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| JP7371029B2 (ja) | 2018-06-13 | 2023-10-30 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | ベンゼンスルホンアミド化合物および治療剤としてのその使用 |
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| JP7450610B2 (ja) | 2018-09-19 | 2024-03-15 | ノヴォ・ノルディスク・ヘルス・ケア・アーゲー | ピルビン酸キナーゼrの活性化 |
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| WO2021132577A1 (ja) * | 2019-12-27 | 2021-07-01 | 日本たばこ産業株式会社 | アシルスルファミド化合物及びその医薬用途 |
| CN111303120A (zh) * | 2020-03-14 | 2020-06-19 | 江巨东 | 一种盐酸法舒地尔的制备方法 |
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| CN115215787A (zh) * | 2021-04-19 | 2022-10-21 | 中国科学院上海药物研究所 | 生长抑素受体5拮抗剂及其用途 |
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-
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- 2014-11-26 KR KR1020167016643A patent/KR20160090846A/ko not_active Withdrawn
- 2014-11-26 AU AU2014356967A patent/AU2014356967A1/en not_active Abandoned
- 2014-11-26 EP EP14865855.2A patent/EP3074377B1/en active Active
- 2014-11-26 MX MX2016006936A patent/MX2016006936A/es unknown
- 2014-11-26 EA EA201691085A patent/EA201691085A1/ru unknown
- 2014-11-26 PE PE2016000696A patent/PE20161247A1/es not_active Application Discontinuation
- 2014-11-26 CA CA2931732A patent/CA2931732A1/en not_active Abandoned
- 2014-11-26 CR CR20160296A patent/CR20160296A/es unknown
- 2014-11-26 EP EP18197734.9A patent/EP3450428A1/en not_active Withdrawn
- 2014-11-26 CN CN201480064734.4A patent/CN105793238B/zh not_active Expired - Fee Related
- 2014-11-26 WO PCT/CN2014/092269 patent/WO2015078374A1/en not_active Ceased
- 2014-11-27 TW TW103141262A patent/TWI560180B/zh not_active IP Right Cessation
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2015
- 2015-01-22 US US14/603,273 patent/US9546164B2/en not_active Expired - Fee Related
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2016
- 2016-05-25 IL IL245844A patent/IL245844A0/en unknown
- 2016-05-26 CL CL2016001287A patent/CL2016001287A1/es unknown
- 2016-05-27 PH PH12016501007A patent/PH12016501007A1/en unknown
- 2016-09-23 US US15/275,131 patent/US9694002B2/en not_active Expired - Fee Related
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2018
- 2018-08-03 JP JP2018146542A patent/JP2018188466A/ja active Pending
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2019
- 2019-04-22 US US16/390,957 patent/US20200108054A1/en not_active Abandoned
- 2019-11-07 US US16/677,487 patent/US20210093618A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN105793238A (zh) | 2016-07-20 |
| JP2018188466A (ja) | 2018-11-29 |
| KR20160090846A (ko) | 2016-08-01 |
| CL2016001287A1 (es) | 2018-03-16 |
| HK1223913A1 (zh) | 2017-08-11 |
| US20200108054A1 (en) | 2020-04-09 |
| US20170087136A1 (en) | 2017-03-30 |
| JP6383418B2 (ja) | 2018-08-29 |
| CN105793238B (zh) | 2019-12-24 |
| MX2016006936A (es) | 2016-10-05 |
| EP3074377B1 (en) | 2018-10-17 |
| TWI560180B (en) | 2016-12-01 |
| US9546164B2 (en) | 2017-01-17 |
| US20150252038A1 (en) | 2015-09-10 |
| PE20161247A1 (es) | 2016-11-30 |
| PH12016501007A1 (en) | 2016-07-18 |
| CA2931732A1 (en) | 2015-06-04 |
| EA201691085A1 (ru) | 2017-02-28 |
| TW201533021A (zh) | 2015-09-01 |
| WO2015078374A1 (en) | 2015-06-04 |
| JP2017504571A (ja) | 2017-02-09 |
| AU2014356967A1 (en) | 2016-07-07 |
| US20210093618A1 (en) | 2021-04-01 |
| EP3074377A4 (en) | 2017-04-19 |
| EP3074377A1 (en) | 2016-10-05 |
| US9694002B2 (en) | 2017-07-04 |
| CR20160296A (es) | 2016-09-20 |
| EP3450428A1 (en) | 2019-03-06 |
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