CA2931732A1 - Substituted benzamides and methods of use thereof - Google Patents

Substituted benzamides and methods of use thereof Download PDF

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Publication number
CA2931732A1
CA2931732A1 CA2931732A CA2931732A CA2931732A1 CA 2931732 A1 CA2931732 A1 CA 2931732A1 CA 2931732 A CA2931732 A CA 2931732A CA 2931732 A CA2931732 A CA 2931732A CA 2931732 A1 CA2931732 A1 CA 2931732A1
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CA
Canada
Prior art keywords
alkyl
group
haloalkyl
compound
optionally substituted
Prior art date
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Abandoned
Application number
CA2931732A
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English (en)
French (fr)
Inventor
Jean-Christophe ANDREZ
Paul Robert BICHLER
Chien-An Chen
Sultan Chowdhury
Shannon Marie DECKER
Christoph Martin Dehnhardt
Thilo FOCKEN
Michael Edward Grimwood
Ivan William Hemeon
Qi Jia
Jun Li
Zhiguo Liu
Daniel F. Ortwine
Brian Safina
Daniel Sutherlin
Tao Sheng
Shaoyi Sun
Andrew D. White
Michael Scott Wilson
Alla Yurevna Zenova
Jiuxiang Zhu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Xenon Pharmaceuticals Inc
Genentech Inc
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Xenon Pharmaceuticals Inc
Genentech Inc
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Publication date
Application filed by Xenon Pharmaceuticals Inc, Genentech Inc filed Critical Xenon Pharmaceuticals Inc
Publication of CA2931732A1 publication Critical patent/CA2931732A1/en
Abandoned legal-status Critical Current

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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