IL147803A0 - 28-epirapalogs - Google Patents

28-epirapalogs

Info

Publication number
IL147803A0
IL147803A0 IL14780300A IL14780300A IL147803A0 IL 147803 A0 IL147803 A0 IL 147803A0 IL 14780300 A IL14780300 A IL 14780300A IL 14780300 A IL14780300 A IL 14780300A IL 147803 A0 IL147803 A0 IL 147803A0
Authority
IL
Israel
Prior art keywords
epirapalogs
epirapamycin
analogs
disclosed
methods
Prior art date
Application number
IL14780300A
Other languages
English (en)
Original Assignee
Ariad Gene Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ariad Gene Therapeutics Inc filed Critical Ariad Gene Therapeutics Inc
Publication of IL147803A0 publication Critical patent/IL147803A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K48/00Medicinal preparations containing genetic material which is inserted into cells of the living body to treat genetic diseases; Gene therapy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/10Transferases (2.)
    • C12N9/12Transferases (2.) transferring phosphorus containing groups, e.g. kinases (2.7)
    • C12N9/1205Phosphotransferases with an alcohol group as acceptor (2.7.1), e.g. protein kinases
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2319/00Fusion polypeptide

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Biotechnology (AREA)
  • Zoology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Wood Science & Technology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Microbiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Saccharide Compounds (AREA)
IL14780300A 1999-08-24 2000-08-24 28-epirapalogs IL147803A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15044799P 1999-08-24 1999-08-24
PCT/US2000/023334 WO2001014387A1 (en) 1999-08-24 2000-08-24 28-epirapalogs

Publications (1)

Publication Number Publication Date
IL147803A0 true IL147803A0 (en) 2002-08-14

Family

ID=22534571

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14780300A IL147803A0 (en) 1999-08-24 2000-08-24 28-epirapalogs
IL147803A IL147803A (en) 1999-08-24 2002-01-23 28-epi-rapamycin derivatives, their preparation, pharmaceutical compositions containing them and preparation of compositions for in vitro and pharmaceutical applications

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL147803A IL147803A (en) 1999-08-24 2002-01-23 28-epi-rapamycin derivatives, their preparation, pharmaceutical compositions containing them and preparation of compositions for in vitro and pharmaceutical applications

Country Status (10)

Country Link
US (1) US7196192B2 (xx)
EP (1) EP1212331B1 (xx)
CN (1) CN1293081C (xx)
AT (1) ATE264863T1 (xx)
AU (1) AU783158B2 (xx)
CA (1) CA2383451A1 (xx)
DE (1) DE60010098T2 (xx)
ES (1) ES2219388T3 (xx)
IL (2) IL147803A0 (xx)
WO (1) WO2001014387A1 (xx)

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* Cited by examiner, † Cited by third party
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