IL147641A0 - Beta-carboline pharmaceutical compositions - Google Patents

Beta-carboline pharmaceutical compositions

Info

Publication number
IL147641A0
IL147641A0 IL14764100A IL14764100A IL147641A0 IL 147641 A0 IL147641 A0 IL 147641A0 IL 14764100 A IL14764100 A IL 14764100A IL 14764100 A IL14764100 A IL 14764100A IL 147641 A0 IL147641 A0 IL 147641A0
Authority
IL
Israel
Prior art keywords
beta
pharmaceutical compositions
carboline
carboline pharmaceutical
disintegrant
Prior art date
Application number
IL14764100A
Other languages
English (en)
Original Assignee
Lilly Icos Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22519593&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL147641(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Icos Llc filed Critical Lilly Icos Llc
Publication of IL147641A0 publication Critical patent/IL147641A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL14764100A 1999-08-03 2000-04-26 Beta-carboline pharmaceutical compositions IL147641A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14692499P 1999-08-03 1999-08-03
PCT/US2000/011130 WO2001008686A1 (en) 1999-08-03 2000-04-26 Beta-carboline pharmaceutical compositions

Publications (1)

Publication Number Publication Date
IL147641A0 true IL147641A0 (en) 2002-08-14

Family

ID=22519593

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14764100A IL147641A0 (en) 1999-08-03 2000-04-26 Beta-carboline pharmaceutical compositions
IL147641A IL147641A (en) 1999-08-03 2002-01-15 Pharmaceutical preparations containing (R6, aR12) - 2,3,4,5,6,7,12, a12 - hexahydro - 2 - methyl - 6 - (3, 4 - methylene dioxyphenyl) pyrazino - [2 ', 1': 6, 1] Pyrido [3, 4 –b] Indole - 1, 4– Dion

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL147641A IL147641A (en) 1999-08-03 2002-01-15 Pharmaceutical preparations containing (R6, aR12) - 2,3,4,5,6,7,12, a12 - hexahydro - 2 - methyl - 6 - (3, 4 - methylene dioxyphenyl) pyrazino - [2 ', 1': 6, 1] Pyrido [3, 4 –b] Indole - 1, 4– Dion

Country Status (29)

Country Link
US (2) US7182958B1 (sk)
EP (3) EP1200091B1 (sk)
JP (2) JP2003505509A (sk)
KR (2) KR20060093355A (sk)
CN (1) CN1213754C (sk)
AT (1) ATE399554T1 (sk)
AU (2) AU776722B2 (sk)
BR (1) BR0012863A (sk)
CA (1) CA2379948C (sk)
CZ (1) CZ304624B6 (sk)
DE (1) DE60039357D1 (sk)
DK (1) DK1200090T3 (sk)
DZ (1) DZ3179A1 (sk)
EA (1) EA004872B1 (sk)
ES (2) ES2310166T3 (sk)
HK (1) HK1044277B (sk)
HR (1) HRP20020090B1 (sk)
HU (1) HU230660B1 (sk)
IL (2) IL147641A0 (sk)
MX (1) MXPA02001196A (sk)
NO (1) NO321649B1 (sk)
NZ (1) NZ516616A (sk)
PL (1) PL199137B1 (sk)
PT (1) PT1200090E (sk)
SI (1) SI1200090T1 (sk)
SK (1) SK287869B6 (sk)
UA (1) UA72922C2 (sk)
WO (2) WO2001008687A1 (sk)
ZA (1) ZA200200823B (sk)

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EP3157530A4 (en) 2014-06-17 2018-01-17 The Research Foundation for The State University of New York Ship inhibition to induce expression of granulocyte colony stimulating factor in a subject
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KR102646431B1 (ko) 2017-09-29 2024-03-12 한미약품 주식회사 생산성 및 균일성이 개선된 타다라필을 함유하는 고형제제 및 그 제조방법
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Also Published As

Publication number Publication date
EA200200118A1 (ru) 2002-06-27
HUP0202513A3 (en) 2004-06-28
DK1200090T3 (da) 2013-11-25
EP1200090B1 (en) 2013-09-11
US7182958B1 (en) 2007-02-27
NO20020532L (no) 2002-03-26
ATE399554T1 (de) 2008-07-15
WO2001008687A1 (en) 2001-02-08
EP1200091B1 (en) 2008-07-02
HUP0202513A2 (en) 2002-10-28
AU4491200A (en) 2001-02-19
KR100738861B1 (ko) 2007-07-16
AU776722B2 (en) 2004-09-16
ES2435816T3 (es) 2013-12-23
EA004872B1 (ru) 2004-08-26
CZ2002386A3 (cs) 2002-07-17
CZ304624B6 (cs) 2014-08-13
EP2338491A2 (en) 2011-06-29
JP2010163464A (ja) 2010-07-29
HU230660B1 (hu) 2017-06-28
US6841167B1 (en) 2005-01-11
PT1200090E (pt) 2013-11-25
JP2003505509A (ja) 2003-02-12
AU4490900A (en) 2001-02-19
DE60039357D1 (de) 2008-08-14
EP1200091A1 (en) 2002-05-02
HK1044277B (zh) 2014-02-28
HRP20020090A2 (en) 2003-12-31
BR0012863A (pt) 2002-04-16
NO20020532D0 (no) 2002-02-01
MXPA02001196A (es) 2003-02-12
NO321649B1 (no) 2006-06-19
ZA200200823B (en) 2003-04-30
EP2338491A3 (en) 2011-11-30
CA2379948C (en) 2008-03-25
DZ3179A1 (fr) 2001-02-08
CN1213754C (zh) 2005-08-10
KR20020014843A (ko) 2002-02-25
EP1200090A1 (en) 2002-05-02
CA2379948A1 (en) 2001-02-08
UA72922C2 (uk) 2005-05-16
CN1365282A (zh) 2002-08-21
SK1732002A3 (en) 2002-05-09
HRP20020090B1 (hr) 2014-03-28
IL147641A (en) 2007-12-03
SK287869B6 (sk) 2012-02-03
PL199137B1 (pl) 2008-08-29
PL353304A1 (en) 2003-11-03
ES2310166T3 (es) 2009-01-01
KR20060093355A (ko) 2006-08-24
NZ516616A (en) 2003-07-25
WO2001008686A1 (en) 2001-02-08
SI1200090T1 (sl) 2013-12-31

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