IL138469A0 - Caspase inhibitors and pharmaceutical compositions containing the same - Google Patents

Caspase inhibitors and pharmaceutical compositions containing the same

Info

Publication number
IL138469A0
IL138469A0 IL138469??A IL13846999A IL138469A0 IL 138469 A0 IL138469 A0 IL 138469A0 IL 13846999 A IL13846999 A IL 13846999A IL 138469 A0 IL138469 A0 IL 138469A0
Authority
IL
Israel
Prior art keywords
same
pharmaceutical compositions
compositions containing
caspase inhibitors
caspase
Prior art date
Application number
IL138469??A
Other languages
English (en)
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of IL138469A0 publication Critical patent/IL138469A0/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
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  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Virology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
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  • Dermatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Urology & Nephrology (AREA)
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IL138469??A 1998-03-19 1999-03-19 Caspase inhibitors and pharmaceutical compositions containing the same IL138469A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7877098P 1998-03-19 1998-03-19
PCT/US1999/005919 WO1999047545A2 (en) 1998-03-19 1999-03-19 Inhibitors of caspases

Publications (1)

Publication Number Publication Date
IL138469A0 true IL138469A0 (en) 2001-10-31

Family

ID=22146109

Family Applications (3)

Application Number Title Priority Date Filing Date
IL138469??A IL138469A0 (en) 1998-03-19 1999-03-19 Caspase inhibitors and pharmaceutical compositions containing the same
IL138469A IL138469A (en) 1998-03-19 2000-09-14 Caspase inhibitors and pharmaceutical compositions containing the same
IL206621A IL206621A0 (en) 1998-03-19 2010-06-24 Caspase inhibitors and pharmaceutical compositions containing the same

Family Applications After (2)

Application Number Title Priority Date Filing Date
IL138469A IL138469A (en) 1998-03-19 2000-09-14 Caspase inhibitors and pharmaceutical compositions containing the same
IL206621A IL206621A0 (en) 1998-03-19 2010-06-24 Caspase inhibitors and pharmaceutical compositions containing the same

Country Status (34)

Country Link
US (3) US6531474B1 (ru)
EP (6) EP2261234A3 (ru)
JP (3) JP4594520B2 (ru)
KR (2) KR100928878B1 (ru)
CN (1) CN1321129C (ru)
AP (1) AP2000001919A0 (ru)
AR (1) AR019011A1 (ru)
AT (1) ATE410439T1 (ru)
AU (1) AU769033B2 (ru)
BG (1) BG104863A (ru)
BR (2) BRPI9909660B8 (ru)
CA (1) CA2324226C (ru)
CZ (1) CZ302281B6 (ru)
DE (1) DE69939689D1 (ru)
DK (1) DK1064298T3 (ru)
ES (1) ES2315010T3 (ru)
GE (1) GEP20043163B (ru)
HK (1) HK1035733A1 (ru)
HU (1) HU227920B1 (ru)
ID (1) ID27002A (ru)
IL (3) IL138469A0 (ru)
IS (1) IS5622A (ru)
NO (1) NO331829B1 (ru)
NZ (2) NZ506963A (ru)
PL (1) PL204619B1 (ru)
PT (1) PT1064298E (ru)
RU (1) RU2274642C2 (ru)
SI (1) SI1064298T1 (ru)
SK (1) SK286736B6 (ru)
TR (1) TR200103406T2 (ru)
TW (1) TWI243828B (ru)
UA (2) UA74133C2 (ru)
WO (1) WO1999047545A2 (ru)
ZA (1) ZA200004652B (ru)

Families Citing this family (77)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI1064298T1 (sl) * 1998-03-19 2009-02-28 Vertex Pharma Inhibitorji kaspaz
US7157430B2 (en) 1998-10-22 2007-01-02 Idun Pharmaceuticals, Inc. (Substituted)acyl dipeptidyl inhibitors of the ICE/CED-3 family of cysteine proteases
US6242422B1 (en) * 1998-10-22 2001-06-05 Idun Pharmacueticals, Inc. (Substituted)Acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
US6720415B2 (en) 1998-12-02 2004-04-13 Princeton University Compositions and methods for regulating bacterial pathogenesis
US7326542B2 (en) 1998-12-02 2008-02-05 Princeton University Compositions and methods for regulating bacterial pathogenesis
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UA74133C2 (ru) 2005-11-15
EP1064298A2 (en) 2001-01-03
EP2261233A3 (en) 2011-04-20
HK1035733A1 (en) 2001-12-07
EP2261235A2 (en) 2010-12-15
WO1999047545A2 (en) 1999-09-23
US20090048226A1 (en) 2009-02-19
EP2261234A2 (en) 2010-12-15
JP4594520B2 (ja) 2010-12-08

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