IL105078A - Pharmaceutical compositions containing 17-(3-pyridyl)- substituted steroids and some new compounds of this type - Google Patents

Pharmaceutical compositions containing 17-(3-pyridyl)- substituted steroids and some new compounds of this type

Info

Publication number
IL105078A
IL105078A IL105078A IL10507893A IL105078A IL 105078 A IL105078 A IL 105078A IL 105078 A IL105078 A IL 105078A IL 10507893 A IL10507893 A IL 10507893A IL 105078 A IL105078 A IL 105078A
Authority
IL
Israel
Prior art keywords
carbon atoms
pyridyl
beta
hydrogen atom
alkyl
Prior art date
Application number
IL105078A
Other languages
English (en)
Other versions
IL105078A0 (en
Original Assignee
British Tech Group
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26300621&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL105078(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB929207057A external-priority patent/GB9207057D0/en
Priority claimed from GB929224880A external-priority patent/GB9224880D0/en
Application filed by British Tech Group filed Critical British Tech Group
Publication of IL105078A0 publication Critical patent/IL105078A0/xx
Publication of IL105078A publication Critical patent/IL105078A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/005—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 16 (17)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
IL105078A 1992-03-31 1993-03-16 Pharmaceutical compositions containing 17-(3-pyridyl)- substituted steroids and some new compounds of this type IL105078A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929207057A GB9207057D0 (en) 1992-03-31 1992-03-31 Steroids
GB929224880A GB9224880D0 (en) 1992-11-27 1992-11-27 Steroids

Publications (2)

Publication Number Publication Date
IL105078A0 IL105078A0 (en) 1993-07-08
IL105078A true IL105078A (en) 1997-11-20

Family

ID=26300621

Family Applications (1)

Application Number Title Priority Date Filing Date
IL105078A IL105078A (en) 1992-03-31 1993-03-16 Pharmaceutical compositions containing 17-(3-pyridyl)- substituted steroids and some new compounds of this type

Country Status (16)

Country Link
EP (1) EP0633893B1 (ko)
JP (1) JP2742331B2 (ko)
KR (1) KR100235135B1 (ko)
AT (1) ATE186913T1 (ko)
AU (1) AU668144B2 (ko)
CA (1) CA2132449C (ko)
CZ (1) CZ287434B6 (ko)
DE (2) DE69327096T2 (ko)
DK (1) DK0633893T3 (ko)
ES (1) ES2138618T3 (ko)
GB (1) GB2265624B (ko)
IL (1) IL105078A (ko)
LU (1) LU91911I2 (ko)
MX (1) MX9301525A (ko)
NZ (1) NZ249911A (ko)
WO (1) WO1993020097A1 (ko)

Families Citing this family (82)

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AU2002214320A1 (en) 2000-11-20 2002-05-27 Takeda Chemical Industries Ltd. Imidazole derivatives, process for their preparation and their use
AU2002221080A1 (en) 2000-12-08 2002-06-18 Masami Kusaka Substituted thiazole derivatives bearing 3-pyridyl groups, process for preparingthe same and use thereof
EP1463505A2 (en) * 2001-12-13 2004-10-06 Abbott Laboratories 3-(phenyl-alkoxy)-5-(phenyl)-pyridine derivatives and related compounds as kinase inhibitors for the treatment of cancer
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WO2014009436A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Nanosuspension of abiraterone acetate
WO2014009437A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Oxidation stability of abiraterone acetate
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WO2014071984A1 (en) 2012-11-09 2014-05-15 Synthon Bv Process for making abiraterone-3-acetate
TWI570131B (zh) * 2012-11-13 2017-02-11 賽克系統公司 製備１７－經取代類固醇之方法
WO2014075978A1 (en) 2012-11-16 2014-05-22 Synthon B.V. Process for the production of abiraterone-3-acetate involving an enol trliflation reaction in the presence of an alkoxy-pyridine compound
CN103059091B (zh) * 2012-11-22 2017-04-19 常州靶点医药科技有限公司 一种避免重金属残留的醋酸阿比特龙的制备方法
CN103864878A (zh) * 2012-12-12 2014-06-18 天津大学 阿比特龙醋酸酯的制备方法
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US20160022606A1 (en) 2013-03-14 2016-01-28 Pellficure Pharmaceuticals Inc. Novel therapy for prostate carcinoma
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EP3013844A4 (en) * 2013-06-24 2017-03-01 Sun Pharmaceutical Industries LTD Process for preparation of abiraterone acetate
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CN110272465A (zh) * 2019-07-15 2019-09-24 成都贝诺科成生物科技有限公司 阿比特龙衍生物、其制备方法与应用
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Also Published As

Publication number Publication date
GB2265624A (en) 1993-10-06
CZ233794A3 (en) 1995-02-15
KR950700923A (ko) 1995-02-20
JP2742331B2 (ja) 1998-04-22
CA2132449A1 (en) 1993-10-14
NZ249911A (en) 1996-06-25
CA2132449C (en) 2002-09-10
AU668144B2 (en) 1996-04-26
ATE186913T1 (de) 1999-12-15
CZ287434B6 (en) 2000-11-15
GB9305269D0 (en) 1993-05-05
EP0633893B1 (en) 1999-11-24
JPH07505377A (ja) 1995-06-15
DE69327096T2 (de) 2000-06-21
IL105078A0 (en) 1993-07-08
DE122012000012I1 (de) 2012-06-14
DK0633893T3 (da) 2000-04-17
ES2138618T3 (es) 2000-01-16
KR100235135B1 (ko) 2000-01-15
EP0633893A1 (en) 1995-01-18
DE69327096D1 (de) 1999-12-30
MX9301525A (es) 1994-02-28
AU3758493A (en) 1993-11-08
GB2265624B (en) 1995-04-19
WO1993020097A1 (en) 1993-10-14
LU91911I2 (fr) 2012-02-07

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