HUE027481T2 - Methods of treating cancer using 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione - Google Patents

Methods of treating cancer using 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione Download PDF

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Publication number
HUE027481T2
HUE027481T2 HUE12710836A HUE12710836A HUE027481T2 HU E027481 T2 HUE027481 T2 HU E027481T2 HU E12710836 A HUE12710836 A HU E12710836A HU E12710836 A HUE12710836 A HU E12710836A HU E027481 T2 HUE027481 T2 HU E027481T2
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HU
Hungary
Prior art keywords
compound
cancer
cell
lymphoma
patient
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HUE12710836A
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English (en)
Hungarian (hu)
Inventor
George W Muller
Peter H Schafer
Hon-Wah Man
Ling-Hua Zhang
Anita Gandhi
Rajesh Chopra
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Celgene Corp
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Publication of HUE027481T2 publication Critical patent/HUE027481T2/en

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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
    • A61B18/00—Surgical instruments, devices or methods for transferring non-mechanical forms of energy to or from the body
    • A61B18/18—Surgical instruments, devices or methods for transferring non-mechanical forms of energy to or from the body by applying electromagnetic radiation, e.g. microwaves
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    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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HUE12710836A 2011-03-11 2012-03-09 Methods of treating cancer using 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione HUE027481T2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161451995P 2011-03-11 2011-03-11
US201161480272P 2011-04-28 2011-04-28

Publications (1)

Publication Number Publication Date
HUE027481T2 true HUE027481T2 (en) 2016-09-28

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HUE12710836A HUE027481T2 (en) 2011-03-11 2012-03-09 Methods of treating cancer using 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione

Country Status (29)

Country Link
US (6) US20140148473A1 (enExample)
EP (3) EP3025715A1 (enExample)
JP (5) JP2014510078A (enExample)
KR (2) KR20140025374A (enExample)
CN (3) CN103561743A (enExample)
AR (1) AR085651A1 (enExample)
AU (4) AU2012229300B2 (enExample)
BR (2) BR112013023277A2 (enExample)
CA (2) CA2829592A1 (enExample)
CY (1) CY1117430T1 (enExample)
DK (1) DK2683384T3 (enExample)
EA (2) EA201691939A1 (enExample)
ES (2) ES2659205T3 (enExample)
HR (1) HRP20160056T1 (enExample)
HU (1) HUE027481T2 (enExample)
IL (2) IL227990B (enExample)
MX (2) MX2013010217A (enExample)
NI (2) NI201300082A (enExample)
PH (2) PH12013501820A1 (enExample)
PL (1) PL2683384T3 (enExample)
PT (1) PT2683384E (enExample)
RS (1) RS54553B1 (enExample)
RU (3) RU2013145524A (enExample)
SG (2) SG193320A1 (enExample)
SI (1) SI2683384T1 (enExample)
SM (1) SMT201600034B (enExample)
TW (2) TWI542349B (enExample)
WO (2) WO2012125459A1 (enExample)
ZA (2) ZA201306148B (enExample)

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