PT2683384E - Métodos de tratamento de cancro utilizando 3-(5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona - Google Patents

Métodos de tratamento de cancro utilizando 3-(5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona Download PDF

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Publication number
PT2683384E
PT2683384E PT127108363T PT12710836T PT2683384E PT 2683384 E PT2683384 E PT 2683384E PT 127108363 T PT127108363 T PT 127108363T PT 12710836 T PT12710836 T PT 12710836T PT 2683384 E PT2683384 E PT 2683384E
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PT
Portugal
Prior art keywords
quinazolin
dione
piperidine
oxo
amino
Prior art date
Application number
PT127108363T
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English (en)
Inventor
Man Hon-Wah
H Schafer Peter
W Muller George
Zhang Ling-Hua
Gandhi Anita
Chopra Rajesh
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
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Application filed by Celgene Corp filed Critical Celgene Corp
Publication of PT2683384E publication Critical patent/PT2683384E/pt

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
    • A61B18/00—Surgical instruments, devices or methods for transferring non-mechanical forms of energy to or from the body
    • A61B18/18—Surgical instruments, devices or methods for transferring non-mechanical forms of energy to or from the body by applying electromagnetic radiation, e.g. microwaves
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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PT127108363T 2011-03-11 2012-03-09 Métodos de tratamento de cancro utilizando 3-(5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona PT2683384E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161451995P 2011-03-11 2011-03-11
US201161480272P 2011-04-28 2011-04-28

Publications (1)

Publication Number Publication Date
PT2683384E true PT2683384E (pt) 2016-03-11

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PT127108363T PT2683384E (pt) 2011-03-11 2012-03-09 Métodos de tratamento de cancro utilizando 3-(5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona

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US (6) US8906932B2 (pt)
EP (3) EP3025715A1 (pt)
JP (5) JP6118273B2 (pt)
KR (2) KR20140025374A (pt)
CN (3) CN103561744A (pt)
AR (1) AR085651A1 (pt)
AU (4) AU2012229300B2 (pt)
BR (2) BR112013023277A2 (pt)
CA (2) CA2829592A1 (pt)
CY (1) CY1117430T1 (pt)
DK (1) DK2683384T3 (pt)
EA (2) EA201391319A1 (pt)
ES (2) ES2562332T3 (pt)
HK (1) HK1191858A1 (pt)
HR (1) HRP20160056T1 (pt)
HU (1) HUE027481T2 (pt)
IL (2) IL227990B (pt)
MX (2) MX2013010217A (pt)
NI (2) NI201300081A (pt)
PL (1) PL2683384T3 (pt)
PT (1) PT2683384E (pt)
RS (1) RS54553B1 (pt)
RU (3) RU2013145556A (pt)
SG (2) SG192947A1 (pt)
SI (1) SI2683384T1 (pt)
SM (1) SMT201600034B (pt)
TW (2) TW201700100A (pt)
WO (2) WO2012125475A1 (pt)
ZA (2) ZA201306148B (pt)

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