HU226982B1 - Novel tiotropium-containing inhalation powder, process for its preperation and its use - Google Patents
Novel tiotropium-containing inhalation powder, process for its preperation and its use Download PDFInfo
- Publication number
- HU226982B1 HU226982B1 HU0203885A HUP0203885A HU226982B1 HU 226982 B1 HU226982 B1 HU 226982B1 HU 0203885 A HU0203885 A HU 0203885A HU P0203885 A HUP0203885 A HU P0203885A HU 226982 B1 HU226982 B1 HU 226982B1
- Authority
- HU
- Hungary
- Prior art keywords
- excipient
- inhalable powder
- tiotropium
- powder according
- inhalable
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Otolaryngology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10050635 | 2000-10-12 | ||
| PCT/EP2001/011227 WO2002030389A1 (de) | 2000-10-12 | 2001-09-28 | Neue tiotropium-haltige inhalationspulver |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HUP0203885A2 HUP0203885A2 (hu) | 2003-03-28 |
| HUP0203885A3 HUP0203885A3 (en) | 2005-01-28 |
| HU226982B1 true HU226982B1 (en) | 2010-04-28 |
Family
ID=7659578
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0203885A HU226982B1 (en) | 2000-10-12 | 2001-09-28 | Novel tiotropium-containing inhalation powder, process for its preperation and its use |
Country Status (48)
Families Citing this family (79)
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| US20030055026A1 (en) | 2001-04-17 | 2003-03-20 | Dey L.P. | Formoterol/steroid bronchodilating compositions and methods of use thereof |
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| DE10128779A1 (de) * | 2001-06-13 | 2003-01-02 | Boehringer Ingelheim Pharma | Verfahren zur Reinigung von Hartgelatinekapseln |
| US20030008001A1 (en) * | 2001-06-13 | 2003-01-09 | Boehringer Ingelheim Pharma Kg | Process for cleaning hard gelatine capsules |
| DE10141376A1 (de) * | 2001-08-23 | 2003-03-13 | Boehringer Ingelheim Pharma | Verfahren zur Herstellung von Inhalationspulvern |
| DE10141377A1 (de) | 2001-08-23 | 2003-03-13 | Boehringer Ingelheim Pharma | Aufstreuverfahren zur Herstellung von Pulverformulierungen |
| DE10212264A1 (de) | 2002-03-20 | 2003-10-02 | Boehringer Ingelheim Pharma | Kristallines Mikronisat, Verfahren zu dessen Herstellung und dessen Verwendung zur Herstellung eines Arzneimittels |
| US7309707B2 (en) * | 2002-03-20 | 2007-12-18 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Crystalline micronisate, process for the manufacture thereof and use thereof for the preparation of a medicament |
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| WO2003084509A1 (en) * | 2002-04-04 | 2003-10-16 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Powder formulations suitable for inhalation |
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| RU2762084C2 (ru) | 2015-12-24 | 2021-12-15 | Филип Моррис Продактс С.А. | Ароматизированный никотиновый порошок |
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| EP4108230A1 (en) | 2021-06-24 | 2022-12-28 | Laboratoires SMB | New dry powder composition of tiotropium for inhalation |
| GR1010358B (el) * | 2021-09-14 | 2022-12-16 | Elpen Ανωνυμος Εταιρεια Φαρμακευτικη Βιομηχανια, | Σταθερο φαρμακευτικο σκευασμα που περιεχει βρωμιουχο τιοτροπιο, για χορηγηση απο το αναπνευστικο |
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| DE10141376A1 (de) | 2001-08-23 | 2003-03-13 | Boehringer Ingelheim Pharma | Verfahren zur Herstellung von Inhalationspulvern |
| US7309707B2 (en) * | 2002-03-20 | 2007-12-18 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Crystalline micronisate, process for the manufacture thereof and use thereof for the preparation of a medicament |
| WO2003084509A1 (en) | 2002-04-04 | 2003-10-16 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Powder formulations suitable for inhalation |
| UA80123C2 (en) | 2002-04-09 | 2007-08-27 | Boehringer Ingelheim Pharma | Inhalation kit comprising inhalable powder of tiotropium |
| US20030235538A1 (en) * | 2002-04-09 | 2003-12-25 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Method for the administration of an anticholinergic by inhalation |
| US7763280B2 (en) | 2002-11-28 | 2010-07-27 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Tiotropium containing powder formulation for inhalation |
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2001
- 2001-09-28 AP APAP/P/2003/002774A patent/AP1712A/en active
- 2001-09-28 SI SI200130160T patent/SI1292281T1/xx unknown
- 2001-09-28 CZ CZ20021785A patent/CZ301465B6/cs not_active IP Right Cessation
- 2001-09-28 NZ NZ519406A patent/NZ519406A/en not_active IP Right Cessation
- 2001-09-28 PT PT01969789T patent/PT1292281E/pt unknown
- 2001-09-28 AT AT01969789T patent/ATE275391T1/de active
- 2001-09-28 WO PCT/EP2001/011227 patent/WO2002030389A1/de not_active Ceased
- 2001-09-28 HU HU0203885A patent/HU226982B1/hu unknown
- 2001-09-28 DK DK01969789T patent/DK1292281T3/da active
- 2001-09-28 DZ DZ013477A patent/DZ3477A1/xx active
- 2001-09-28 BR BR0107304-4A patent/BR0107304A/pt not_active Application Discontinuation
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- 2001-09-28 CN CNB01803098XA patent/CN1210017C/zh not_active Ceased
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- 2001-09-28 UA UA2002064932A patent/UA72014C2/uk unknown
- 2001-09-28 MX MXPA02005666A patent/MXPA02005666A/es active IP Right Grant
- 2001-09-28 SK SK706-2002A patent/SK285389B6/sk not_active IP Right Cessation
- 2001-09-28 EA EA200200551A patent/EA004034B1/ru not_active IP Right Cessation
- 2001-09-28 EP EP04006349A patent/EP1430887A1/de not_active Withdrawn
- 2001-09-28 HR HR20020437A patent/HRP20020437B1/xx not_active IP Right Cessation
- 2001-09-28 KR KR10-2002-7007877A patent/KR100488644B1/ko not_active Expired - Lifetime
- 2001-09-28 JP JP2002533832A patent/JP3870159B2/ja not_active Expired - Lifetime
- 2001-09-28 IL IL14998401A patent/IL149984A0/xx active IP Right Grant
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- 2001-10-09 TW TW090124971A patent/TWI285553B/zh not_active IP Right Cessation
- 2001-10-09 EG EG20011059A patent/EG24139A/xx active
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- 2001-10-10 PE PE2001001001A patent/PE20020577A1/es active IP Right Grant
- 2001-10-10 UY UY26959A patent/UY26959A1/es not_active IP Right Cessation
- 2001-10-11 US US09/975,418 patent/US7070800B2/en not_active Expired - Lifetime
- 2001-10-12 AR ARP010104783A patent/AR031819A1/es not_active Application Discontinuation
- 2001-10-15 SA SA01220460A patent/SA01220460B1/ar unknown
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2002
- 2002-05-21 ZA ZA200204378A patent/ZA200204378B/xx unknown
- 2002-05-21 BG BG106730A patent/BG65753B1/bg unknown
- 2002-05-22 NO NO20022414A patent/NO331956B1/no not_active IP Right Cessation
- 2002-05-28 EC EC2002004268A patent/ECSP024268A/es unknown
- 2002-06-03 IL IL149984A patent/IL149984A/en unknown
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2003
- 2003-03-26 CR CR6937A patent/CR6937A/es not_active Application Discontinuation
- 2003-04-08 IS IS6771A patent/IS2360B/is unknown
- 2003-04-08 MA MA27103A patent/MA25843A1/fr unknown
- 2003-04-08 EC EC2003004546A patent/ECSP034546A/es unknown
- 2003-04-11 CU CU20030082A patent/CU23284B7/es unknown
- 2003-12-05 US US10/729,543 patent/US20040228806A1/en not_active Abandoned
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2005
- 2005-10-20 US US11/254,573 patent/US20060039868A1/en not_active Abandoned
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2008
- 2008-07-29 US US12/181,651 patent/US20080292563A1/en not_active Abandoned
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