HRP950321B1 - Cortricitropin releasing factor antagonists - Google Patents

Cortricitropin releasing factor antagonists

Info

Publication number
HRP950321B1
HRP950321B1 HR950321A HRP950321A HRP950321B1 HR P950321 B1 HRP950321 B1 HR P950321B1 HR 950321 A HR950321 A HR 950321A HR P950321 A HRP950321 A HR P950321A HR P950321 B1 HRP950321 B1 HR P950321B1
Authority
HR
Croatia
Prior art keywords
pct
releasing factor
cortricitropin
factor antagonists
date dec
Prior art date
Application number
HR950321A
Other languages
English (en)
Inventor
L Chen Yuhpung
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of HRP950321A2 publication Critical patent/HRP950321A2/hr
Publication of HRP950321B1 publication Critical patent/HRP950321B1/xx

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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/69—Two or more oxygen atoms
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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HR950321A 1994-06-08 1995-06-07 Cortricitropin releasing factor antagonists HRP950321B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25551494A 1994-06-08 1994-06-08

Publications (2)

Publication Number Publication Date
HRP950321A2 HRP950321A2 (en) 1998-02-28
HRP950321B1 true HRP950321B1 (en) 2001-08-31

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Family Applications (1)

Application Number Title Priority Date Filing Date
HR950321A HRP950321B1 (en) 1994-06-08 1995-06-07 Cortricitropin releasing factor antagonists

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Country Link
US (1) US5962479A (de)
EP (1) EP0764166B1 (de)
JP (3) JP3193055B2 (de)
KR (2) KR20030096422A (de)
CN (2) CN1049659C (de)
AT (1) ATE196295T1 (de)
AU (1) AU692548B2 (de)
BR (1) BR9502708A (de)
CA (1) CA2192354C (de)
CO (1) CO4440627A1 (de)
CZ (1) CZ293752B6 (de)
DE (1) DE69518841T2 (de)
DK (1) DK0764166T3 (de)
ES (1) ES2150567T3 (de)
FI (2) FI114469B (de)
GR (1) GR3034765T3 (de)
HR (1) HRP950321B1 (de)
HU (1) HUT75774A (de)
IL (1) IL114004A0 (de)
MY (1) MY114522A (de)
NO (2) NO308994B1 (de)
NZ (1) NZ285442A (de)
PE (1) PE32596A1 (de)
PL (1) PL320631A1 (de)
PT (1) PT764166E (de)
RU (1) RU2221799C2 (de)
SK (1) SK155596A3 (de)
TW (2) TW574214B (de)
UA (1) UA71535C2 (de)
WO (1) WO1995033750A1 (de)
YU (1) YU38795A (de)
ZA (1) ZA954677B (de)

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DE69533284T2 (de) * 1994-04-29 2005-07-21 Pfizer Inc. Neue cyclische und acyclische amide zur erhöhung der neurotransmitter ausschüttung
EP0729758A3 (de) * 1995-03-02 1997-10-29 Pfizer Pyrazolopyrimidine und Pyrrolopyrimidine zur Behandlung von neuronalen und anderen Krankheiten
US6956047B1 (en) 1995-06-06 2005-10-18 Pfizer Inc. Corticotropin releasing factor antagonists
US7125880B1 (en) 1995-06-06 2006-10-24 Pfizer Inc. Corticotropin releasing factor antagonists
US6403599B1 (en) * 1995-11-08 2002-06-11 Pfizer Inc Corticotropin releasing factor antagonists
US5955613A (en) * 1995-10-13 1999-09-21 Neurogen Corporation Certain pyrrolopyridine derivatives; novel CRF1 specific ligands
AU738304B2 (en) 1995-10-13 2001-09-13 Neurogen Corporation Certain pyrrolopyridine derivatives; novel CRF 1 specific ligands
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