HK1214527A1 - 酪蛋白激酶1δ(CK1δ)抑制剂 - Google Patents

酪蛋白激酶1δ(CK1δ)抑制剂 Download PDF

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Publication number
HK1214527A1
HK1214527A1 HK16102571.5A HK16102571A HK1214527A1 HK 1214527 A1 HK1214527 A1 HK 1214527A1 HK 16102571 A HK16102571 A HK 16102571A HK 1214527 A1 HK1214527 A1 HK 1214527A1
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Hong Kong
Prior art keywords
alkyl
aryl
compound
group
heteroaryl
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HK16102571.5A
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English (en)
Chinese (zh)
Inventor
Joseph M. Sheridan
Jonathan R. Heal
William D.O. Hamilton
Ian Pike
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Electrophoretics Limited
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Priority claimed from GBGB1021161.3A external-priority patent/GB201021161D0/en
Priority claimed from GBGB1109162.6A external-priority patent/GB201109162D0/en
Application filed by Electrophoretics Limited filed Critical Electrophoretics Limited
Publication of HK1214527A1 publication Critical patent/HK1214527A1/zh

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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