HK1137938A1 - Quinoline derivatives as pi3 kinase inhibitors - Google Patents
Quinoline derivatives as pi3 kinase inhibitorsInfo
- Publication number
- HK1137938A1 HK1137938A1 HK10104231.9A HK10104231A HK1137938A1 HK 1137938 A1 HK1137938 A1 HK 1137938A1 HK 10104231 A HK10104231 A HK 10104231A HK 1137938 A1 HK1137938 A1 HK 1137938A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- kinase inhibitors
- quinoline derivatives
- quinoline
- derivatives
- kinase
- Prior art date
Links
- 229940027991 antiseptic and disinfectant quinoline derivative Drugs 0.000 title 1
- 239000002935 phosphatidylinositol 3 kinase inhibitor Substances 0.000 title 1
- 125000002943 quinolinyl group Chemical class N1=C(C=CC2=CC=CC=C12)* 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US93876107P | 2007-05-18 | 2007-05-18 | |
PCT/US2008/063819 WO2008144463A1 (en) | 2007-05-18 | 2008-05-16 | Quinoline derivatives as pi3 kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1137938A1 true HK1137938A1 (en) | 2010-08-13 |
Family
ID=40088996
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK10104231.9A HK1137938A1 (en) | 2007-05-18 | 2010-04-29 | Quinoline derivatives as pi3 kinase inhibitors |
Country Status (32)
Country | Link |
---|---|
US (6) | US20100168100A1 (xx) |
EP (3) | EP2596793B1 (xx) |
JP (3) | JP4814396B2 (xx) |
KR (1) | KR101458660B1 (xx) |
CN (1) | CN101754759B (xx) |
AR (1) | AR066614A1 (xx) |
AU (1) | AU2008254915B2 (xx) |
BR (1) | BRPI0811761A2 (xx) |
CA (1) | CA2686016C (xx) |
CL (1) | CL2008001457A1 (xx) |
CO (1) | CO6241101A2 (xx) |
CR (1) | CR11165A (xx) |
CY (1) | CY1114070T1 (xx) |
DK (1) | DK2162131T3 (xx) |
EA (1) | EA019540B1 (xx) |
ES (2) | ES2404557T3 (xx) |
HK (1) | HK1137938A1 (xx) |
HR (1) | HRP20130252T1 (xx) |
IL (1) | IL202018A (xx) |
JO (1) | JO2891B1 (xx) |
MA (1) | MA31443B1 (xx) |
MX (2) | MX342959B (xx) |
MY (1) | MY158843A (xx) |
NZ (1) | NZ580979A (xx) |
PE (1) | PE20090717A1 (xx) |
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PT (1) | PT2162131E (xx) |
SI (1) | SI2162131T1 (xx) |
TW (1) | TWI410417B (xx) |
UA (1) | UA104408C2 (xx) |
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- 2008-05-16 WO PCT/US2008/063819 patent/WO2008144463A1/en active Application Filing
- 2008-05-16 US US12/600,752 patent/US20100168100A1/en not_active Abandoned
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