MX315904B - Inhibidores de fosfoinosituro-3 cinasa. - Google Patents

Inhibidores de fosfoinosituro-3 cinasa.

Info

Publication number
MX315904B
MX315904B MX2010013110A MX2010013110A MX315904B MX 315904 B MX315904 B MX 315904B MX 2010013110 A MX2010013110 A MX 2010013110A MX 2010013110 A MX2010013110 A MX 2010013110A MX 315904 B MX315904 B MX 315904B
Authority
MX
Mexico
Prior art keywords
kinase
inhibitors
Prior art date
Application number
MX2010013110A
Other languages
English (en)
Other versions
MX2010013110A (es
Inventor
Shon Booker
Mark H Norman
Yunxin Y Bo
Longbin Liu
Kevin Yang
Nobuko Nishimura
Holly L Deak
Aaron C Siegmund
Laurie Schenkel
Kathleen Panter
Nuria A Tamayo
Marian Bryan
Kristin Andrews
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of MX2010013110A publication Critical patent/MX2010013110A/es
Publication of MX315904B publication Critical patent/MX315904B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2010013110A 2008-05-30 2009-05-29 Inhibidores de fosfoinosituro-3 cinasa. MX315904B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5774508P 2008-05-30 2008-05-30
PCT/US2009/045713 WO2009155121A2 (en) 2008-05-30 2009-05-29 Inhibitors of pi3 kinase

Publications (2)

Publication Number Publication Date
MX2010013110A MX2010013110A (es) 2010-12-20
MX315904B true MX315904B (es) 2013-11-29

Family

ID=40902593

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010013110A MX315904B (es) 2008-05-30 2009-05-29 Inhibidores de fosfoinosituro-3 cinasa.

Country Status (8)

Country Link
US (1) US8415376B2 (es)
EP (1) EP2307400B1 (es)
JP (1) JP5599783B2 (es)
AU (1) AU2009260447B2 (es)
CA (1) CA2725014C (es)
ES (1) ES2474147T3 (es)
MX (1) MX315904B (es)
WO (1) WO2009155121A2 (es)

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US8415376B2 (en) 2013-04-09
AU2009260447B2 (en) 2012-03-29
WO2009155121A3 (en) 2010-02-18
MX2010013110A (es) 2010-12-20
EP2307400A2 (en) 2011-04-13
CA2725014A1 (en) 2009-12-23
AU2009260447A1 (en) 2009-12-23
EP2307400B1 (en) 2014-04-23
JP5599783B2 (ja) 2014-10-01
JP2011522806A (ja) 2011-08-04
ES2474147T3 (es) 2014-07-08

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