GB0810902D0 - New compounds - Google Patents

New compounds

Info

Publication number
GB0810902D0
GB0810902D0 GBGB0810902.7A GB0810902A GB0810902D0 GB 0810902 D0 GB0810902 D0 GB 0810902D0 GB 0810902 A GB0810902 A GB 0810902A GB 0810902 D0 GB0810902 D0 GB 0810902D0
Authority
GB
United Kingdom
Prior art keywords
new compounds
compounds
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0810902.7A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astex Therapeutics Ltd
Original Assignee
Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astex Therapeutics Ltd filed Critical Astex Therapeutics Ltd
Priority to GBGB0810902.7A priority Critical patent/GB0810902D0/en
Publication of GB0810902D0 publication Critical patent/GB0810902D0/en
Priority to CN200980122215.8A priority patent/CN102137859B/zh
Priority to US12/997,754 priority patent/US8796244B2/en
Priority to BRPI0915084A priority patent/BRPI0915084B8/pt
Priority to LTEP09761801.1T priority patent/LT2300465T/lt
Priority to HUE09761801A priority patent/HUE045300T2/hu
Priority to SI200931974T priority patent/SI2300465T1/sl
Priority to JP2011512999A priority patent/JP5596023B2/ja
Priority to DK09761801.1T priority patent/DK2300465T3/da
Priority to KR1020117000791A priority patent/KR101745730B1/ko
Priority to NZ589781A priority patent/NZ589781A/xx
Priority to EP09761801.1A priority patent/EP2300465B1/en
Priority to CA2727062A priority patent/CA2727062A1/en
Priority to HRP20191027 priority patent/HRP20191027T1/hr
Priority to AU2009256584A priority patent/AU2009256584B2/en
Priority to ES09761801T priority patent/ES2735979T3/es
Priority to RU2011100786/04A priority patent/RU2518089C2/ru
Priority to PCT/EP2009/057318 priority patent/WO2009150240A1/en
Priority to MX2010013743A priority patent/MX2010013743A/es
Priority to IL209864A priority patent/IL209864A/en
Priority to ZA2010/08961A priority patent/ZA201008961B/en
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
GBGB0810902.7A 2008-06-13 2008-06-13 New compounds Ceased GB0810902D0 (en)

Priority Applications (21)

Application Number Priority Date Filing Date Title
GBGB0810902.7A GB0810902D0 (en) 2008-06-13 2008-06-13 New compounds
MX2010013743A MX2010013743A (es) 2008-06-13 2009-06-12 Derivados de imidazopiridina como inhibidores de receptor de tirosina-cinasas.
NZ589781A NZ589781A (en) 2008-06-13 2009-06-12 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
CA2727062A CA2727062A1 (en) 2008-06-13 2009-06-12 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
BRPI0915084A BRPI0915084B8 (pt) 2008-06-13 2009-06-12 composto, e, composição farmacêutica
LTEP09761801.1T LT2300465T (lt) 2008-06-13 2009-06-12 Imidazopiridino dariniai kaip receptoriaus tirozino kinazių inhibitoriai
HUE09761801A HUE045300T2 (hu) 2008-06-13 2009-06-12 Imidazopiridin származékok, mint receptor tirozin kinázok inhibitorai
SI200931974T SI2300465T1 (sl) 2008-06-13 2009-06-12 Imidazopiridinski derivati kot inhibitorji receptorskih tirozin kinaz
JP2011512999A JP5596023B2 (ja) 2008-06-13 2009-06-12 レセプターチロシンキナーゼのインヒビターとしてのイミダゾピリジン誘導体
DK09761801.1T DK2300465T3 (da) 2008-06-13 2009-06-12 Imidazopyridinderivater som hæmmere af receptortyrosinkinaser
KR1020117000791A KR101745730B1 (ko) 2008-06-13 2009-06-12 수용체 티로신 키나제의 억제제로서의 이미다조피리딘 유도체
CN200980122215.8A CN102137859B (zh) 2008-06-13 2009-06-12 作为受体酪氨酸激酶的抑制剂的咪唑并吡啶衍生物
EP09761801.1A EP2300465B1 (en) 2008-06-13 2009-06-12 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
US12/997,754 US8796244B2 (en) 2008-06-13 2009-06-12 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
HRP20191027 HRP20191027T1 (hr) 2008-06-13 2009-06-12 Derivati imidazopiridina kao inhibitori tiposinskih receptora kinaza
AU2009256584A AU2009256584B2 (en) 2008-06-13 2009-06-12 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
ES09761801T ES2735979T3 (es) 2008-06-13 2009-06-12 Derivados de la imidazopiridina como inhibidores de tirosina quinasas receptoras
RU2011100786/04A RU2518089C2 (ru) 2008-06-13 2009-06-12 Производные имидазопиридина в качестве ингибиторов рецепторных тирозинкиназ
PCT/EP2009/057318 WO2009150240A1 (en) 2008-06-13 2009-06-12 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
IL209864A IL209864A (en) 2008-06-13 2010-12-09 History of imidazopyridine as tyrosine receptor kinase inhibitors
ZA2010/08961A ZA201008961B (en) 2008-06-13 2010-12-13 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0810902.7A GB0810902D0 (en) 2008-06-13 2008-06-13 New compounds

Publications (1)

Publication Number Publication Date
GB0810902D0 true GB0810902D0 (en) 2008-07-23

Family

ID=39672279

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0810902.7A Ceased GB0810902D0 (en) 2008-06-13 2008-06-13 New compounds

Country Status (21)

Country Link
US (1) US8796244B2 (enExample)
EP (1) EP2300465B1 (enExample)
JP (1) JP5596023B2 (enExample)
KR (1) KR101745730B1 (enExample)
CN (1) CN102137859B (enExample)
AU (1) AU2009256584B2 (enExample)
BR (1) BRPI0915084B8 (enExample)
CA (1) CA2727062A1 (enExample)
DK (1) DK2300465T3 (enExample)
ES (1) ES2735979T3 (enExample)
GB (1) GB0810902D0 (enExample)
HR (1) HRP20191027T1 (enExample)
HU (1) HUE045300T2 (enExample)
IL (1) IL209864A (enExample)
LT (1) LT2300465T (enExample)
MX (1) MX2010013743A (enExample)
NZ (1) NZ589781A (enExample)
RU (1) RU2518089C2 (enExample)
SI (1) SI2300465T1 (enExample)
WO (1) WO2009150240A1 (enExample)
ZA (1) ZA201008961B (enExample)

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CN101679408B (zh) 2006-12-22 2016-04-27 Astex治疗学有限公司 作为fgfr抑制剂的双环杂环化合物
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JP2011522866A (ja) 2011-08-04
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IL209864A (en) 2015-10-29
AU2009256584B2 (en) 2014-06-12
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AU2009256584A1 (en) 2009-12-17
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DK2300465T3 (da) 2019-06-24
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