FR2338271A1 - Derives du phtalane, procede pour leur preparation, et compositions pharmaceutiques contenant de tels derives - Google Patents

Derives du phtalane, procede pour leur preparation, et compositions pharmaceutiques contenant de tels derives

Info

Publication number
FR2338271A1
FR2338271A1 FR7701079A FR7701079A FR2338271A1 FR 2338271 A1 FR2338271 A1 FR 2338271A1 FR 7701079 A FR7701079 A FR 7701079A FR 7701079 A FR7701079 A FR 7701079A FR 2338271 A1 FR2338271 A1 FR 2338271A1
Authority
FR
France
Prior art keywords
derivatives
phthalane
preparation
pharmaceutical compositions
compositions containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7701079A
Other languages
English (en)
French (fr)
Other versions
FR2338271B1 (forum.php
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
H Lundbeck AS
Original Assignee
Kefalas AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9722860&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR2338271(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kefalas AS filed Critical Kefalas AS
Publication of FR2338271A1 publication Critical patent/FR2338271A1/fr
Application granted granted Critical
Publication of FR2338271B1 publication Critical patent/FR2338271B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR7701079A 1976-01-14 1977-01-14 Derives du phtalane, procede pour leur preparation, et compositions pharmaceutiques contenant de tels derives Granted FR2338271A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1486/76A GB1526331A (en) 1976-01-14 1976-01-14 Phthalanes

Publications (2)

Publication Number Publication Date
FR2338271A1 true FR2338271A1 (fr) 1977-08-12
FR2338271B1 FR2338271B1 (forum.php) 1982-11-05

Family

ID=9722860

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7701079A Granted FR2338271A1 (fr) 1976-01-14 1977-01-14 Derives du phtalane, procede pour leur preparation, et compositions pharmaceutiques contenant de tels derives

Country Status (19)

Country Link
US (1) US4136193A (forum.php)
JP (1) JPS52105162A (forum.php)
AT (1) AT359488B (forum.php)
AU (1) AU509445B2 (forum.php)
BE (1) BE850401A (forum.php)
CA (1) CA1094087A (forum.php)
CH (3) CH626886A5 (forum.php)
DE (1) DE2657013C2 (forum.php)
DK (1) DK143275C (forum.php)
ES (1) ES454980A1 (forum.php)
FI (1) FI63754C (forum.php)
FR (1) FR2338271A1 (forum.php)
GB (1) GB1526331A (forum.php)
IE (1) IE44055B1 (forum.php)
NL (2) NL192451C (forum.php)
NO (2) NO147243C (forum.php)
NZ (1) NZ183001A (forum.php)
SE (1) SE429551B (forum.php)
ZA (1) ZA7757B (forum.php)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003087081A1 (en) * 2002-04-09 2003-10-23 Torcan Chemical Ltd. Process and intermediates for preparing escitalopram

Families Citing this family (161)

* Cited by examiner, † Cited by third party
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US4602035A (en) * 1983-12-07 1986-07-22 Hoechst-Roussel Pharmaceuticals Inc. Antidepressant (3-aryl-2,3-dihydrobenzofuran-3-yl)alkylamines
GB8419963D0 (en) * 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
ES2145977T3 (es) * 1995-08-16 2000-07-16 Lilly Co Eli Potenciacion de la respuesta de la serotonina.
SK283309B6 (sk) * 1997-07-08 2003-05-02 H. Lundbeck A/S Spôsob výroby citalopramu a medziprodukty
UA62985C2 (en) * 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
HUP0002953A3 (en) 1997-11-11 2002-12-28 Lundbeck & Co As H Method for preparation of citalopram and intermediates used for them
PL199423B1 (pl) 1998-10-20 2008-09-30 Lundbeck & Co As H Sposób wytwarzania citalopramu
AR021509A1 (es) * 1998-12-08 2002-07-24 Lundbeck & Co As H Derivados de benzofurano, su preparacion y uso
HRP20010418A2 (en) 1998-12-08 2002-06-30 Lundbeck & Co As H Benzofuran derivatives, their preparation and use
ATE236145T1 (de) 1998-12-23 2003-04-15 Lundbeck & Co As H Verfahren zur herstellung von 5-cyanophthalid
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
PL198024B1 (pl) * 1999-04-14 2008-05-30 Lundbeck & Co As H Sposób wytwarzania citalopramu, związki pośrednie i ich zastosowanie do wytwarzania citalopramu
ITMI991581A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991579A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991486A1 (it) * 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
AR021155A1 (es) * 1999-07-08 2002-06-12 Lundbeck & Co As H Tratamiento de desordenes neuroticos
EP1298124B1 (en) 1999-10-25 2007-02-28 H. Lundbeck A/S Method For the Preparation of Citalopram
WO2000012044A2 (en) 1999-10-25 2000-03-09 H. Lundbeck A/S Method for the preparation of citalopram
US6310222B1 (en) * 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
KR20020073489A (ko) * 1999-12-28 2002-09-26 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
TR200201688T2 (tr) * 1999-12-30 2002-11-21 H. Lundbeck A/S Sitalopram hazırlama yöntemi.
SK286879B6 (sk) * 2000-01-14 2009-07-06 H. Lundbeck A/S Spôsob prípravy 5-kyanoftalidu
US6433196B1 (en) 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017415C1 (nl) * 2000-02-24 2001-05-18 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
IES20010143A2 (en) * 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
NL1017417C1 (nl) * 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
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AU2001239210A1 (en) * 2000-03-13 2001-09-24 H. Lundbeck A/S Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
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TR200202166T2 (tr) * 2000-03-13 2002-12-23 H. Lndbeck A/S Sitalopramın preparasyon metodu
GB2357762B (en) * 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
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US6977306B2 (en) * 2000-05-02 2005-12-20 Sumitomo Chemical Company, Limited Citalopram hydrobromide crystal and method for crystallization thereof
AR032455A1 (es) * 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
KR100821912B1 (ko) * 2000-05-12 2008-04-16 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
SK3362002A3 (en) * 2000-07-06 2002-08-06 Lundbeck & Co As H Method for the preparation of citalopram
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US20030109577A1 (en) * 2000-10-27 2003-06-12 Ken Liljegren Pharmaceutical composition containing citalopram
US20030232881A1 (en) * 2000-10-27 2003-12-18 H. Lundbeck A/S Crystals of pharmaceutically acceptable salts of citalopram, methods of crystallization, and pharmaceutical compositions comprising them
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US4136193A (en) 1979-01-23
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NL192451C (nl) 1997-08-04
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NO1996001I1 (no) 1996-01-05
BE850401A (fr) 1977-07-14
SE429551B (sv) 1983-09-12
DK143275B (da) 1981-08-03
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NL192451B (nl) 1997-04-01
NL970031I1 (nl) 1997-10-01
FR2338271B1 (forum.php) 1982-11-05
CA1094087A (en) 1981-01-20
DE2657013A1 (de) 1977-07-28
FI770073A7 (forum.php) 1977-07-15
IE44055B1 (en) 1981-07-29
NL970031I2 (nl) 1997-10-01
NO147243C (no) 1983-03-02
NL7700244A (nl) 1977-07-18
DK143275C (da) 1982-01-18
DK13177A (da) 1977-07-15
AU2107377A (en) 1978-07-13
ZA7757B (en) 1977-11-30
IE44055L (en) 1977-07-14
AU509445B2 (en) 1980-05-15
ATA947276A (de) 1980-04-15
CH626886A5 (forum.php) 1981-12-15
CH632259A5 (de) 1982-09-30
NZ183001A (en) 1978-06-02
NO147243B (no) 1982-11-22
FI63754B (fi) 1983-04-29
AT359488B (de) 1980-11-10
JPS6135986B2 (forum.php) 1986-08-15
DE2657013C2 (de) 1985-11-14
GB1526331A (en) 1978-09-27
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CH632258A5 (de) 1982-09-30

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