FI66618C - Foerfarande foer framstaellning av terapeutiskt verkande 7-(2-(2-aminotiazol-4-yl)-2-(syn)-metoxi-iminoacetamido-cefalosporinderivat - Google Patents

Foerfarande foer framstaellning av terapeutiskt verkande 7-(2-(2-aminotiazol-4-yl)-2-(syn)-metoxi-iminoacetamido-cefalosporinderivat Download PDF

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Publication number
FI66618C
FI66618C FI771176A FI771176A FI66618C FI 66618 C FI66618 C FI 66618C FI 771176 A FI771176 A FI 771176A FI 771176 A FI771176 A FI 771176A FI 66618 C FI66618 C FI 66618C
Authority
FI
Finland
Prior art keywords
compound
ppm
alkyl
syn
mixture
Prior art date
Application number
FI771176A
Other languages
English (en)
Finnish (fi)
Other versions
FI66618B (fi
FI771176A (fr
Inventor
Michihiko Ochiai
Akira Morimoto
Yoshihiro Matsushita
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP4288576A external-priority patent/JPS52125188A/ja
Priority claimed from JP51108102A external-priority patent/JPS597717B2/ja
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of FI771176A publication Critical patent/FI771176A/fi
Priority to FI830278A priority Critical patent/FI830278A0/fi
Publication of FI66618B publication Critical patent/FI66618B/fi
Application granted granted Critical
Publication of FI66618C publication Critical patent/FI66618C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI771176A 1976-04-14 1977-04-14 Foerfarande foer framstaellning av terapeutiskt verkande 7-(2-(2-aminotiazol-4-yl)-2-(syn)-metoxi-iminoacetamido-cefalosporinderivat FI66618C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI830278A FI830278A0 (fi) 1976-04-14 1983-01-26 Som mellanprodukter anvaendbara 2-(2-aminotiazol-4-yl)-2-oxiiminoaettiksyrederivat

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP4288576 1976-04-14
JP4288576A JPS52125188A (en) 1976-04-14 1976-04-14 Cephalosporin derivatives and their preparation
JP51108102A JPS597717B2 (ja) 1976-09-08 1976-09-08 セフアロスポリン誘導体およびその製造法
JP10810276 1976-09-08

Publications (3)

Publication Number Publication Date
FI771176A FI771176A (fr) 1977-10-15
FI66618B FI66618B (fi) 1984-07-31
FI66618C true FI66618C (fi) 1984-11-12

Family

ID=26382633

Family Applications (1)

Application Number Title Priority Date Filing Date
FI771176A FI66618C (fi) 1976-04-14 1977-04-14 Foerfarande foer framstaellning av terapeutiskt verkande 7-(2-(2-aminotiazol-4-yl)-2-(syn)-metoxi-iminoacetamido-cefalosporinderivat

Country Status (23)

Country Link
US (4) US4520194A (fr)
AT (1) AT351164B (fr)
AU (1) AU508449B2 (fr)
BG (1) BG60438B2 (fr)
CA (1) CA1308708C (fr)
CH (4) CH629499A5 (fr)
DE (2) DE2760484C2 (fr)
DK (1) DK158671C (fr)
ES (1) ES457751A1 (fr)
FI (1) FI66618C (fr)
FR (1) FR2348218A1 (fr)
GB (1) GB1581854A (fr)
GR (1) GR63088B (fr)
HK (1) HK27684A (fr)
HU (1) HU182052B (fr)
MX (1) MX4879E (fr)
MY (1) MY8500265A (fr)
NL (1) NL7704057A (fr)
NO (1) NO771285L (fr)
PH (2) PH23284A (fr)
PT (1) PT66435B (fr)
SE (2) SE464580B (fr)
SG (1) SG76183G (fr)

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CN114014823B (zh) * 2021-12-15 2023-07-07 山东金城医药化工有限公司 反式去甲氨噻肟酸乙酯的制备方法

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FR2345153A1 (fr) * 1976-03-25 1977-10-21 Roussel Uclaf Nouvelles alcoyloximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
DK162391C (da) * 1976-04-12 1992-03-09 Fujisawa Pharmaceutical Co Analogifremgangsmaade til fremstilling af syn-isomerer af 3,7-disubstituerede 3-cephem-4-carboxylsyreforbindelser
US4304770A (en) * 1976-04-12 1981-12-08 Fujisawa Pharmaceutical Co., Ltd. Syn-isomer of 3,7-disubstituted-3-cephem-4-carboxylic acid compounds and processes for the preparation thereof
US4066762A (en) * 1976-07-12 1978-01-03 Smithkline Corporation Derivatives of 7-(2-substituted-2-hydroxyiminoacetamido)-3-(1-substituted tetrazol-5-ylthiomethyl-3-cephem-4-carboxylic acid

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CH629499A5 (de) 1982-04-30
US4278671A (en) 1981-07-14
MX4879E (es) 1982-11-26
DE2760484C2 (fr) 1992-12-03
FI66618B (fi) 1984-07-31
PH22747A (en) 1988-11-28
DE2715385A1 (de) 1977-11-10
NL7704057A (nl) 1977-10-18
PH23284A (en) 1989-06-30
US4520194A (en) 1985-05-28
CH650503A5 (de) 1985-07-31
DK158671C (da) 1990-12-31
CH630635A5 (de) 1982-06-30
SE453086B (sv) 1988-01-11
PT66435A (en) 1977-05-01
SE464580B (sv) 1991-05-13
NO771285L (no) 1977-10-17
AU2421977A (en) 1978-10-19
FR2348218B1 (fr) 1981-12-04
AT351164B (de) 1979-07-10
SE8306702D0 (sv) 1983-12-05
SE8306702L (sv) 1983-12-05
ATA256577A (de) 1978-12-15
DE2715385C2 (fr) 1991-10-17
PT66435B (en) 1978-09-20
MY8500265A (en) 1985-12-31
HU182052B (en) 1983-12-28
US4510138A (en) 1985-04-09
FR2348218A1 (fr) 1977-11-10
ES457751A1 (es) 1978-08-01
GR63088B (en) 1979-08-09
CA1308708C (fr) 1992-10-13
FI771176A (fr) 1977-10-15
CH630632A5 (de) 1982-06-30
AU508449B2 (en) 1980-03-20
HK27684A (en) 1984-03-30
BG60438B2 (bg) 1995-03-31
US4680390A (en) 1987-07-14
GB1581854A (en) 1980-12-31
SG76183G (en) 1984-08-03
DK158671B (da) 1990-07-02
DK164177A (da) 1977-10-15
SE7704233L (sv) 1977-10-15

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