FI63406C - Foerfarande foer framstaellning av terapeutiskt anvaendbara 5-entsoyl-1,2-dihydro-3h-pyrrolo(1,2-a)pyrrol-1-karboxylsyr adrivat - Google Patents
Foerfarande foer framstaellning av terapeutiskt anvaendbara 5-entsoyl-1,2-dihydro-3h-pyrrolo(1,2-a)pyrrol-1-karboxylsyr adrivat Download PDFInfo
- Publication number
- FI63406C FI63406C FI772153A FI772153A FI63406C FI 63406 C FI63406 C FI 63406C FI 772153 A FI772153 A FI 772153A FI 772153 A FI772153 A FI 772153A FI 63406 C FI63406 C FI 63406C
- Authority
- FI
- Finland
- Prior art keywords
- dihydro
- pyrrolo
- pyrrole
- formula
- carboxylic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70490976A | 1976-07-14 | 1976-07-14 | |
US70490976 | 1976-07-14 | ||
US77128677 | 1977-02-23 | ||
US05/771,286 US4089969A (en) | 1976-07-14 | 1977-02-23 | 5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof |
Publications (3)
Publication Number | Publication Date |
---|---|
FI772153A FI772153A (ja) | 1978-01-15 |
FI63406B FI63406B (fi) | 1983-02-28 |
FI63406C true FI63406C (fi) | 1983-06-10 |
Family
ID=27107410
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI772153A FI63406C (fi) | 1976-07-14 | 1977-07-11 | Foerfarande foer framstaellning av terapeutiskt anvaendbara 5-entsoyl-1,2-dihydro-3h-pyrrolo(1,2-a)pyrrol-1-karboxylsyr adrivat |
Country Status (27)
Country | Link |
---|---|
JP (1) | JPS539788A (ja) |
AR (1) | AR224997A1 (ja) |
CA (1) | CA1102809A (ja) |
CH (3) | CH641458A5 (ja) |
CS (1) | CS204954B2 (ja) |
DE (2) | DE2760330C2 (ja) |
DK (1) | DK151886C (ja) |
ES (2) | ES460706A1 (ja) |
FI (1) | FI63406C (ja) |
FR (2) | FR2358406A1 (ja) |
GB (1) | GB1554075A (ja) |
GR (1) | GR61111B (ja) |
HK (1) | HK15981A (ja) |
HU (1) | HU174224B (ja) |
IE (1) | IE45253B1 (ja) |
IL (2) | IL52493A (ja) |
IT (1) | IT1117313B (ja) |
MX (1) | MX163202B (ja) |
MY (1) | MY8100357A (ja) |
NL (2) | NL186318C (ja) |
NO (1) | NO147564C (ja) |
NZ (1) | NZ184610A (ja) |
PL (4) | PL109390B1 (ja) |
PT (1) | PT66780B (ja) |
SE (1) | SE434643B (ja) |
SU (1) | SU695558A3 (ja) |
YU (1) | YU40816B (ja) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4140698A (en) * | 1977-07-25 | 1979-02-20 | Syntex (Usa) Inc. | 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles |
JPS55124633A (en) * | 1979-03-19 | 1980-09-25 | Sohachi Takeuchi | Manufacturing method of tubular vessel |
US4344943A (en) * | 1980-06-09 | 1982-08-17 | Syntex (U.S.A.) Inc. | 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof |
US4353829A (en) * | 1980-11-21 | 1982-10-12 | Syntex (U.S.A.) Inc. | Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters |
US4511724A (en) * | 1982-06-10 | 1985-04-16 | Merck & Co., Inc. | 5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents |
JPS5910589A (ja) * | 1982-06-10 | 1984-01-20 | メルク エンド カムパニー インコーポレーテツド | 抗炎症剤および鎮痛剤として新規な5−(ピロ−ル−2−オイル)−1,2−ジヒドロ−3H−ピロロ〔1,2−a〕ピロ−ル誘導体 |
US4874871A (en) * | 1987-03-25 | 1989-10-17 | Syntex (U.S.A.) Inc. | Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds |
JPH0739418B2 (ja) * | 1987-09-10 | 1995-05-01 | 久光製薬株式会社 | 新規な3−アロイル−6,7−ジヒドロ−5H−ピロロ〔1,2−c〕イミダゾール−7−カルボン酸誘導体 |
JP2649168B2 (ja) * | 1988-02-25 | 1997-09-03 | 久光製薬株式会社 | 新規な5,6−ジフェニル−1,2−ジヒドロ−3H−ピロロ[1,2−a]ピロール−1−カルボン酸誘導体 |
IT1250691B (it) * | 1991-07-22 | 1995-04-21 | Giancarlo Santus | Composizioni terapeutiche per somministrazione intranasale comprendenti ketorolac. |
JP2902113B2 (ja) * | 1991-11-11 | 1999-06-07 | 久光製薬株式会社 | ケトロラク含有シップ剤 |
DE4300697C1 (de) * | 1993-01-13 | 1994-05-19 | Roemmers Sa | Keterolac-Derivat mit wesentlich geringerer gastrointestinaler Reizung und Ulzeration |
US5622948A (en) * | 1994-12-01 | 1997-04-22 | Syntex (U.S.A.) Inc. | Pyrrole pyridazine and pyridazinone anti-inflammatory agents |
JP2008210666A (ja) * | 2007-02-27 | 2008-09-11 | Okamura Corp | 商品陳列棚における照明装置 |
-
1977
- 1977-05-17 JP JP5697777A patent/JPS539788A/ja active Granted
- 1977-07-07 GR GR53907A patent/GR61111B/el unknown
- 1977-07-07 AR AR268356A patent/AR224997A1/es active
- 1977-07-07 DK DK307577A patent/DK151886C/da active
- 1977-07-08 IL IL52493A patent/IL52493A/xx unknown
- 1977-07-08 PT PT66780A patent/PT66780B/pt unknown
- 1977-07-08 NL NLAANVRAGE7707651,A patent/NL186318C/xx not_active IP Right Cessation
- 1977-07-08 CH CH850077A patent/CH641458A5/de not_active IP Right Cessation
- 1977-07-08 IE IE1423/77A patent/IE45253B1/en not_active IP Right Cessation
- 1977-07-11 FR FR7721356A patent/FR2358406A1/fr active Granted
- 1977-07-11 GB GB28919/77A patent/GB1554075A/en not_active Expired
- 1977-07-11 NZ NZ184610A patent/NZ184610A/xx unknown
- 1977-07-11 YU YU1721/77A patent/YU40816B/xx unknown
- 1977-07-11 FI FI772153A patent/FI63406C/fi not_active IP Right Cessation
- 1977-07-12 CA CA282,599A patent/CA1102809A/en not_active Expired
- 1977-07-12 CS CS774646A patent/CS204954B2/cs unknown
- 1977-07-13 PL PL1977199603A patent/PL109390B1/pl unknown
- 1977-07-13 DE DE2760330A patent/DE2760330C2/de not_active Expired
- 1977-07-13 DE DE19772731678 patent/DE2731678A1/de active Granted
- 1977-07-13 SU SU772501050A patent/SU695558A3/ru active
- 1977-07-13 ES ES460706A patent/ES460706A1/es not_active Expired
- 1977-07-13 PL PL1977227289A patent/PL124711B1/pl unknown
- 1977-07-13 PL PL1977227291A patent/PL124445B1/pl unknown
- 1977-07-13 PL PL1977227290A patent/PL124444B1/pl unknown
- 1977-07-13 NO NO772494A patent/NO147564C/no unknown
- 1977-07-13 IT IT68630/77A patent/IT1117313B/it active Protection Beyond IP Right Term
- 1977-07-13 SE SE7708141A patent/SE434643B/xx not_active IP Right Cessation
- 1977-07-14 HU HU77SI1582A patent/HU174224B/hu unknown
- 1977-12-20 FR FR7738508A patent/FR2375234A1/fr active Granted
-
1978
- 1978-05-24 ES ES470214A patent/ES470214A1/es not_active Expired
-
1979
- 1979-11-22 IL IL58779A patent/IL58779A0/xx unknown
-
1981
- 1981-04-23 HK HK159/81A patent/HK15981A/xx unknown
- 1981-12-30 MY MY357/81A patent/MY8100357A/xx unknown
-
1984
- 1984-02-22 CH CH86684A patent/CH646973A5/de not_active IP Right Cessation
- 1984-02-22 CH CH86584A patent/CH646972A5/de not_active IP Right Cessation
-
1991
- 1991-07-05 MX MX9100104A patent/MX163202B/es unknown
-
1993
- 1993-03-23 NL NL930021C patent/NL930021I2/nl unknown
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MA | Patent expired | ||
ND | Supplementary protection certificate (spc) granted | ||
SPCG | Supplementary protection certificate granted |
Spc suppl protection certif: L4 Extension date: 20020711 |
|
MA | Patent expired |
Owner name: SYNTEX (U.S.A.) INC. |