YU172177A - Process for obtaining 5-aroyl-1,2-dihydro-3h-pyrrolo (1,2-a) pyrrol-1-carboxylic derivatives - Google Patents

Process for obtaining 5-aroyl-1,2-dihydro-3h-pyrrolo (1,2-a) pyrrol-1-carboxylic derivatives

Info

Publication number
YU172177A
YU172177A YU01721/77A YU172177A YU172177A YU 172177 A YU172177 A YU 172177A YU 01721/77 A YU01721/77 A YU 01721/77A YU 172177 A YU172177 A YU 172177A YU 172177 A YU172177 A YU 172177A
Authority
YU
Yugoslavia
Prior art keywords
aroyl
pyrrol
pyrrolo
dihydro
obtaining
Prior art date
Application number
YU01721/77A
Other versions
YU40816B (en
Inventor
J M Muchowski
A F Kluge
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=YU172177(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US05/771,286 external-priority patent/US4089969A/en
Application filed by Syntex Inc filed Critical Syntex Inc
Priority to SI7711721A priority Critical patent/SI7711721A8/en
Publication of YU172177A publication Critical patent/YU172177A/en
Publication of YU40816B publication Critical patent/YU40816B/en
Priority to HRP-1721/77A priority patent/HRP940490B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
YU1721/77A 1976-07-14 1977-07-11 Process for obtaining 5-aroyl-1,2 dihydro-3h-pyrrolo (1,2-a)pyrrol-1-carboxylic derivatives YU40816B (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
SI7711721A SI7711721A8 (en) 1976-07-14 1977-07-11 Process for obtaining 5-aroyl-1,2 dehydro-3h-pyrrolo (1,2-a)pyrrol-1-carboxylic derivatives
HRP-1721/77A HRP940490B1 (en) 1976-07-14 1994-08-31 5-AROYL-1,2-DIHYDRO-3H-PYRROLO(1,2-a)PYRROLE-1-CARBOXYLIC ACID DERIVATIVES AND PROCESS FOR THE PRODUCTION THEREOF

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70490976A 1976-07-14 1976-07-14
US05/771,286 US4089969A (en) 1976-07-14 1977-02-23 5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (2)

Publication Number Publication Date
YU172177A true YU172177A (en) 1983-09-30
YU40816B YU40816B (en) 1986-06-30

Family

ID=27107410

Family Applications (1)

Application Number Title Priority Date Filing Date
YU1721/77A YU40816B (en) 1976-07-14 1977-07-11 Process for obtaining 5-aroyl-1,2 dihydro-3h-pyrrolo (1,2-a)pyrrol-1-carboxylic derivatives

Country Status (27)

Country Link
JP (1) JPS539788A (en)
AR (1) AR224997A1 (en)
CA (1) CA1102809A (en)
CH (3) CH641458A5 (en)
CS (1) CS204954B2 (en)
DE (2) DE2760330C2 (en)
DK (1) DK151886C (en)
ES (2) ES460706A1 (en)
FI (1) FI63406C (en)
FR (2) FR2358406A1 (en)
GB (1) GB1554075A (en)
GR (1) GR61111B (en)
HK (1) HK15981A (en)
HU (1) HU174224B (en)
IE (1) IE45253B1 (en)
IL (2) IL52493A (en)
IT (1) IT1117313B (en)
MX (1) MX163202B (en)
MY (1) MY8100357A (en)
NL (2) NL186318C (en)
NO (1) NO147564C (en)
NZ (1) NZ184610A (en)
PL (4) PL124445B1 (en)
PT (1) PT66780B (en)
SE (1) SE434643B (en)
SU (1) SU695558A3 (en)
YU (1) YU40816B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4140698A (en) * 1977-07-25 1979-02-20 Syntex (Usa) Inc. 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) * 1979-03-19 1980-09-25 Sohachi Takeuchi Manufacturing method of tubular vessel
US4344943A (en) * 1980-06-09 1982-08-17 Syntex (U.S.A.) Inc. 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) * 1980-11-21 1982-10-12 Syntex (U.S.A.) Inc. Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) * 1982-06-10 1985-04-16 Merck & Co., Inc. 5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
JPS5910589A (en) * 1982-06-10 1984-01-20 メルク　エンド　カムパニー　インコーポレーテツド Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
US4874871A (en) * 1987-03-25 1989-10-17 Syntex (U.S.A.) Inc. Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (en) * 1987-09-10 1995-05-01 久光製薬株式会社 Novel 3-aroyl-6,7-dihydro-5H-pyrrolo [1,2-c] imidazole-7-carboxylic acid derivative
JP2649168B2 (en) * 1988-02-25 1997-09-03 久光製薬株式会社 Novel 5,6-diphenyl-1,2-dihydro-3H-pyrrolo [1,2-a] pyrrole-1-carboxylic acid derivatives
IT1250691B (en) * 1991-07-22 1995-04-21 Giancarlo Santus THERAPEUTIC COMPOSITIONS FOR INTRANASAL ADMINISTRATION INCLUDING KETOROLAC.
AU669492B2 (en) * 1991-11-11 1996-06-13 Hisamitsu Pharmaceutical Co., Inc. Fomentation containing ketorolac
DE4300697C1 (en) * 1993-01-13 1994-05-19 Roemmers Sa New 2-pyrrolidino-ethyl ester of ketorolac - useful as analgesic, antiinflammatory and antipyretic agent with low ulcerogenicity
US5622948A (en) * 1994-12-01 1997-04-22 Syntex (U.S.A.) Inc. Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (en) * 2007-02-27 2008-09-11 Okamura Corp Lighting system in merchandise display shelf

Also Published As

Publication number Publication date
NO772494L (en) 1978-01-17
IE45253B1 (en) 1982-07-14
CS204954B2 (en) 1981-04-30
SU695558A3 (en) 1979-10-30
DK151886B (en) 1988-01-11
AU513384B2 (en) 1980-11-27
AR224997A1 (en) 1982-02-15
HK15981A (en) 1981-05-01
MX163202B (en) 1992-02-20
PT66780A (en) 1977-08-01
YU40816B (en) 1986-06-30
NL930021I2 (en) 1997-03-03
NO147564C (en) 1983-05-18
PL109390B1 (en) 1980-05-31
PL124444B1 (en) 1983-01-31
CH646972A5 (en) 1984-12-28
PT66780B (en) 1978-12-18
FR2375234A1 (en) 1978-07-21
NL7707651A (en) 1978-01-17
DE2760330C2 (en) 1989-06-15
NL930021I1 (en) 1993-05-03
HU174224B (en) 1979-11-28
FI772153A (en) 1978-01-15
ES460706A1 (en) 1978-12-01
IL52493A0 (en) 1977-10-31
AU2697577A (en) 1979-01-18
SE434643B (en) 1984-08-06
GB1554075A (en) 1979-10-17
IT1117313B (en) 1986-02-17
NO147564B (en) 1983-01-24
FI63406C (en) 1983-06-10
CH641458A5 (en) 1984-02-29
FR2375234B1 (en) 1980-11-07
NL186318C (en) 1990-11-01
DE2731678A1 (en) 1978-03-16
IL58779A0 (en) 1980-02-29
PL124711B1 (en) 1983-02-28
NL186318B (en) 1990-06-01
ES470214A1 (en) 1979-09-16
DK307577A (en) 1978-01-15
FR2358406A1 (en) 1978-02-10
DK151886C (en) 1988-06-06
FR2358406B1 (en) 1981-04-17
PL199603A1 (en) 1978-04-24
IL52493A (en) 1982-02-28
CA1102809A (en) 1981-06-09
GR61111B (en) 1978-09-12
MY8100357A (en) 1981-12-31
DE2731678C2 (en) 1989-06-08
PL124445B1 (en) 1983-01-31
FI63406B (en) 1983-02-28
JPS6254109B2 (en) 1987-11-13
CH646973A5 (en) 1984-12-28
JPS539788A (en) 1978-01-28
SE7708141L (en) 1978-01-15
NZ184610A (en) 1979-03-28
IE45253L (en) 1978-01-14

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